BR112017021631A2 - composto, composição farmacêutica, combinação farmacêutica, método de tratamento, uso de um composto e processo para preparação de dito composto - Google Patents
composto, composição farmacêutica, combinação farmacêutica, método de tratamento, uso de um composto e processo para preparação de dito compostoInfo
- Publication number
- BR112017021631A2 BR112017021631A2 BR112017021631-0A BR112017021631A BR112017021631A2 BR 112017021631 A2 BR112017021631 A2 BR 112017021631A2 BR 112017021631 A BR112017021631 A BR 112017021631A BR 112017021631 A2 BR112017021631 A2 BR 112017021631A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- pharmaceutical composition
- preparing
- treatment
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4436—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
- C07C53/126—Acids containing more than four carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
a presente invenção refere-se a novos compostos de piridínio, seus isômeros, esterômeros, atropisômeros, conformadores, tautômeros, polimorfos, hidratos e solvatos. o presente invento engloba também um processo para a preparação de novos compostos, e uma composição farmacêutica dos referidos compostos. a invenção refere-se ainda à utilização dos compostos acima mencionados para a preparação de um medicamento para uso como produtos farmacêuticos.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1473MU2015 | 2015-04-08 | ||
IN1473/MUM/2015 | 2015-04-08 | ||
PCT/IB2016/051917 WO2016162785A1 (en) | 2015-04-08 | 2016-04-05 | Novel pyridinium compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112017021631A2 true BR112017021631A2 (pt) | 2018-07-03 |
Family
ID=55808799
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112017021631-0A BR112017021631A2 (pt) | 2015-04-08 | 2016-04-05 | composto, composição farmacêutica, combinação farmacêutica, método de tratamento, uso de um composto e processo para preparação de dito composto |
Country Status (19)
Country | Link |
---|---|
US (2) | US10233175B2 (pt) |
EP (1) | EP3280711A1 (pt) |
JP (1) | JP6782763B2 (pt) |
KR (1) | KR20170134661A (pt) |
CN (1) | CN107438604B (pt) |
AR (1) | AR104274A1 (pt) |
AU (1) | AU2016245418B2 (pt) |
BR (1) | BR112017021631A2 (pt) |
CA (1) | CA2997364A1 (pt) |
EA (1) | EA035406B1 (pt) |
IL (1) | IL254792B (pt) |
MX (1) | MX2017012943A (pt) |
MY (1) | MY182914A (pt) |
PH (1) | PH12017501830A1 (pt) |
SG (1) | SG11201708140RA (pt) |
TW (1) | TWI710559B (pt) |
UA (1) | UA120389C2 (pt) |
WO (1) | WO2016162785A1 (pt) |
ZA (1) | ZA201707090B (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2997364A1 (en) * | 2015-04-08 | 2016-10-13 | Torrent Pharmaceuticals Limited | Novel pyridinium compounds |
LT3762368T (lt) | 2018-03-08 | 2022-06-10 | Incyte Corporation | Aminopirazindiolio junginiai, kaip pi3k-γ inhibitoriai |
WO2020010003A1 (en) | 2018-07-02 | 2020-01-09 | Incyte Corporation | AMINOPYRAZINE DERIVATIVES AS PI3K-γ INHIBITORS |
US20200338058A1 (en) * | 2019-04-28 | 2020-10-29 | King Faisal University | Therapeutic agents for treating and preventing autoimmune diseases and cancer and a screening method |
WO2022238921A1 (en) * | 2021-05-14 | 2022-11-17 | Torrent Pharmaceuticals Limited | In-situ synthesis of 3-substituted pyridinium compounds |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
RU2215000C2 (ru) * | 1999-10-06 | 2003-10-27 | Торрент Фармасьютикалз Лтд. | Производные солей пиридиния, способ их получения, фармацевтические композиции на их основе и способы лечения |
PL348049A1 (en) * | 1999-10-06 | 2002-05-06 | Torrent Pharmaceuticals Ltd | Pyridinium derivatives for the treatment of diabetic and aging−related vascular complications |
US6608094B2 (en) * | 1999-10-06 | 2003-08-19 | Torrent Pharmaceuticals Ltd. | Compounds for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof |
DK1243581T3 (da) | 2001-03-21 | 2005-10-31 | Torrent Pharmaceuticals Ltd | Pyridiniumforbindelser til behandling af AGE-relaterede sygdomme |
PT1373263E (pt) | 2001-04-05 | 2005-03-31 | Torrent Pharmaceuticals Ltd | Compostos heterociclicos para complicacoes relacionadas com a idade e complicacoes vasculares diabeticas |
EP1996588A4 (en) | 2006-03-03 | 2011-10-05 | Torrent Pharmaceuticals Ltd | NEW DUAL ACTION RECEPTOR (DARA) ANTAGONISTS OF ATI AND ETA RECEPTORS |
CA2997364A1 (en) * | 2015-04-08 | 2016-10-13 | Torrent Pharmaceuticals Limited | Novel pyridinium compounds |
-
2016
- 2016-04-05 CA CA2997364A patent/CA2997364A1/en not_active Abandoned
- 2016-04-05 BR BR112017021631-0A patent/BR112017021631A2/pt not_active Application Discontinuation
- 2016-04-05 JP JP2018503834A patent/JP6782763B2/ja active Active
- 2016-04-05 CN CN201680020723.5A patent/CN107438604B/zh active Active
- 2016-04-05 UA UAA201710766A patent/UA120389C2/uk unknown
- 2016-04-05 KR KR1020177032034A patent/KR20170134661A/ko not_active Application Discontinuation
- 2016-04-05 SG SG11201708140RA patent/SG11201708140RA/en unknown
- 2016-04-05 EP EP16718473.8A patent/EP3280711A1/en not_active Withdrawn
- 2016-04-05 AR ARP160100917A patent/AR104274A1/es unknown
- 2016-04-05 EA EA201792234A patent/EA035406B1/ru not_active IP Right Cessation
- 2016-04-05 AU AU2016245418A patent/AU2016245418B2/en not_active Ceased
- 2016-04-05 MX MX2017012943A patent/MX2017012943A/es unknown
- 2016-04-05 US US15/564,715 patent/US10233175B2/en active Active
- 2016-04-05 MY MYPI2017001476A patent/MY182914A/en unknown
- 2016-04-05 WO PCT/IB2016/051917 patent/WO2016162785A1/en active Application Filing
- 2016-04-06 TW TW105110717A patent/TWI710559B/zh active
-
2017
- 2017-09-28 IL IL254792A patent/IL254792B/en active IP Right Grant
- 2017-10-06 PH PH12017501830A patent/PH12017501830A1/en unknown
- 2017-10-19 ZA ZA2017/07090A patent/ZA201707090B/en unknown
-
2019
- 2019-02-04 US US16/267,224 patent/US10717727B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
AR104274A1 (es) | 2017-07-12 |
IL254792A0 (en) | 2017-12-31 |
KR20170134661A (ko) | 2017-12-06 |
CA2997364A1 (en) | 2016-10-13 |
TW201639834A (zh) | 2016-11-16 |
CN107438604B (zh) | 2021-12-03 |
US10717727B2 (en) | 2020-07-21 |
EA035406B1 (ru) | 2020-06-09 |
US20190169175A1 (en) | 2019-06-06 |
AU2016245418B2 (en) | 2020-03-26 |
UA120389C2 (uk) | 2019-11-25 |
WO2016162785A1 (en) | 2016-10-13 |
JP2018511658A (ja) | 2018-04-26 |
EP3280711A1 (en) | 2018-02-14 |
MX2017012943A (es) | 2018-01-30 |
MY182914A (en) | 2021-02-05 |
JP6782763B2 (ja) | 2020-11-11 |
US20180118728A1 (en) | 2018-05-03 |
EA201792234A1 (ru) | 2018-02-28 |
AU2016245418A1 (en) | 2017-11-02 |
TWI710559B (zh) | 2020-11-21 |
SG11201708140RA (en) | 2017-11-29 |
PH12017501830A1 (en) | 2018-04-23 |
US10233175B2 (en) | 2019-03-19 |
CN107438604A (zh) | 2017-12-05 |
ZA201707090B (en) | 2021-03-31 |
IL254792B (en) | 2021-01-31 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BR112018005497A2 (pt) | compostos heterocíclicos e usos dos mesmos | |
CL2018000542A1 (es) | Nuevos derivados de fenoximetilo. | |
CL2018002009A1 (es) | Compuestos derivados de ciclopentanoperhidofenantreno, moduladores de fxr; composicion farmaceutica que comprende dichos compuestos; y su uso para el tratamiento de enfermedades colestásicas, fibróticas, hipercolesterolemia, entre otras. | |
BR112017022604A2 (pt) | composto, composição farmacêutica, uso de um composto e de uma combinação, e, combinação | |
BR112017010354B8 (pt) | Compostos de triazolopirimidina, seu uso, e composição farmacêutica | |
MX2018004175A (es) | Derivado oxa espiro, su metodo de preparacion, y sus aplicaciones en medicinas. | |
CL2015001733A1 (es) | Compuestos derivados de lactamas fusionadas de arilo y heteroarilo, moduladores de ezh2; composicion farmaceutica que los comprende; uso del compuesto para el tratamiento del cancer. | |
BR112014021531A8 (pt) | composto, composição farmacêutica e usos dos mesmos | |
BR112016023558A2 (pt) | compostos úteis como imunomoduladores | |
PH12017500416A1 (en) | Compounds and compositions as raf kinase inhibitors | |
BR112014012878A8 (pt) | composto, uso de um composto, composição farmacêutica e processos de fabricação de um composto | |
BR112016014020A8 (pt) | moduladores de tetra-hidropiridopirazinas de gpr6. | |
CL2014000311A1 (es) | Compuestos derivados de benzotiazepinas sustituidas; composicion farmaceutica que los contiene; y su uso para el tratamiento o profilaxis de la infeccion del virus sincicial respiratorio. | |
BR112014018990A8 (pt) | Derivados de ácido benzotiazol-6-il acético e seu uso para tratamento de uma infecção | |
CL2014000543A1 (es) | Compuestos derivados de imidazopiridazinas sustituidas con amino, inhibidores de la quinasa ,mknk2; metodo de preparacion; compuestos intermediarios y su uso; composicion farmaceutica; combinacion farmaceutica; y su uso para el tratamiento del cancer. | |
MX2017014035A (es) | Formas solidas novedosas. | |
BR112017021631A2 (pt) | composto, composição farmacêutica, combinação farmacêutica, método de tratamento, uso de um composto e processo para preparação de dito composto | |
MX364376B (es) | Derivado de fenol y metodo de preparacion y uso en la medicina del mismo. | |
BR112018070123A2 (pt) | oxiesterós e métodos de uso dos mesmos | |
BR112017004173A2 (pt) | composto, composição farmacêutica, e, método para tratar uma doença ou condição patológica. | |
BR112017010311A2 (pt) | 4-oxo-3,4-dihidro-1,2,3-benzotriazinas como moduladores de gpr139 | |
EA201790949A1 (ru) | Замещенные 2,4-диаминохинолины в качестве новых противораковых средств | |
BR112017005242A2 (pt) | composto, composição farmacêutica, e, composto para uso. | |
CL2014002845A1 (es) | Compuestos derivados de pirazol inhibidores de sglt1; metodo para tratar la diabetes; composicion farmaceutica; uso del compuesto para el tratamiento de la diabetes tipo 1 y tipo 2. | |
BR112017002852A2 (pt) | compostos de azetidiniloxifenilpirrolidina |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] |
Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS. |
|
B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
B06U | Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette] | ||
B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements |