BR9701672A - Processo para a preparação de ácidos ciclo-alcano-indol-e azaindol-e pirimido(1,2a)-indol-carboxílicos enantiomericamente puros e seus derivados ativados - Google Patents

Processo para a preparação de ácidos ciclo-alcano-indol-e azaindol-e pirimido(1,2a)-indol-carboxílicos enantiomericamente puros e seus derivados ativados

Info

Publication number
BR9701672A
BR9701672A BR9701672A BR9701672A BR9701672A BR 9701672 A BR9701672 A BR 9701672A BR 9701672 A BR9701672 A BR 9701672A BR 9701672 A BR9701672 A BR 9701672A BR 9701672 A BR9701672 A BR 9701672A
Authority
BR
Brazil
Prior art keywords
indole
azaindole
pyrimido
cycloalkane
preparation
Prior art date
Application number
BR9701672A
Other languages
English (en)
Inventor
Jan-Bernd Lenfers
Kai Van Laak
Peter Fey
Paul Naab
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of BR9701672A publication Critical patent/BR9701672A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/612Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/612Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
    • C07C69/616Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety polycyclic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/62Halogen-containing esters
    • C07C69/65Halogen-containing esters of unsaturated acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BR9701672A 1996-04-04 1997-04-04 Processo para a preparação de ácidos ciclo-alcano-indol-e azaindol-e pirimido(1,2a)-indol-carboxílicos enantiomericamente puros e seus derivados ativados BR9701672A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19613549A DE19613549A1 (de) 1996-04-04 1996-04-04 Verfahren zur Herstellung von enantiomerenreinen Cycloalkano-indol- und azaindol-carbonsäuren und deren aktivierte Derivate

Publications (1)

Publication Number Publication Date
BR9701672A true BR9701672A (pt) 1998-11-03

Family

ID=7790501

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9701672A BR9701672A (pt) 1996-04-04 1997-04-04 Processo para a preparação de ácidos ciclo-alcano-indol-e azaindol-e pirimido(1,2a)-indol-carboxílicos enantiomericamente puros e seus derivados ativados

Country Status (27)

Country Link
US (1) US5952498A (pt)
EP (1) EP0799829B1 (pt)
JP (2) JP4235268B2 (pt)
KR (1) KR970069988A (pt)
CN (2) CN1067394C (pt)
AR (2) AR006544A1 (pt)
AT (1) ATE246193T1 (pt)
AU (1) AU722592B2 (pt)
BR (1) BR9701672A (pt)
CA (1) CA2201435C (pt)
CZ (1) CZ102197A3 (pt)
DE (2) DE19613549A1 (pt)
DZ (1) DZ2202A1 (pt)
EE (1) EE9700079A (pt)
ES (1) ES2202506T3 (pt)
HR (1) HRP970178A2 (pt)
HU (1) HU218494B (pt)
ID (1) ID16794A (pt)
IL (1) IL120591A (pt)
MA (1) MA24130A1 (pt)
NO (2) NO308301B1 (pt)
NZ (1) NZ314498A (pt)
PL (1) PL319269A1 (pt)
SG (1) SG60050A1 (pt)
SK (1) SK42897A3 (pt)
TN (1) TNSN97060A1 (pt)
ZA (1) ZA972831B (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4435477A1 (de) 1994-10-04 1996-04-11 Bayer Ag Cycloalkano-indol- und -azaindol-derivate
WO2001074817A1 (fr) * 2000-03-30 2001-10-11 Yamanouchi Pharmaceutical Co., Ltd. Derives d'hydrazide
WO2005051382A1 (ja) * 2003-11-28 2005-06-09 Astellas Pharma Inc. 脂質低下作用増強剤
ES2399721T5 (es) * 2004-03-05 2016-05-25 Univ Pennsylvania Métodos para tratar trastornos o enfermedades asociados a la hiperlipidemia e hipercolesterolemia minimizando los efectos adversos
CA2562015A1 (en) * 2004-04-09 2005-10-20 Janssen Pharmaceutica Nv Intermittent dosing regimens of apob secretion/mtp inhibitors for overweith and obese subjects
JP2009511639A (ja) * 2005-10-18 2009-03-19 エージェリオン ファーマシューティカルズ 血清コレステロールおよび/または血清トリグリセリドを低下させるための組成物
CA2652751A1 (en) * 2006-05-18 2007-11-29 Bayer Healthcare Ag Pharmaceutical compositions and methods of using same
JP2010513534A (ja) * 2006-12-21 2010-04-30 エージェリオン ファーマシューティカルズ, インコーポレイテッド Mtpインヒビターおよびコレステロール吸収インヒビターを含む組み合わせを用いて肥満症を処置する方法
WO2008124384A2 (en) * 2007-04-03 2008-10-16 Aegerion Pharmaceuticals, Inc. Combinations of mtp inhibitors with cholesterol absorption inhibitors or interferon for treating hepatitis c
ES2971913T3 (es) 2013-03-14 2024-06-10 Osteoqc Inc Derivados de un alquil-amina harmina para la promoción del crecimiento de los huesos
KR20210075071A (ko) 2018-08-14 2021-06-22 오스테오큐씨 인코포레이티드 피롤로-디피리딘 화합물
EP3837241A4 (en) 2018-08-14 2022-05-18 Osteoqc Inc. FLUORINATED ß-CARBOLINE COMPOUNDS

