BR112019006963A2 - método para preparar acetofenonas substituídas por ciclopropil - Google Patents

método para preparar acetofenonas substituídas por ciclopropil

Info

Publication number
BR112019006963A2
BR112019006963A2 BR112019006963A BR112019006963A BR112019006963A2 BR 112019006963 A2 BR112019006963 A2 BR 112019006963A2 BR 112019006963 A BR112019006963 A BR 112019006963A BR 112019006963 A BR112019006963 A BR 112019006963A BR 112019006963 A2 BR112019006963 A2 BR 112019006963A2
Authority
BR
Brazil
Prior art keywords
cyclopropyl substituted
substituted acetophenones
preparing cyclopropyl
preparing
acetophenones
Prior art date
Application number
BR112019006963A
Other languages
English (en)
Other versions
BR112019006963B1 (pt
Inventor
Schotes Christoph
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BR112019006963A2 publication Critical patent/BR112019006963A2/pt
Publication of BR112019006963B1 publication Critical patent/BR112019006963B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/20—Unsaturated compounds containing keto groups bound to acyclic carbon atoms
    • C07C49/225—Unsaturated compounds containing keto groups bound to acyclic carbon atoms containing six-membered aromatic rings and other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C29/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
    • C07C29/36—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring increasing the number of carbon atoms by reactions with formation of hydroxy groups, which may occur via intermediates being derivatives of hydroxy, e.g. O-metal
    • C07C29/38—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring increasing the number of carbon atoms by reactions with formation of hydroxy groups, which may occur via intermediates being derivatives of hydroxy, e.g. O-metal by reaction with aldehydes or ketones
    • C07C29/40—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring increasing the number of carbon atoms by reactions with formation of hydroxy groups, which may occur via intermediates being derivatives of hydroxy, e.g. O-metal by reaction with aldehydes or ketones with compounds containing carbon-to-metal bonds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C29/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
    • C07C29/62—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00—Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40—Halogenated unsaturated alcohols
    • C07C33/50—Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/56—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds
    • C07C45/57—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom
    • C07C45/58—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom in three-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
    • C07C49/813—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen polycyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/08—Compounds containing oxirane rings with hydrocarbon radicals, substituted by halogen atoms, nitro radicals or nitroso radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/02—Systems containing only non-condensed rings with a three-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

método para preparar acetofenonas substituídas por ciclopropil. é descrito um método para preparação de acetofenonas substituídas por ciclopropil da fórmula geral (i).
BR112019006963-1A 2016-10-05 2017-09-29 Método para preparar acetofenonas substituídas por ciclopropil, e seus intermediários BR112019006963B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP16192300.8 2016-10-05
EP16192300 2016-10-05
PCT/EP2017/074802 WO2018065316A1 (de) 2016-10-05 2017-09-29 Verfahren zur herstellung von cyclopropyl-substituierten acetophenonen

Publications (2)

Publication Number Publication Date
BR112019006963A2 true BR112019006963A2 (pt) 2019-07-02
BR112019006963B1 BR112019006963B1 (pt) 2023-02-14

Family

ID=57103867

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112019006963-1A BR112019006963B1 (pt) 2016-10-05 2017-09-29 Método para preparar acetofenonas substituídas por ciclopropil, e seus intermediários

Country Status (12)

Country Link
US (1) US10633321B2 (pt)
EP (1) EP3523270B1 (pt)
JP (1) JP6944519B2 (pt)
KR (1) KR102440434B1 (pt)
CN (1) CN109715595B (pt)
BR (1) BR112019006963B1 (pt)
DK (1) DK3523270T3 (pt)
ES (1) ES2849961T3 (pt)
IL (1) IL265779B (pt)
MX (1) MX2019004024A (pt)
TW (1) TWI751203B (pt)
WO (1) WO2018065316A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113121321B (zh) * 2019-12-30 2023-11-24 江苏剑牌农化股份有限公司 一种a-R烷氧基对氯苄基磷酸单酯的回收及其再利用方法
CN113121322A (zh) * 2019-12-30 2021-07-16 辽宁众辉生物科技有限公司 1-(4-氯苯基)-2-环丙基-1-丙酮的合成方法
CN116396151B (zh) * 2022-12-06 2023-11-03 如东众意化工有限公司 一种1-(4-氯苯基)-2-环丙基-1-丙酮的合成方法
CN117402044A (zh) * 2023-10-17 2024-01-16 辽宁众辉生物科技有限公司 一种1-（4-氯苯基）-2-环丙基-1-丙酮的合成方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101857576B (zh) 2010-06-18 2012-07-25 中国科学院上海有机化学研究所 通过环丙基甲基酮制备环唑醇的方法
CN102603508B (zh) * 2012-04-17 2014-03-12 江苏澄扬作物科技有限公司 1-(4-氯苯基)-2-环丙基-1-丙酮的制备方法及其中间体和中间体的制备方法
CN102942465B (zh) * 2012-11-22 2015-10-28 江苏澄扬作物科技有限公司 1-(4-氯苯基)-2-环丙基-1-丙酮的制备方法及其中间体

Also Published As

Publication number Publication date
CN109715595A (zh) 2019-05-03
JP6944519B2 (ja) 2021-10-06
BR112019006963B1 (pt) 2023-02-14
MX2019004024A (es) 2019-08-05
US20200002259A1 (en) 2020-01-02
ES2849961T3 (es) 2021-08-24
KR102440434B1 (ko) 2022-09-05
TW201833065A (zh) 2018-09-16
US10633321B2 (en) 2020-04-28
IL265779A (en) 2019-06-30
CN109715595B (zh) 2022-03-11
WO2018065316A1 (de) 2018-04-12
TWI751203B (zh) 2022-01-01
EP3523270A1 (de) 2019-08-14
EP3523270B1 (de) 2020-10-21
JP2019531300A (ja) 2019-10-31
DK3523270T3 (da) 2021-01-11
IL265779B (en) 2021-04-29
KR20190055837A (ko) 2019-05-23

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Legal Events

Date Code Title Description
B350 Update of information on the portal [chapter 15.35 patent gazette]
B06W Patent application suspended after preliminary examination (for patents with searches from other patent authorities) chapter 6.23 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

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