BR112021021838A8 - Método para tratar dor associada à endometriose com uso de composto de diaminopirimidina - Google Patents

Método para tratar dor associada à endometriose com uso de composto de diaminopirimidina

Info

Publication number
BR112021021838A8
BR112021021838A8 BR112021021838A BR112021021838A BR112021021838A8 BR 112021021838 A8 BR112021021838 A8 BR 112021021838A8 BR 112021021838 A BR112021021838 A BR 112021021838A BR 112021021838 A BR112021021838 A BR 112021021838A BR 112021021838 A8 BR112021021838 A8 BR 112021021838A8
Authority
BR
Brazil
Prior art keywords
endometriosis
pain associated
treatment
compound
diaminopyrimidine
Prior art date
Application number
BR112021021838A
Other languages
English (en)
Portuguese (pt)
Other versions
BR112021021838A2 (pt
Inventor
Zhao Yanping
Huang Huai
Wang Hongjun
Jiang Yuanyuan
Liang Huining
An Ran
Lan Zhou
Wang Jin
Zhou Liying
Liu Yanan
Original Assignee
Beijing Tide Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beijing Tide Pharmaceutical Co Ltd filed Critical Beijing Tide Pharmaceutical Co Ltd
Publication of BR112021021838A2 publication Critical patent/BR112021021838A2/pt
Publication of BR112021021838A8 publication Critical patent/BR112021021838A8/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BR112021021838A 2019-04-30 2020-04-29 Método para tratar dor associada à endometriose com uso de composto de diaminopirimidina BR112021021838A8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN2019085209 2019-04-30
PCT/CN2020/087689 WO2020221277A1 (zh) 2019-04-30 2020-04-29 二氨基嘧啶类化合物治疗子宫内膜异位相关的疼痛的方法

Publications (2)

Publication Number Publication Date
BR112021021838A2 BR112021021838A2 (pt) 2022-01-04
BR112021021838A8 true BR112021021838A8 (pt) 2023-02-28

Family

ID=73028778

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112021021838A BR112021021838A8 (pt) 2019-04-30 2020-04-29 Método para tratar dor associada à endometriose com uso de composto de diaminopirimidina

Country Status (12)

Country Link
US (1) US12605381B2 (https=)
EP (1) EP3960178B1 (https=)
JP (1) JP7663508B2 (https=)
KR (1) KR102935431B1 (https=)
CN (1) CN114007620B (https=)
AU (1) AU2020266947B2 (https=)
BR (1) BR112021021838A8 (https=)
CA (1) CA3138238A1 (https=)
MX (1) MX2021013347A (https=)
SG (1) SG11202111960PA (https=)
TW (1) TWI737285B (https=)
WO (1) WO2020221277A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN117186068A (zh) * 2017-11-01 2023-12-08 北京泰德制药股份有限公司 P2x3和/或p2x2/3受体拮抗剂、包含其的药物组合物及其用途
WO2023081800A1 (en) * 2021-11-05 2023-05-11 The Regents Of The University Of California Alpha-2a adrenergic receptor modulators and uses thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008104474A1 (en) * 2007-02-28 2008-09-04 F. Hoffmann-La Roche Ag Diaminopyrimidines
WO2017160569A1 (en) 2016-03-14 2017-09-21 Afferent Pharmaceuticals Inc. Pyrimidines and variants thereof, and uses therefor
AU2017237929B2 (en) * 2016-03-25 2021-04-15 Afferent Pharmaceuticals Inc. Pyrimidines and variants thereof, and uses therefor
CN117186068A (zh) * 2017-11-01 2023-12-08 北京泰德制药股份有限公司 P2x3和/或p2x2/3受体拮抗剂、包含其的药物组合物及其用途

Also Published As

Publication number Publication date
WO2020221277A1 (zh) 2020-11-05
KR102935431B1 (ko) 2026-03-05
JP7663508B2 (ja) 2025-04-16
MX2021013347A (es) 2022-01-24
CN114007620A (zh) 2022-02-01
CA3138238A1 (en) 2020-11-05
AU2020266947B2 (en) 2025-10-09
SG11202111960PA (en) 2021-12-30
BR112021021838A2 (pt) 2022-01-04
US12605381B2 (en) 2026-04-21
JP2022531570A (ja) 2022-07-07
AU2020266947A1 (en) 2021-12-16
KR20220008286A (ko) 2022-01-20
EP3960178A1 (en) 2022-03-02
US20220249478A1 (en) 2022-08-11
TW202106303A (zh) 2021-02-16
TWI737285B (zh) 2021-08-21
CN114007620B (zh) 2024-08-06
EP3960178B1 (en) 2026-03-18
EP3960178A4 (en) 2023-01-25

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