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3900261A1 (de) * 1988-05-31 1989-12-07 Bayer Ag Substituierte 4-(chinolin-2-yl-methoxy) phenyl-essigsaeure-derivate
DE4200954A1 (de) * 1991-04-26 1992-10-29 Bayer Ag Heterocyclisch substituierte phenylessigsaeurederivate
DE4208051A1 (de) * 1992-03-13 1993-09-16 Bayer Ag Substituierte phenylessigsaeureamide
DE4302956A1 (de) * 1993-02-03 1994-08-04 Bayer Ag Substituierte Imidazo(4,5-b)pyridine und Benzimidazole
DE4435477A1 (de) * 1994-10-04 1996-04-11 Bayer Ag Cycloalkano-indol- und -azaindol-derivate

Also Published As

Publication number Publication date
ATE246193T1 (de) 2003-08-15
HUP9700698A1 (hu) 1998-01-28
SK42897A3 (en) 1997-10-08
HU218494B (hu) 2000-09-28
JP4235268B2 (ja) 2009-03-11
CN1067394C (zh) 2001-06-20
JP2008169218A (ja) 2008-07-24
MX9702446A (es) 1997-10-31
NO20003784L (no) 1997-10-06
PL319269A1 (en) 1997-10-13
TNSN97060A1 (fr) 2005-03-15
EE9700079A (et) 1997-10-15
CA2201435A1 (en) 1997-10-04
JPH1045759A (ja) 1998-02-17
NZ314498A (en) 1999-09-29
CN1184109A (zh) 1998-06-10
DZ2202A1 (fr) 2002-12-03
IL120591A0 (en) 1997-08-14
CN1330065A (zh) 2002-01-09
ID16794A (id) 1997-11-13
AR012048A2 (es) 2000-09-27
AR006544A1 (es) 1999-09-08
US5952498A (en) 1999-09-14
EP0799829A1 (de) 1997-10-08
NO308301B1 (no) 2000-08-28
AU722592B2 (en) 2000-08-10
CZ102197A3 (en) 1997-10-15
DE19613549A1 (de) 1997-10-09
DE59710487D1 (de) 2003-09-04
NO971513D0 (no) 1997-04-03
CA2201435C (en) 2006-12-12
IL120591A (en) 2000-11-21
KR970069988A (ko) 1997-11-07
ZA972831B (en) 1997-10-31
AU1660297A (en) 1997-10-09
ES2202506T3 (es) 2004-04-01
NO971513L (no) 1997-10-06
MA24130A1 (fr) 1997-10-01
SG60050A1 (en) 1999-02-22
EP0799829B1 (de) 2003-07-30
HU9700698D0 (en) 1997-05-28
NO20003784D0 (no) 2000-07-24
HRP970178A2 (en) 1998-04-30

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Legal Events

Date Code Title Description
FB34 Technical and formal requirements: requirement - article 34 of industrial property law
B11T Dismissal of application maintained [chapter 11.20 patent gazette]