BR9712930A - produtos de condensação de knoevenagel, processos para a sua preparação e aplicação - Google Patents

produtos de condensação de knoevenagel, processos para a sua preparação e aplicação

Info

Publication number
BR9712930A
BR9712930A BRPI9712930-5A BR9712930A BR9712930A BR 9712930 A BR9712930 A BR 9712930A BR 9712930 A BR9712930 A BR 9712930A BR 9712930 A BR9712930 A BR 9712930A
Authority
BR
Brazil
Prior art keywords
processes
preparation
application
condensation products
knoevenagel condensation
Prior art date
Application number
BRPI9712930-5A
Other languages
English (en)
Inventor
Andreas Johannes Kesel
Walter Oberthur
Original Assignee
Andreas Johannes Kesel
Walter Oberthur
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Andreas Johannes Kesel, Walter Oberthur filed Critical Andreas Johannes Kesel
Publication of BR9712930A publication Critical patent/BR9712930A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576Six-membered rings
    • C07F9/58Pyridine rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Polyesters Or Polycarbonates (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)

Abstract

"PRODUTOS DE CONDENSAçãO DE KNOEVENAGEL, PROCESSOS PARA A SUA PREPARAçãO E APLICAçãO". A presente invenção refere-se a novos produtos de condensação de Knoevenagel, processos para a sua preparação e sua aplicação, especialmente para finalidades farmacêuticas e analíticas. Além disso, são publicados conjugados dos condensados de Knoevenagel com biomoléculas. Típico para a invenção é o composto da fórmula (3).
BRPI9712930-5A 1996-11-07 1997-11-07 produtos de condensação de knoevenagel, processos para a sua preparação e aplicação BR9712930A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19645974A DE19645974C1 (de) 1996-11-07 1996-11-07 (Z)-5-[[3-Hydroxy-2-methyl-5-[(phosphonooxy)methyl]-4-pyridinyl]methylen]-2-thioxo-4- thiazolidinon, Verfahren zu dessen Herstellung und Verwendung
PCT/EP1997/006184 WO1998020013A1 (de) 1996-11-07 1997-11-07 Neue knoevenagel-kondensationsprodukte, verfahren zu deren herstellung und verwendung

Publications (1)

Publication Number Publication Date
BR9712930A true BR9712930A (pt) 2006-04-18

Family

ID=7810958

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9712930-5A BR9712930A (pt) 1996-11-07 1997-11-07 produtos de condensação de knoevenagel, processos para a sua preparação e aplicação

Country Status (17)

Country Link
EP (1) EP0937089A1 (pt)
JP (1) JP2001503752A (pt)
KR (1) KR20000053141A (pt)
CN (1) CN1236369A (pt)
AU (1) AU728345B2 (pt)
BR (1) BR9712930A (pt)
CA (1) CA2270973A1 (pt)
CZ (1) CZ160999A3 (pt)
DE (1) DE19645974C1 (pt)
HU (1) HUP9904289A3 (pt)
IL (1) IL129826A0 (pt)
NO (1) NO992209L (pt)
NZ (1) NZ335977A (pt)
PL (1) PL333128A1 (pt)
SK (1) SK61799A3 (pt)
TR (1) TR199901733T2 (pt)
WO (1) WO1998020013A1 (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU3826099A (en) 1998-05-04 1999-11-23 Andreas Johannes Kesel Monomeric, oligomeric and polymeric knoevenagel condensation products
WO2000010573A1 (en) * 1998-08-21 2000-03-02 Viropharma Incorporated Compounds, compositions and methods for treating or preventing viral infections and associated diseases
WO2000066599A1 (en) * 1999-04-30 2000-11-09 Oberthuer Walter Antioxidative vitamin b6 analogs
US6940497B2 (en) 2001-10-16 2005-09-06 Hewlett-Packard Development Company, L.P. Portable electronic reading apparatus
US20030071780A1 (en) * 2001-10-16 2003-04-17 Vincent Kent D. High resolution display

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9103776D0 (sv) * 1991-12-19 1991-12-19 Astra Ab New compounds
IT1266570B1 (it) * 1993-07-30 1997-01-09 Zambon Spa Derivati della propanammide n-eteroaril sostituiti utili nel trattamento delle malattie cardiovascolari
FR2722790B1 (fr) * 1994-07-19 1996-10-04 Roussel Uclaf Nouvelles cephalosporines comportant en position 7 un radical benzyloxymino subtitue, leur procede de preparation leur application comme medicaments

Also Published As

Publication number Publication date
AU728345B2 (en) 2001-01-04
DE19645974C1 (de) 1998-08-13
IL129826A0 (en) 2000-02-29
WO1998020013A1 (de) 1998-05-14
CA2270973A1 (en) 1998-05-14
TR199901733T2 (xx) 1999-09-21
PL333128A1 (en) 1999-11-22
KR20000053141A (ko) 2000-08-25
CZ160999A3 (cs) 1999-09-15
EP0937089A1 (de) 1999-08-25
AU5479898A (en) 1998-05-29
CN1236369A (zh) 1999-11-24
NZ335977A (en) 2000-12-22
NO992209D0 (no) 1999-05-06
JP2001503752A (ja) 2001-03-21
HUP9904289A2 (hu) 2001-04-28
HUP9904289A3 (en) 2001-08-28
SK61799A3 (en) 2000-01-18
NO992209L (no) 1999-07-01

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Legal Events

Date Code Title Description
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1861 DE 05/09/2006.