IL120591A - Process for preparation of enantiomerically pure carbazole-,cycloalkanoindole-,cycloalkanoazaindole-,carboline-and pyrimido[1,2-a]indolemethyl-alpha-substituted-benzeneacetic acids and their derivatives and some novel intermediates therefor - Google Patents

Process for preparation of enantiomerically pure carbazole-,cycloalkanoindole-,cycloalkanoazaindole-,carboline-and pyrimido[1,2-a]indolemethyl-alpha-substituted-benzeneacetic acids and their derivatives and some novel intermediates therefor

Info

Publication number
IL120591A
IL120591A IL12059197A IL12059197A IL120591A IL 120591 A IL120591 A IL 120591A IL 12059197 A IL12059197 A IL 12059197A IL 12059197 A IL12059197 A IL 12059197A IL 120591 A IL120591 A IL 120591A
Authority
IL
Israel
Prior art keywords
cycloalkanoazaindole
cycloalkanoindole
indolemethyl
pyrimido
carboline
Prior art date
Application number
IL12059197A
Other languages
English (en)
Other versions
IL120591A0 (en
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Priority to IL13692297A priority Critical patent/IL136922A0/xx
Publication of IL120591A0 publication Critical patent/IL120591A0/xx
Publication of IL120591A publication Critical patent/IL120591A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/612Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/612Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
    • C07C69/616Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety polycyclic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/62Halogen-containing esters
    • C07C69/65Halogen-containing esters of unsaturated acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL12059197A 1996-04-04 1997-04-02 Process for preparation of enantiomerically pure carbazole-,cycloalkanoindole-,cycloalkanoazaindole-,carboline-and pyrimido[1,2-a]indolemethyl-alpha-substituted-benzeneacetic acids and their derivatives and some novel intermediates therefor IL120591A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IL13692297A IL136922A0 (en) 1996-04-04 1997-04-02 Process for the preparation of enantiomerically pure indolecarboxylic acid derivatives and some such new compounds

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19613549A DE19613549A1 (de) 1996-04-04 1996-04-04 Verfahren zur Herstellung von enantiomerenreinen Cycloalkano-indol- und azaindol-carbonsäuren und deren aktivierte Derivate

Publications (2)

Publication Number Publication Date
IL120591A0 IL120591A0 (en) 1997-08-14
IL120591A true IL120591A (en) 2000-11-21

Family

ID=7790501

Family Applications (1)

Application Number Title Priority Date Filing Date
IL12059197A IL120591A (en) 1996-04-04 1997-04-02 Process for preparation of enantiomerically pure carbazole-,cycloalkanoindole-,cycloalkanoazaindole-,carboline-and pyrimido[1,2-a]indolemethyl-alpha-substituted-benzeneacetic acids and their derivatives and some novel intermediates therefor

Country Status (27)

Country Link
US (1) US5952498A (xx)
EP (1) EP0799829B1 (xx)
JP (2) JP4235268B2 (xx)
KR (1) KR970069988A (xx)
CN (2) CN1067394C (xx)
AR (2) AR006544A1 (xx)
AT (1) ATE246193T1 (xx)
AU (1) AU722592B2 (xx)
BR (1) BR9701672A (xx)
CA (1) CA2201435C (xx)
CZ (1) CZ102197A3 (xx)
DE (2) DE19613549A1 (xx)
DZ (1) DZ2202A1 (xx)
EE (1) EE9700079A (xx)
ES (1) ES2202506T3 (xx)
HR (1) HRP970178A2 (xx)
HU (1) HU218494B (xx)
ID (1) ID16794A (xx)
IL (1) IL120591A (xx)
MA (1) MA24130A1 (xx)
NO (2) NO308301B1 (xx)
NZ (1) NZ314498A (xx)
PL (1) PL319269A1 (xx)
SG (1) SG60050A1 (xx)
SK (1) SK42897A3 (xx)
TN (1) TNSN97060A1 (xx)
ZA (1) ZA972831B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4435477A1 (de) 1994-10-04 1996-04-11 Bayer Ag Cycloalkano-indol- und -azaindol-derivate
AU2001244635A1 (en) * 2000-03-30 2001-10-15 Yamanouchi Pharmaceutical Co..Ltd. Hydrazide derivatives
WO2005051382A1 (ja) * 2003-11-28 2005-06-09 Astellas Pharma Inc. 脂質低下作用増強剤
WO2005087234A1 (en) * 2004-03-05 2005-09-22 The Trustees Of The University Of Pennsylvania Methods for treating disorders or diseases associated with hyperlipidemia and hypercholesterolemia while minimizing side-effects
AU2005230397B2 (en) * 2004-04-09 2010-04-08 Elanco Animal Health Ireland Limited Intermittent dosing regimen for the treatment of overweight with MTP-inhibitors
EP1951220A2 (en) * 2005-10-18 2008-08-06 Aegerion Pharmaceuticals Compositions for lowering serum cholesterol and/or triglycerides
US20080051427A1 (en) * 2006-05-18 2008-02-28 Fritz Schuckler Pharmaceutical Compositions and Methods of Using Same
WO2008079398A1 (en) * 2006-12-21 2008-07-03 Aegerion Pharmaceuticals, Inc. Methods for treating obesity with a combination comprising a mtp inhibitor and a cholesterol absorption inhibitor
WO2008124384A2 (en) * 2007-04-03 2008-10-16 Aegerion Pharmaceuticals, Inc. Combinations of mtp inhibitors with cholesterol absorption inhibitors or interferon for treating hepatitis c
JP6721499B2 (ja) 2013-03-14 2020-07-15 オステオーク インコーポレイティド 骨の成長を促進するためのアルキルアミンハルミン誘導体
MX2021001752A (es) 2018-08-14 2021-06-23 Osteoqc Inc Compuestos de pirrolo-dipiridina.
AU2019320773A1 (en) 2018-08-14 2021-03-04 Osteoqc Inc. Fluoro β-carboline compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3900261A1 (de) * 1988-05-31 1989-12-07 Bayer Ag Substituierte 4-(chinolin-2-yl-methoxy) phenyl-essigsaeure-derivate
DE4200954A1 (de) * 1991-04-26 1992-10-29 Bayer Ag Heterocyclisch substituierte phenylessigsaeurederivate
DE4208051A1 (de) * 1992-03-13 1993-09-16 Bayer Ag Substituierte phenylessigsaeureamide
DE4302956A1 (de) * 1993-02-03 1994-08-04 Bayer Ag Substituierte Imidazo(4,5-b)pyridine und Benzimidazole
DE4435477A1 (de) * 1994-10-04 1996-04-11 Bayer Ag Cycloalkano-indol- und -azaindol-derivate

Also Published As

Publication number Publication date
SK42897A3 (en) 1997-10-08
JP4235268B2 (ja) 2009-03-11
CN1184109A (zh) 1998-06-10
BR9701672A (pt) 1998-11-03
NO971513L (no) 1997-10-06
EP0799829B1 (de) 2003-07-30
ZA972831B (en) 1997-10-31
HUP9700698A1 (hu) 1998-01-28
KR970069988A (ko) 1997-11-07
NZ314498A (en) 1999-09-29
DE19613549A1 (de) 1997-10-09
CN1330065A (zh) 2002-01-09
EE9700079A (et) 1997-10-15
NO20003784L (no) 1997-10-06
NO308301B1 (no) 2000-08-28
NO20003784D0 (no) 2000-07-24
HU9700698D0 (en) 1997-05-28
MX9702446A (es) 1997-10-31
MA24130A1 (fr) 1997-10-01
JPH1045759A (ja) 1998-02-17
AU1660297A (en) 1997-10-09
NO971513D0 (no) 1997-04-03
DZ2202A1 (fr) 2002-12-03
CZ102197A3 (en) 1997-10-15
HRP970178A2 (en) 1998-04-30
HU218494B (hu) 2000-09-28
EP0799829A1 (de) 1997-10-08
ID16794A (id) 1997-11-13
CA2201435C (en) 2006-12-12
DE59710487D1 (de) 2003-09-04
AR012048A2 (es) 2000-09-27
PL319269A1 (en) 1997-10-13
US5952498A (en) 1999-09-14
AU722592B2 (en) 2000-08-10
SG60050A1 (en) 1999-02-22
JP2008169218A (ja) 2008-07-24
IL120591A0 (en) 1997-08-14
TNSN97060A1 (fr) 2005-03-15
ES2202506T3 (es) 2004-04-01
ATE246193T1 (de) 2003-08-15
CN1067394C (zh) 2001-06-20
AR006544A1 (es) 1999-09-08
CA2201435A1 (en) 1997-10-04

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Legal Events

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KB Patent renewed
RH1 Patent not in force