BR112015024522A8 - éter de celulose esterificado, composição, dispersão sólida, forma de dosagem, invólucro de cápsula e processo para produzir o éter de celulose esterificado - Google Patents

éter de celulose esterificado, composição, dispersão sólida, forma de dosagem, invólucro de cápsula e processo para produzir o éter de celulose esterificado Download PDF

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Publication number
BR112015024522A8
BR112015024522A8 BR112015024522A BR112015024522A BR112015024522A8 BR 112015024522 A8 BR112015024522 A8 BR 112015024522A8 BR 112015024522 A BR112015024522 A BR 112015024522A BR 112015024522 A BR112015024522 A BR 112015024522A BR 112015024522 A8 BR112015024522 A8 BR 112015024522A8
Authority
BR
Brazil
Prior art keywords
esterified cellulose
cellulose ether
chr
composition
dosage form
Prior art date
Application number
BR112015024522A
Other languages
English (en)
Portuguese (pt)
Other versions
BR112015024522A2 (cg-RX-API-DMAC7.html
Inventor
Yin Ligeng
A Hillmyer Marc
L Schmitt Robert
J Guillaudeu Steven
Original Assignee
Dow Global Technologies Llc
Univ Minnesota
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Global Technologies Llc, Univ Minnesota filed Critical Dow Global Technologies Llc
Publication of BR112015024522A2 publication Critical patent/BR112015024522A2/pt
Publication of BR112015024522A8 publication Critical patent/BR112015024522A8/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08B—POLYSACCHARIDES; DERIVATIVES THEREOF
    • C08B13/00—Preparation of cellulose ether-esters
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Materials Engineering (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Polymers & Plastics (AREA)
  • Organic Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BR112015024522A 2013-05-14 2014-05-07 éter de celulose esterificado, composição, dispersão sólida, forma de dosagem, invólucro de cápsula e processo para produzir o éter de celulose esterificado BR112015024522A8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361822977P 2013-05-14 2013-05-14
PCT/US2014/037070 WO2014186185A1 (en) 2013-05-14 2014-05-07 Cellulose ethers esterified with dicarboxylic acids

Publications (2)

Publication Number Publication Date
BR112015024522A2 BR112015024522A2 (cg-RX-API-DMAC7.html) 2017-08-22
BR112015024522A8 true BR112015024522A8 (pt) 2019-12-10

Family

ID=50977076

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015024522A BR112015024522A8 (pt) 2013-05-14 2014-05-07 éter de celulose esterificado, composição, dispersão sólida, forma de dosagem, invólucro de cápsula e processo para produzir o éter de celulose esterificado

Country Status (7)

Country Link
US (1) US9890221B2 (cg-RX-API-DMAC7.html)
EP (1) EP2997046B1 (cg-RX-API-DMAC7.html)
JP (1) JP6306691B2 (cg-RX-API-DMAC7.html)
KR (1) KR20160006788A (cg-RX-API-DMAC7.html)
CN (1) CN105164162B (cg-RX-API-DMAC7.html)
BR (1) BR112015024522A8 (cg-RX-API-DMAC7.html)
WO (1) WO2014186185A1 (cg-RX-API-DMAC7.html)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6683561B2 (ja) * 2016-07-12 2020-04-22 信越化学工業株式会社 腸溶性硬カプセル用組成物及び腸溶性硬カプセルの製造方法
CN112704671B (zh) * 2020-12-28 2022-04-19 普洛药业股份有限公司 一种阿莫西林克拉维酸钾胶囊及其制备方法

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4226981A (en) 1977-09-28 1980-10-07 Shin-Etsu Chemical Co., Ltd. Ether-ester derivatives of cellulose and their applications
DE2917104A1 (de) 1979-04-27 1980-11-06 Hoechst Ag Verfahren zur viskositaetserniedrigung von celluloseethern durch ozon und seine verwendung
JPS607492B2 (ja) * 1979-04-28 1985-02-25 信越化学工業株式会社 腸溶性カプセル
US4365060A (en) 1979-04-28 1982-12-21 Shin-Etsu Chemical Co. Ltd. Enterosoluble capsules
JPS5632424A (en) * 1979-08-27 1981-04-01 Shin Etsu Chem Co Ltd Preparation of formed enteric product
JPS6225101A (ja) 1985-07-24 1987-02-03 Shin Etsu Chem Co Ltd 低重合度セルロ−スエ−テルの製造方法
JPS6281402A (ja) 1985-10-07 1987-04-14 Shin Etsu Chem Co Ltd セルロ−スエ−テル酸性ジカルボン酸エステルの製造方法
DE3620991A1 (de) 1986-06-23 1988-01-14 Henkel Kgaa Wasserloesliche alkenyl- oder alkylbernsteinsaeureester enthaltende celluloseether
DE4404840A1 (de) * 1994-02-16 1995-08-17 Wolff Walsrode Ag Thermoplastische biologisch abbaubare Polysaccharidderivate, Verfahren zu ihrer Herstellung und ihre Verwendung
DE19529409A1 (de) 1995-08-10 1997-02-13 Wolff Walsrode Ag Maleinsäureadditionsproduktgruppen enthaltende, thermoplastische und biologisch abbaubare Polysaccharidester/-etherester
EP0872233A1 (en) 1997-04-14 1998-10-21 Janssen Pharmaceutica N.V. Antiretroviral compositions with improved bioavailability
US6261218B1 (en) 1998-12-01 2001-07-17 The Dow Chemical Company Process and apparatus for making low molecular weight cellulose ethers
WO2000078285A1 (en) * 1999-06-18 2000-12-28 University Of Medicine And Dentistry Of New Jersey Controlled release of therapeutics by in-situ entrapment by matrix cross-linking
US20020076443A1 (en) * 2000-06-19 2002-06-20 Stanley Stein Multiple phase cross-linked compositions and uses thereof
DE10141680B4 (de) 2001-08-25 2004-02-26 Clariant Gmbh Verfahren zur Herstellung niederviskoser Celluloseether durch sauer-oxidativen Abbau von gemahlenen und getrockneten Celluloseethern
JP2003073443A (ja) * 2001-08-31 2003-03-12 Hiroshi Takimoto 生分解性高吸水性樹脂
JP2003160694A (ja) * 2001-11-28 2003-06-03 Hiroshi Takimoto 生分解性組成物
EP1753402B1 (en) 2004-05-28 2008-10-01 Pfizer Products Incorporated Pharmaceutical compositions with enhanced performance comprising a hpmca polymer
WO2009061815A1 (en) 2007-11-09 2009-05-14 Union Carbide Chemicals & Plastics Technology Llc Method for preparing very low viscosity cellulose ether and product
JP2011504524A (ja) 2007-11-09 2011-02-10 ダウ グローバル テクノロジーズ インコーポレイティド セルロースエーテルコーティング組成物および方法
CN102933615B (zh) * 2010-06-08 2015-08-12 陶氏环球技术有限责任公司 制备粒状可逆交联的聚合物材料的方法
WO2011159626A1 (en) 2010-06-14 2011-12-22 Bend Research, Inc. Hydroxypropyl methyl cellulose acetate succinate with enhanced acetate and succinate substitution
US9320799B2 (en) * 2012-04-11 2016-04-26 Dow Global Technologies Llc Esterified cellulose ethers having a specific substituent distribution
CN102807625A (zh) * 2012-08-23 2012-12-05 浙江中维药业有限公司 一种醋酸羟丙甲纤维素琥珀酸酯的制备方法

Also Published As

Publication number Publication date
BR112015024522A2 (cg-RX-API-DMAC7.html) 2017-08-22
KR20160006788A (ko) 2016-01-19
EP2997046B1 (en) 2019-09-25
US9890221B2 (en) 2018-02-13
CN105164162A (zh) 2015-12-16
CN105164162B (zh) 2017-11-28
JP6306691B2 (ja) 2018-04-04
US20160289344A1 (en) 2016-10-06
JP2016519198A (ja) 2016-06-30
WO2014186185A1 (en) 2014-11-20
EP2997046A1 (en) 2016-03-23

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B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements