BR112016030599A8 - novos derivados de aminoalquilbenzotiazepina e suas utilizações - Google Patents
novos derivados de aminoalquilbenzotiazepina e suas utilizaçõesInfo
- Publication number
- BR112016030599A8 BR112016030599A8 BR112016030599A BR112016030599A BR112016030599A8 BR 112016030599 A8 BR112016030599 A8 BR 112016030599A8 BR 112016030599 A BR112016030599 A BR 112016030599A BR 112016030599 A BR112016030599 A BR 112016030599A BR 112016030599 A8 BR112016030599 A8 BR 112016030599A8
- Authority
- BR
- Brazil
- Prior art keywords
- new
- aminoalkylbenzothiazepine
- derivatives
- aminoalkylbenzothiazepine derivatives
- constipation
- Prior art date
Links
- 206010010774 Constipation Diseases 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D281/02—Seven-membered rings
- C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C13/00—Cyclic hydrocarbons containing rings other than, or in addition to, six-membered aromatic rings
- C07C13/02—Monocyclic hydrocarbons or acyclic hydrocarbon derivatives thereof
- C07C13/24—Monocyclic hydrocarbons or acyclic hydrocarbon derivatives thereof with a seven-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C13/00—Cyclic hydrocarbons containing rings other than, or in addition to, six-membered aromatic rings
- C07C13/28—Polycyclic hydrocarbons or acyclic hydrocarbon derivatives thereof
- C07C13/32—Polycyclic hydrocarbons or acyclic hydrocarbon derivatives thereof with condensed rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/02—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms
- C07C317/06—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms of a saturated carbon skeleton containing rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D281/02—Seven-membered rings
- C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Abstract
novos derivados de aminoalquilbenzotiazepina e suas utilizações. a presente invenção refere-se a um novo derivado de aminoalquilobenzotiazepina ou a um seu sal farmaceuticamente aceitável, e a uma composição farmacêutica para a prevenção ou tratamento de obstipação que compreende o mesmo como ingrediente ativo.
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR20140141869 | 2014-10-20 | ||
KR10-2014-0141869 | 2014-10-20 | ||
KR10-2015-0069949 | 2015-05-19 | ||
KR1020150069949A KR101674806B1 (ko) | 2014-10-20 | 2015-05-19 | 신규한 아미노알킬벤조티아제핀 유도체 및 이의 용도 |
PCT/KR2015/009044 WO2016064082A2 (ko) | 2014-10-20 | 2015-08-28 | 신규한 아미노알킬벤조티아제핀 유도체 및 이의 용도 |
Publications (3)
Publication Number | Publication Date |
---|---|
BR112016030599A2 BR112016030599A2 (pt) | 2017-08-15 |
BR112016030599A8 true BR112016030599A8 (pt) | 2021-07-06 |
BR112016030599B1 BR112016030599B1 (pt) | 2023-07-04 |
Family
ID=
Also Published As
Publication number | Publication date |
---|---|
CA2951824C (en) | 2019-01-08 |
UY36342A (es) | 2016-06-01 |
AU2015336400A1 (en) | 2016-12-22 |
RU2017103920A (ru) | 2018-11-22 |
JP2017527589A (ja) | 2017-09-21 |
CN106573902B (zh) | 2019-10-08 |
CA2951824A1 (en) | 2016-04-28 |
MX2016016593A (es) | 2017-04-27 |
JP6386171B2 (ja) | 2018-09-05 |
DK3210977T3 (da) | 2019-07-01 |
CN106573902A (zh) | 2017-04-19 |
ES2729305T3 (es) | 2019-10-31 |
EP3210977B1 (en) | 2019-03-20 |
AU2015336400B8 (en) | 2018-04-05 |
IL250668B (en) | 2019-07-31 |
KR101674806B1 (ko) | 2016-11-10 |
AU2015336400B2 (en) | 2017-12-07 |
KR20160047378A (ko) | 2016-05-02 |
BR112016030599A2 (pt) | 2017-08-15 |
EP3210977A2 (en) | 2017-08-30 |
US20170283386A1 (en) | 2017-10-05 |
EP3210977A4 (en) | 2018-04-11 |
AU2015336400A8 (en) | 2018-04-05 |
IL250668A0 (en) | 2017-04-30 |
RU2679891C2 (ru) | 2019-02-14 |
RU2017103920A3 (pt) | 2018-11-22 |
AR102204A1 (es) | 2017-02-08 |
WO2016064082A2 (ko) | 2016-04-28 |
WO2016064082A3 (ko) | 2016-06-09 |
US9890129B2 (en) | 2018-02-13 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] |
Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI |
|
B06U | Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette] | ||
B25D | Requested change of name of applicant approved |
Owner name: HK. INNO.N CORPORATION (KR) |
|
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 28/08/2015, OBSERVADAS AS CONDICOES LEGAIS |