BR112019003139A2 - processo para a preparação de 3-amino-1-((2,6-dissubstituído)fenil)pirazóis - Google Patents

processo para a preparação de 3-amino-1-((2,6-dissubstituído)fenil)pirazóis

Info

Publication number
BR112019003139A2
BR112019003139A2 BR112019003139A BR112019003139A BR112019003139A2 BR 112019003139 A2 BR112019003139 A2 BR 112019003139A2 BR 112019003139 A BR112019003139 A BR 112019003139A BR 112019003139 A BR112019003139 A BR 112019003139A BR 112019003139 A2 BR112019003139 A2 BR 112019003139A2
Authority
BR
Brazil
Prior art keywords
disubstituted
phenyl
amino
preparation
pyrazols
Prior art date
Application number
BR112019003139A
Other languages
English (en)
Other versions
BR112019003139B1 (pt
Inventor
Sämann Christoph
W J Kennedy Jason
Von Morgenstern Sascha
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BR112019003139A2 publication Critical patent/BR112019003139A2/pt
Publication of BR112019003139B1 publication Critical patent/BR112019003139B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/63—Carboxylic acid nitriles containing cyano groups and nitrogen atoms further bound to other hetero atoms, other than oxygen atoms of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C255/65—Carboxylic acid nitriles containing cyano groups and nitrogen atoms further bound to other hetero atoms, other than oxygen atoms of nitro or nitroso groups, bound to the same carbon skeleton with the nitrogen atoms further bound to nitrogen atoms
    • C07C255/66—Carboxylic acid nitriles containing cyano groups and nitrogen atoms further bound to other hetero atoms, other than oxygen atoms of nitro or nitroso groups, bound to the same carbon skeleton with the nitrogen atoms further bound to nitrogen atoms having cyano groups and nitrogen atoms being part of hydrazine or hydrazone groups bound to the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C07D231/40—Acylated on said nitrogen atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

a presente invenção revela uma preparação eficiente de 3-amino-1-((2,6-dissubstituído)fenil)pirazóis.
BR112019003139-1A 2016-08-15 2017-08-10 Processo para preparação de 3-amino-1-((2,6-dissubstituído)fenil)pirazóis BR112019003139B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP16184135 2016-08-15
EP16184135.8 2016-08-15
PCT/EP2017/070305 WO2018033467A1 (en) 2016-08-15 2017-08-10 Process for the preparation of 3-amino-1-(2,6-disubstituted-phenyl)pyrazoles

Publications (2)

Publication Number Publication Date
BR112019003139A2 true BR112019003139A2 (pt) 2019-05-21
BR112019003139B1 BR112019003139B1 (pt) 2022-11-01

Family

ID=56684544

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112019003139-1A BR112019003139B1 (pt) 2016-08-15 2017-08-10 Processo para preparação de 3-amino-1-((2,6-dissubstituído)fenil)pirazóis

Country Status (12)

Country Link
US (1) US10738012B2 (pt)
EP (1) EP3497084B1 (pt)
JP (1) JP6994498B2 (pt)
KR (1) KR102467045B1 (pt)
CN (1) CN109563048B (pt)
BR (1) BR112019003139B1 (pt)
DK (1) DK3497084T3 (pt)
ES (1) ES2863853T3 (pt)
IL (1) IL264586B (pt)
MX (1) MX2019001813A (pt)
TW (1) TWI777969B (pt)
WO (1) WO2018033467A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022096295A1 (en) 2020-11-03 2022-05-12 Basf Se Fertilizer compatible agrochemical suspensions

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4419078B2 (ja) 2002-12-02 2010-02-24 アステラス製薬株式会社 ピラゾール誘導体
WO2007054480A1 (en) 2005-11-08 2007-05-18 N.V. Organon 2-(benzimidazol-1-yl)-acetamide biaryl derivatives and their use as inhibitors of the trpv1 receptor
CA2732038A1 (en) 2008-07-31 2010-02-04 Merck Sharp & Dohme Corp. Inhibitors of janus kinases
WO2011132017A1 (en) 2010-04-19 2011-10-27 Glenmark Pharmaceuticals S.A. Pyrido[3,4-d]pyrimidinyl acetamide derivatives as trpa1 modulators
AR087701A1 (es) 2011-08-31 2014-04-09 Japan Tobacco Inc Derivados de pirazol con actividad inhibidora de sglt1
AU2013326600B2 (en) * 2012-10-02 2017-03-30 Bayer Cropscience Ag Heterocyclic compounds as pesticides
WO2015144652A2 (en) 2014-03-27 2015-10-01 Bayer Cropscience Ag Heterocyclic compounds for the control of unwanted microorganisms
JP6464190B2 (ja) 2014-04-01 2019-02-06 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 複素環化合物の線虫防除のための使用
WO2015172196A1 (en) 2014-05-13 2015-11-19 Monash University Heterocyclic compounds and use of same

Also Published As

Publication number Publication date
IL264586B (en) 2021-09-30
EP3497084B1 (en) 2021-01-13
CN109563048A (zh) 2019-04-02
MX2019001813A (es) 2019-05-20
TWI777969B (zh) 2022-09-21
WO2018033467A1 (en) 2018-02-22
CN109563048B (zh) 2022-05-06
JP6994498B2 (ja) 2022-02-04
TW201817719A (zh) 2018-05-16
JP2019527723A (ja) 2019-10-03
KR102467045B1 (ko) 2022-11-11
US20190177280A1 (en) 2019-06-13
IL264586A (en) 2019-02-28
EP3497084A1 (en) 2019-06-19
ES2863853T3 (es) 2021-10-11
KR20190039177A (ko) 2019-04-10
US10738012B2 (en) 2020-08-11
DK3497084T3 (da) 2021-04-06
BR112019003139B1 (pt) 2022-11-01

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Legal Events

Date Code Title Description
B350 Update of information on the portal [chapter 15.35 patent gazette]
B06W Patent application suspended after preliminary examination (for patents with searches from other patent authorities) chapter 6.23 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 10/08/2017, OBSERVADAS AS CONDICOES LEGAIS