BR112017009850A2 - composto, composição, e, uso de uma quantidade melhoradora de hiv de um composto - Google Patents
composto, composição, e, uso de uma quantidade melhoradora de hiv de um compostoInfo
- Publication number
- BR112017009850A2 BR112017009850A2 BR112017009850A BR112017009850A BR112017009850A2 BR 112017009850 A2 BR112017009850 A2 BR 112017009850A2 BR 112017009850 A BR112017009850 A BR 112017009850A BR 112017009850 A BR112017009850 A BR 112017009850A BR 112017009850 A2 BR112017009850 A2 BR 112017009850A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- composition
- hiv
- compounds
- enhancer amount
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
- C07J63/008—Expansion of ring D by one atom, e.g. D homo steroids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201462079977P | 2014-11-14 | 2014-11-14 | |
PCT/US2015/060344 WO2016077561A1 (en) | 2014-11-14 | 2015-11-12 | Oxolupene derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112017009850A2 true BR112017009850A2 (pt) | 2018-01-16 |
Family
ID=54697682
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112017009850A BR112017009850A2 (pt) | 2014-11-14 | 2015-11-12 | composto, composição, e, uso de uma quantidade melhoradora de hiv de um composto |
Country Status (10)
Country | Link |
---|---|
US (1) | US9969767B2 (pt) |
EP (1) | EP3218387A1 (pt) |
JP (1) | JP2017533937A (pt) |
KR (1) | KR20170087478A (pt) |
CN (1) | CN107250153A (pt) |
AU (1) | AU2015346303B2 (pt) |
BR (1) | BR112017009850A2 (pt) |
CA (1) | CA2967679A1 (pt) |
RU (1) | RU2017118489A (pt) |
WO (1) | WO2016077561A1 (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2016298669A1 (en) * | 2015-07-28 | 2018-02-22 | Glaxosmithkline Intellectual Property (No.2) Limited | Betuin derivatives for preventing or treating HIV infections |
EP3328875A1 (en) * | 2015-07-28 | 2018-06-06 | Glaxosmithkline Intellectual Property (No. 2) Limited | Betuin derivatives for preventing or treating hiv infections |
US20180273579A1 (en) * | 2015-09-24 | 2018-09-27 | Glaxosmithkline Intellectual Property (No.2) Limited | Compounds with hiv maturation inhibitory activity |
WO2017125870A1 (en) * | 2016-01-20 | 2017-07-27 | Glaxosmithkline Intellectual Property (No.2) Limited | Amine derivatives of lupanes with hiv maturation inhibitory activity |
Family Cites Families (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5413999A (en) | 1991-11-08 | 1995-05-09 | Merck & Co., Inc. | HIV protease inhibitors useful for the treatment of AIDS |
US5679828A (en) | 1995-06-05 | 1997-10-21 | Biotech Research Labs, Inc. | Betulinic acid and dihydrobetulinic acid derivatives and uses therefor |
US20040110785A1 (en) | 2001-02-02 | 2004-06-10 | Tao Wang | Composition and antiviral activity of substituted azaindoleoxoacetic piperazine derivatives |
US7365221B2 (en) | 2002-09-26 | 2008-04-29 | Panacos Pharmaceuticals, Inc. | Monoacylated betulin and dihydrobetulin derivatives, preparation thereof and use thereof |
US7745625B2 (en) | 2004-03-15 | 2010-06-29 | Bristol-Myers Squibb Company | Prodrugs of piperazine and substituted piperidine antiviral agents |
CA2560266A1 (en) | 2004-03-17 | 2005-09-29 | Panacos Pharmaceuticals, Inc. | Pharmaceutical salts of 3-o-(3',3'-dimethylsuccinyl) betulinic acid |
TW200628161A (en) | 2004-11-12 | 2006-08-16 | Panacos Pharmaceuticals Inc | Novel betulin derivatives, preparation thereof and use thereof |
US20090105203A1 (en) | 2006-10-16 | 2009-04-23 | Myriad Genetics, Incorporated | Compounds for treating viral infections |
TW200837074A (en) * | 2006-11-03 | 2008-09-16 | Panacos Pharmaceuticals Inc | Extended triterpene derivatives |
EP2250185A4 (en) * | 2008-01-03 | 2011-11-16 | Virochem Pharma Inc | NEW LUPANDERIVATE |
CA2714049A1 (en) | 2008-02-14 | 2009-08-20 | Virochem Pharma Inc. | Novel 17.beta. lupane derivatives |
US8431556B2 (en) * | 2008-03-26 | 2013-04-30 | Vertex Pharmaceuticals Incorporated | C-21-keto lupane derivatives preparation and use thereof |
US9067966B2 (en) | 2009-07-14 | 2015-06-30 | Hetero Research Foundation, Hetero Drugs Ltd. | Lupeol-type triterpene derivatives as antivirals |
WO2011100308A1 (en) * | 2010-02-11 | 2011-08-18 | Glaxosmithkline Llc | Derivatives of betulin |
PT2576586E (pt) * | 2010-06-04 | 2015-10-23 | Bristol Myers Squibb Co | Amidas c-28 de derivados de ácido betulínico c-3 modificadas como inibidores de maturação de hiv |
BR112012030818A2 (pt) * | 2010-06-04 | 2019-09-24 | Bristol-Myers Squibb Company | "derivados de ácido c-3 betulínico modificado como inibidores da maturação do hiv" |
AU2012212509B2 (en) | 2011-01-31 | 2016-01-21 | ViiV Healthcare UK (No.4) Limited | C-17 and C-3 modified triterpenoids with HIV maturation inhibitory activity |
EA023578B1 (ru) * | 2011-01-31 | 2016-06-30 | Бристол-Маерс Сквибб Компани | C28-амины c3-модифицированных производных бетулиновой кислоты в качестве ингибиторов созревания вич |
JO3387B1 (ar) * | 2011-12-16 | 2019-03-13 | Glaxosmithkline Llc | مشتقات بيتولين |
CN103242413B (zh) * | 2012-02-08 | 2015-08-26 | 江西青峰药业有限公司 | Lupane三萜系衍生物及其药学用途 |
US8906889B2 (en) | 2012-02-15 | 2014-12-09 | Bristol-Myers Squibb Company | C-3 cycloalkenyl triterpenoids with HIV maturation inhibitory activity |
-
2015
- 2015-11-12 JP JP2017525933A patent/JP2017533937A/ja active Pending
- 2015-11-12 US US15/524,298 patent/US9969767B2/en not_active Expired - Fee Related
- 2015-11-12 RU RU2017118489A patent/RU2017118489A/ru not_active Application Discontinuation
- 2015-11-12 BR BR112017009850A patent/BR112017009850A2/pt not_active IP Right Cessation
- 2015-11-12 KR KR1020177016222A patent/KR20170087478A/ko unknown
- 2015-11-12 CA CA2967679A patent/CA2967679A1/en not_active Abandoned
- 2015-11-12 CN CN201580071098.2A patent/CN107250153A/zh active Pending
- 2015-11-12 AU AU2015346303A patent/AU2015346303B2/en not_active Ceased
- 2015-11-12 EP EP15798639.9A patent/EP3218387A1/en not_active Ceased
- 2015-11-12 WO PCT/US2015/060344 patent/WO2016077561A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
JP2017533937A (ja) | 2017-11-16 |
US9969767B2 (en) | 2018-05-15 |
EP3218387A1 (en) | 2017-09-20 |
RU2017118489A (ru) | 2018-12-14 |
US20170334946A1 (en) | 2017-11-23 |
AU2015346303A1 (en) | 2017-06-08 |
RU2017118489A3 (pt) | 2019-02-13 |
CA2967679A1 (en) | 2016-05-19 |
CN107250153A (zh) | 2017-10-13 |
WO2016077561A1 (en) | 2016-05-19 |
AU2015346303B2 (en) | 2018-03-15 |
KR20170087478A (ko) | 2017-07-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07D | Technical examination (opinion) related to article 229 of industrial property law |
Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS. |
|
B07E | Notice of approval relating to section 229 industrial property law | ||
B08F | Application fees: dismissal - article 86 of industrial property law |
Free format text: REFERENTE A 5A ANUIDADE. |
|
B08K | Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87) |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2603 DE 24-11-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |