BR112021017198A2 - Uso de vibegron para tratar bexiga hiperativa - Google Patents

Uso de vibegron para tratar bexiga hiperativa

Info

Publication number
BR112021017198A2
BR112021017198A2 BR112021017198A BR112021017198A BR112021017198A2 BR 112021017198 A2 BR112021017198 A2 BR 112021017198A2 BR 112021017198 A BR112021017198 A BR 112021017198A BR 112021017198 A BR112021017198 A BR 112021017198A BR 112021017198 A2 BR112021017198 A2 BR 112021017198A2
Authority
BR
Brazil
Prior art keywords
vibegron
overactive bladder
treat overactive
treat
directed
Prior art date
Application number
BR112021017198A
Other languages
English (en)
Portuguese (pt)
Inventor
N Mudd Paul Jr
Original Assignee
Urovant Sciences Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Urovant Sciences Gmbh filed Critical Urovant Sciences Gmbh
Publication of BR112021017198A2 publication Critical patent/BR112021017198A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BR112021017198A 2019-03-18 2020-03-18 Uso de vibegron para tratar bexiga hiperativa BR112021017198A2 (pt)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201962820230P 2019-03-18 2019-03-18
US201962830302P 2019-04-05 2019-04-05
US201962842435P 2019-05-02 2019-05-02
US201962885767P 2019-08-12 2019-08-12
US201962897019P 2019-09-06 2019-09-06
US201962904429P 2019-09-23 2019-09-23
PCT/IB2020/052484 WO2020188505A1 (en) 2019-03-18 2020-03-18 Use of vibegron to treat overactive bladder

Publications (1)

Publication Number Publication Date
BR112021017198A2 true BR112021017198A2 (pt) 2021-11-16

Family

ID=70166082

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112021017198A BR112021017198A2 (pt) 2019-03-18 2020-03-18 Uso de vibegron para tratar bexiga hiperativa

Country Status (14)

Country Link
US (1) US20230027066A1 (https=)
EP (1) EP3941473A1 (https=)
JP (2) JP2022524576A (https=)
KR (2) KR20210142004A (https=)
CN (2) CN121489955A (https=)
AU (2) AU2020243514A1 (https=)
BR (1) BR112021017198A2 (https=)
CA (1) CA3129024A1 (https=)
IL (1) IL285910A (https=)
MX (1) MX2021009488A (https=)
PH (1) PH12021551975A1 (https=)
SG (1) SG11202108810YA (https=)
TW (2) TW202102221A (https=)
WO (1) WO2020188505A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3634420A1 (en) 2017-06-06 2020-04-15 Urovant Sciences GmbH Use of vibegron to treat overactive bladder
SG11202103662VA (en) 2018-12-05 2021-06-29 Urovant Sciences Gmbh Vibegron for the treatment of overactive bladder symptoms
TW202245781A (zh) * 2021-02-16 2022-12-01 瑞士商優洛凡特科學公司 用維貝格龍(vibegron)治療心臟衰竭之方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20091825A1 (es) 2008-04-04 2009-12-04 Merck & Co Inc Hidroximetil pirrolidinas como agonistas del receptor adrenergico beta 3
ES2584427T3 (es) 2011-10-27 2016-09-27 Merck Sharp & Dohme Corp. Proceso para la preparación de agonistas beta 3 y productos intermedios
WO2013062881A1 (en) 2011-10-27 2013-05-02 Merck Sharp & Dohme Corp. Process for making beta 3 agonists and intermediates
RS59402B1 (sr) 2013-03-15 2019-11-29 Merck Sharp & Dohme Postupak za pripremu beta 3 agonista i međuproizvoda
JP6197971B1 (ja) * 2016-04-22 2017-09-20 小野薬品工業株式会社 Kcnq2〜5チャネル関連疾患の予防および/または治療剤
US20170348288A1 (en) * 2016-06-03 2017-12-07 Velicept Therapeutics, Inc. Dosing regimens for beta-3 adrenoceptor agonists and anti-muscarinic agents for the treatment and prevention of lower urinary tract symptoms and overactive bladder
US10057209B2 (en) * 2016-07-28 2018-08-21 Qualcomm Incorporated Time-sequenced multi-device address assignment
JP7670461B2 (ja) * 2017-06-06 2025-04-30 ウロバント サイエンシズ ゲゼルシャフト ミット ベシュレンクター ハフトゥング 過活動膀胱の治療のためのビベグロンの投薬
EP3634420A1 (en) * 2017-06-06 2020-04-15 Urovant Sciences GmbH Use of vibegron to treat overactive bladder
EP3583905A1 (en) * 2018-06-20 2019-12-25 Arthrex Inc Percutaneous targeting device

Also Published As

Publication number Publication date
CN113840607A (zh) 2021-12-24
SG11202108810YA (en) 2021-10-28
AU2020243514A1 (en) 2021-08-26
AU2025256180A1 (en) 2025-11-13
MX2021009488A (es) 2021-09-21
TW202506129A (zh) 2025-02-16
WO2020188505A1 (en) 2020-09-24
CN121489955A (zh) 2026-02-10
JP2022524576A (ja) 2022-05-09
EP3941473A1 (en) 2022-01-26
JP2025084777A (ja) 2025-06-03
CA3129024A1 (en) 2020-09-24
TW202102221A (zh) 2021-01-16
PH12021551975A1 (en) 2022-07-04
IL285910A (en) 2021-10-31
KR20210142004A (ko) 2021-11-23
KR20260049872A (ko) 2026-04-14
US20230027066A1 (en) 2023-01-26

Similar Documents

Publication Publication Date Title
CO2020013600A2 (es) Tratamiento de la hidradenitis supurativa mediante el uso de inhibidores de jak
CO2017011038A2 (es) Derivados de (s)-2-((2-oxooxazolidin-3-il)-5,6-dihidrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-il)amino)amidas como inhibidores de pi3kca”
MX2021002322A (es) Nuevos metodos.
CL2019000935A1 (es) Composición farmacéutica, métodos para tratamiento y usos de la misma.
MX2020009602A (es) Formulaciones de pulverizacion de epinefrina.
BR112016014481A2 (pt) tratamento de câncer utilizando combinações de inibidores de erk e raf
BRPI0510094A (pt) uso de flibanserina no tratamento pré-menstrual e outros distúrbios sexuais femininos
PH12017500746A1 (en) Carbidopa and l-dopa prodrugs and their use to treat parkinson's disease
AR044007A1 (es) Metodos para el tratamiento de la enfermedad de parkinson
BR112021017198A2 (pt) Uso de vibegron para tratar bexiga hiperativa
MX2020009773A (es) Terapia de combinacion.
MX2016015434A (es) Combinaciones farmaceuticas para tratar cancer.
BR112015026247A2 (pt) métodos para o tratamento de câncer com o uso de terapia combinada com inibidor de cinase tor
MX2024002360A (es) Uso de estimuladores de la guanilato ciclasa soluble (sgc) para el tratamiento de trastornos mitocondriales.
MX2018012165A (es) Metodos de tratamiento de canceres pediatricos.
BR112019002945A2 (pt) terapia de combinação para o tratamento de câncer pancreático
ZA202002626B (en) Use of riluzole prodrugs to treat ataxias
ZA202000028B (en) Use of vibegron to treat overactive bladder
AU2018282105A1 (en) Dosing of vibegron for treatment of overactive bladder
MX389282B (es) Composiciones y métodos para tratar sinucleinopatías.
MX2022012632A (es) Uso de inhibidores del bromodominio para el tratamiento de la enfermedad de huntington.
MX2019000849A (es) Gel intestinal de levodopa y carbidopa y metodos de uso.
BR112021010856A2 (pt) Vibegron para o tratamento de sintomas de bexiga hiperativa
MX2018015208A (es) Andrografolido para tratar formas progresivas de esclerosis multiple.
CL2023002236A1 (es) Métodos para tratar la amiloidosis primaria

Legal Events

Date Code Title Description
B06W Patent application suspended after preliminary examination (for patents with searches from other patent authorities) chapter 6.23 patent gazette]