BR112016028698A2 - preparação de piperidina-4-carbotioamida - Google Patents

preparação de piperidina-4-carbotioamida

Info

Publication number
BR112016028698A2
BR112016028698A2 BR112016028698A BR112016028698A BR112016028698A2 BR 112016028698 A2 BR112016028698 A2 BR 112016028698A2 BR 112016028698 A BR112016028698 A BR 112016028698A BR 112016028698 A BR112016028698 A BR 112016028698A BR 112016028698 A2 BR112016028698 A2 BR 112016028698A2
Authority
BR
Brazil
Prior art keywords
carbothioamide
piperidine
preparation
present
invention describes
Prior art date
Application number
BR112016028698A
Other languages
English (en)
Other versions
BR112016028698B1 (pt
Inventor
Brünjes Marco
James Ford Mark
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BR112016028698A2 publication Critical patent/BR112016028698A2/pt
Publication of BR112016028698B1 publication Critical patent/BR112016028698B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4465—Non condensed piperidines, e.g. piperocaine only substituted in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Plant Pathology (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

preparação de piperidina-4-carbotioamida. a presente invenção descreve um novo processo de preparação de piperidina-4-carbotioamida.
BR112016028698-7A 2014-06-11 2015-06-08 preparação de piperidina-4-carbotioamida BR112016028698B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14172038 2014-06-11
EP14172038.3 2014-06-11
PCT/EP2015/062650 WO2015189115A1 (en) 2014-06-11 2015-06-08 Preparation of piperidine-4-carbothioamide

Publications (2)

Publication Number Publication Date
BR112016028698A2 true BR112016028698A2 (pt) 2017-08-22
BR112016028698B1 BR112016028698B1 (pt) 2021-05-04

Family

ID=50896206

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112016028698-7A BR112016028698B1 (pt) 2014-06-11 2015-06-08 preparação de piperidina-4-carbotioamida

Country Status (12)

Country Link
US (1) US9790182B2 (pt)
EP (1) EP3154942B1 (pt)
JP (1) JP6603242B2 (pt)
KR (1) KR102430612B1 (pt)
CN (1) CN106458898B (pt)
BR (1) BR112016028698B1 (pt)
DK (1) DK3154942T3 (pt)
ES (1) ES2753582T3 (pt)
IL (1) IL249130B (pt)
MX (1) MX2016016398A (pt)
TW (1) TWI666199B (pt)
WO (1) WO2015189115A1 (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10093626B2 (en) * 2015-03-05 2018-10-09 Bayer Cropscience Aktiengesellschaft Process for preparing piperidine-4-carbothioamide hydrochloride
DE102018212696B3 (de) 2018-07-30 2019-11-07 Thyssenkrupp Ag Verstellantrieb für eine Lenksäule und Lenksäule für ein Kraftfahrzeug

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1143364A (zh) * 1994-03-11 1997-02-19 山之内制药株式会社 5-ht3受体激动剂、新颖的噻唑衍生物及其中间体
DE10252102A1 (de) * 2002-11-08 2004-05-27 Merck Patent Gmbh Indolderivate
KR20060017929A (ko) * 2004-08-04 2006-02-28 동화약품공업주식회사 티아졸 유도체가 치환된 신규한 벤즈아미딘 유도체, 그의제조방법 및 이를 유효성분으로 하는 약학 조성물
CN1807409A (zh) * 2006-02-09 2006-07-26 朱凯琴 硫代酰胺类化合物的合成方法
WO2008013622A2 (en) * 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
WO2009019295A2 (en) 2007-08-06 2009-02-12 Nv Remynd Phenyl- and benzylthiazolylpiperazine derivatives for the treatment of neurodegenerative diseases
US20090054392A1 (en) * 2007-08-20 2009-02-26 Wyeth Naphthylpyrimidine, naphthylpyrazine and naphthylpyridazine analogs and their use as agonists of the wnt-beta-catenin cellular messaging system
TWI428091B (zh) 2007-10-23 2014-03-01 Du Pont 殺真菌劑混合物
WO2009094407A2 (en) 2008-01-25 2009-07-30 E. I. Du Pont De Nemours And Company Fungicidal amides
EP2509978A1 (en) 2009-12-11 2012-10-17 E.I. Du Pont De Nemours And Company Azocyclic inhibitors of fatty acid amide hydrolase
CN102781937B (zh) 2009-12-21 2015-09-30 拜尔农作物科学股份公司 用作杀菌剂的双(二氟甲基)吡唑
WO2011146182A1 (en) 2010-05-20 2011-11-24 E. I. Du Pont De Nemours And Company Fungicidal oximes and hydrazones
EP2585048B1 (en) * 2010-06-23 2018-04-11 CymaBay Therapeutics, Inc. Compositions of 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine
WO2013127808A1 (en) 2012-03-02 2013-09-06 Syngenta Participations Ag Microbiocidal pyrazole derivatives

Also Published As

Publication number Publication date
MX2016016398A (es) 2017-04-06
CN106458898A (zh) 2017-02-22
JP2017517531A (ja) 2017-06-29
JP6603242B2 (ja) 2019-11-06
US9790182B2 (en) 2017-10-17
KR20170016387A (ko) 2017-02-13
WO2015189115A1 (en) 2015-12-17
BR112016028698B1 (pt) 2021-05-04
CN106458898B (zh) 2019-11-12
IL249130B (en) 2018-12-31
TWI666199B (zh) 2019-07-21
ES2753582T3 (es) 2020-04-13
EP3154942B1 (en) 2019-08-28
DK3154942T3 (da) 2019-11-18
EP3154942A1 (en) 2017-04-19
KR102430612B1 (ko) 2022-08-08
TW201625530A (zh) 2016-07-16
US20170137381A1 (en) 2017-05-18
IL249130A0 (en) 2017-01-31

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07G Grant request does not fulfill article 229-c lpi (prior consent of anvisa) [chapter 7.7 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 08/06/2015, OBSERVADAS AS CONDICOES LEGAIS.