BR112017021631A2 - composto, composição farmacêutica, combinação farmacêutica, método de tratamento, uso de um composto e processo para preparação de dito composto - Google Patents

composto, composição farmacêutica, combinação farmacêutica, método de tratamento, uso de um composto e processo para preparação de dito composto

Info

Publication number
BR112017021631A2
BR112017021631A2 BR112017021631-0A BR112017021631A BR112017021631A2 BR 112017021631 A2 BR112017021631 A2 BR 112017021631A2 BR 112017021631 A BR112017021631 A BR 112017021631A BR 112017021631 A2 BR112017021631 A2 BR 112017021631A2
Authority
BR
Brazil
Prior art keywords
compound
pharmaceutical composition
preparing
treatment
compounds
Prior art date
Application number
BR112017021631-0A
Other languages
English (en)
Inventor
Dutt Chaitanya
Chandra Gupta Ramesh
Patel Manish
Abraham Jaya
Mishra Vivek
Kesarwani Amit
Deshpande Shailesh
Kumar Zambad Shital
Mathur Anoop
Kotecha Jignesh
Latad Sachin
Chaudhari Anita
Original Assignee
Torrent Pharmaceuticals Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Torrent Pharmaceuticals Limited filed Critical Torrent Pharmaceuticals Limited
Publication of BR112017021631A2 publication Critical patent/BR112017021631A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4436Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C53/00Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
    • C07C53/126Acids containing more than four carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

a presente invenção refere-se a novos compostos de piridínio, seus isômeros, esterômeros, atropisômeros, conformadores, tautômeros, polimorfos, hidratos e solvatos. o presente invento engloba também um processo para a preparação de novos compostos, e uma composição farmacêutica dos referidos compostos. a invenção refere-se ainda à utilização dos compostos acima mencionados para a preparação de um medicamento para uso como produtos farmacêuticos.
BR112017021631-0A 2015-04-08 2016-04-05 composto, composição farmacêutica, combinação farmacêutica, método de tratamento, uso de um composto e processo para preparação de dito composto BR112017021631A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN1473MU2015 2015-04-08
IN1473/MUM/2015 2015-04-08
PCT/IB2016/051917 WO2016162785A1 (en) 2015-04-08 2016-04-05 Novel pyridinium compounds

Publications (1)

Publication Number Publication Date
BR112017021631A2 true BR112017021631A2 (pt) 2018-07-03

Family

ID=55808799

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112017021631-0A BR112017021631A2 (pt) 2015-04-08 2016-04-05 composto, composição farmacêutica, combinação farmacêutica, método de tratamento, uso de um composto e processo para preparação de dito composto

Country Status (19)

Country Link
US (2) US10233175B2 (pt)
EP (1) EP3280711A1 (pt)
JP (1) JP6782763B2 (pt)
KR (1) KR20170134661A (pt)
CN (1) CN107438604B (pt)
AR (1) AR104274A1 (pt)
AU (1) AU2016245418B2 (pt)
BR (1) BR112017021631A2 (pt)
CA (1) CA2997364A1 (pt)
EA (1) EA035406B1 (pt)
IL (1) IL254792B (pt)
MX (1) MX2017012943A (pt)
MY (1) MY182914A (pt)
PH (1) PH12017501830A1 (pt)
SG (1) SG11201708140RA (pt)
TW (1) TWI710559B (pt)
UA (1) UA120389C2 (pt)
WO (1) WO2016162785A1 (pt)
ZA (1) ZA201707090B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2997364A1 (en) * 2015-04-08 2016-10-13 Torrent Pharmaceuticals Limited Novel pyridinium compounds
LT3762368T (lt) 2018-03-08 2022-06-10 Incyte Corporation Aminopirazindiolio junginiai, kaip pi3k-γ inhibitoriai
WO2020010003A1 (en) 2018-07-02 2020-01-09 Incyte Corporation AMINOPYRAZINE DERIVATIVES AS PI3K-γ INHIBITORS
US20200338058A1 (en) * 2019-04-28 2020-10-29 King Faisal University Therapeutic agents for treating and preventing autoimmune diseases and cancer and a screening method
WO2022238921A1 (en) * 2021-05-14 2022-11-17 Torrent Pharmaceuticals Limited In-situ synthesis of 3-substituted pyridinium compounds

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2215000C2 (ru) * 1999-10-06 2003-10-27 Торрент Фармасьютикалз Лтд. Производные солей пиридиния, способ их получения, фармацевтические композиции на их основе и способы лечения
PL348049A1 (en) * 1999-10-06 2002-05-06 Torrent Pharmaceuticals Ltd Pyridinium derivatives for the treatment of diabetic and aging−related vascular complications
US6608094B2 (en) * 1999-10-06 2003-08-19 Torrent Pharmaceuticals Ltd. Compounds for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof
DK1243581T3 (da) 2001-03-21 2005-10-31 Torrent Pharmaceuticals Ltd Pyridiniumforbindelser til behandling af AGE-relaterede sygdomme
PT1373263E (pt) 2001-04-05 2005-03-31 Torrent Pharmaceuticals Ltd Compostos heterociclicos para complicacoes relacionadas com a idade e complicacoes vasculares diabeticas
EP1996588A4 (en) 2006-03-03 2011-10-05 Torrent Pharmaceuticals Ltd NEW DUAL ACTION RECEPTOR (DARA) ANTAGONISTS OF ATI AND ETA RECEPTORS
CA2997364A1 (en) * 2015-04-08 2016-10-13 Torrent Pharmaceuticals Limited Novel pyridinium compounds

Also Published As

Publication number Publication date
AR104274A1 (es) 2017-07-12
IL254792A0 (en) 2017-12-31
KR20170134661A (ko) 2017-12-06
CA2997364A1 (en) 2016-10-13
TW201639834A (zh) 2016-11-16
CN107438604B (zh) 2021-12-03
US10717727B2 (en) 2020-07-21
EA035406B1 (ru) 2020-06-09
US20190169175A1 (en) 2019-06-06
AU2016245418B2 (en) 2020-03-26
UA120389C2 (uk) 2019-11-25
WO2016162785A1 (en) 2016-10-13
JP2018511658A (ja) 2018-04-26
EP3280711A1 (en) 2018-02-14
MX2017012943A (es) 2018-01-30
MY182914A (en) 2021-02-05
JP6782763B2 (ja) 2020-11-11
US20180118728A1 (en) 2018-05-03
EA201792234A1 (ru) 2018-02-28
AU2016245418A1 (en) 2017-11-02
TWI710559B (zh) 2020-11-21
SG11201708140RA (en) 2017-11-29
PH12017501830A1 (en) 2018-04-23
US10233175B2 (en) 2019-03-19
CN107438604A (zh) 2017-12-05
ZA201707090B (en) 2021-03-31
IL254792B (en) 2021-01-31

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements