BR112015009936A8 - uso de uma dose de formulação; bremelanotide para uso em um método para tratar disfunção sexual feminina; e unidade de dose pré-carregada - Google Patents

uso de uma dose de formulação; bremelanotide para uso em um método para tratar disfunção sexual feminina; e unidade de dose pré-carregada Download PDF

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Publication number
BR112015009936A8
BR112015009936A8 BR112015009936A BR112015009936A BR112015009936A8 BR 112015009936 A8 BR112015009936 A8 BR 112015009936A8 BR 112015009936 A BR112015009936 A BR 112015009936A BR 112015009936 A BR112015009936 A BR 112015009936A BR 112015009936 A8 BR112015009936 A8 BR 112015009936A8
Authority
BR
Brazil
Prior art keywords
bremelanotide
sexual dysfunction
dose
female sexual
treating female
Prior art date
Application number
BR112015009936A
Other languages
English (en)
Other versions
BR112015009936A2 (pt
Inventor
Spana Carl
D Edelson Jeffrey
Jordan Robert
Original Assignee
Palatin Technologies Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50628268&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112015009936(A8) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Palatin Technologies Inc filed Critical Palatin Technologies Inc
Publication of BR112015009936A2 publication Critical patent/BR112015009936A2/pt
Publication of BR112015009936A8 publication Critical patent/BR112015009936A8/pt

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/33Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • A61K38/34Melanocyte stimulating hormone [MSH], e.g. alpha- or beta-melanotropin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/06Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Reproductive Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Zoology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Dermatology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Peptides Or Proteins (AREA)

Abstract

método para tratar disfunção sexual feminina em uma paciente do sexo feminino diagnosticada com disfunção sexual feminina, mas desejando ter atividade sexual; uso de uma dose de formulação; bremelanotide para uso em um método para tratar disfunção sexual feminina; e unidade de dose pré-carregada trata-se do uso de uma dose administrada por via subcutânea entre cerca de 1,0 mg e 175 mg de bremelanotide ou um sal farmaceuticamente aceitável de bremelanotide para o tratamento de disfunção sexual feminina em mulheres enquanto reduz ou minimiza efeitos colaterais indesejáveis.
BR112015009936A 2012-11-05 2013-11-05 uso de uma dose de formulação; bremelanotide para uso em um método para tratar disfunção sexual feminina; e unidade de dose pré-carregada BR112015009936A8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261722511P 2012-11-05 2012-11-05
US201361770535P 2013-02-28 2013-02-28
PCT/US2013/068386 WO2014071339A2 (en) 2012-11-05 2013-11-05 Uses of bremelanotide in therapy for female sexual dysfunction

Publications (2)

Publication Number Publication Date
BR112015009936A2 BR112015009936A2 (pt) 2017-07-11
BR112015009936A8 true BR112015009936A8 (pt) 2019-09-17

Family

ID=50628268

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015009936A BR112015009936A8 (pt) 2012-11-05 2013-11-05 uso de uma dose de formulação; bremelanotide para uso em um método para tratar disfunção sexual feminina; e unidade de dose pré-carregada

Country Status (24)

Country Link
US (6) US9352013B2 (pt)
EP (1) EP2916856B2 (pt)
JP (1) JP6567971B2 (pt)
KR (1) KR102253526B1 (pt)
CN (2) CN104755094A (pt)
AU (1) AU2013337341B2 (pt)
BR (1) BR112015009936A8 (pt)
CA (1) CA2890081A1 (pt)
DK (1) DK2916856T4 (pt)
EA (1) EA032959B9 (pt)
ES (1) ES2701444T5 (pt)
FI (1) FI2916856T4 (pt)
GE (1) GEP20196947B (pt)
HK (1) HK1211227A1 (pt)
IL (1) IL238276B (pt)
MX (1) MX362610B (pt)
MY (1) MY179755A (pt)
NZ (1) NZ707246A (pt)
PH (1) PH12015500915B1 (pt)
PL (1) PL2916856T5 (pt)
SG (1) SG11201502949QA (pt)
UA (1) UA118656C2 (pt)
WO (1) WO2014071339A2 (pt)
ZA (1) ZA201503128B (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11590209B2 (en) * 2020-01-21 2023-02-28 Palatin Technologies, Inc. Use of bremelanotide in patients with controlled hypertension

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6579968B1 (en) 1999-06-29 2003-06-17 Palatin Technologies, Inc. Compositions and methods for treatment of sexual dysfunction
US7176279B2 (en) 2000-06-28 2007-02-13 Palatin Technologies, Inc. Cyclic peptide compositions and methods for treatment of sexual dysfunction
US7235625B2 (en) * 1999-06-29 2007-06-26 Palatin Technologies, Inc. Multiple agent therapy for sexual dysfunction
US7022674B2 (en) 1999-12-16 2006-04-04 Eli Lilly And Company Polypeptide compositions with improved stability
AU2001263766A1 (en) * 2000-05-31 2001-12-11 Novo-Nordisk A/S A disposable double pointed injection needle, and an insulin injection system comprising a disposable double pointed injection needle
CA2453515A1 (en) 2001-07-11 2003-01-23 Palatin Technologies, Inc. Linear and cyclic melanocortin receptor-specific peptides
CN101146562B (zh) * 2004-12-09 2011-11-30 韦斯特制药服务公司 自动注射装置的联结器
WO2009120656A1 (en) * 2008-03-24 2009-10-01 Palatin Technologies, Inc. Pharmaceutical for ocular indications
WO2009152079A1 (en) * 2008-06-09 2009-12-17 Palatin Technologies, Inc. Melanocortin receptor-specific peptides for treatment of sexual dysfunction
CN102665401A (zh) * 2009-11-16 2012-09-12 益普生制药股份有限公司 黑皮质素受体配体的药物组合物
RU2695703C2 (ru) * 2010-04-21 2019-07-25 Эббви Байотекнолоджи Лтд. Носимое устройство для автоматической инъекции для управляемой подачи терапевтических агентов

Also Published As

Publication number Publication date
US20220362328A1 (en) 2022-11-17
KR102253526B1 (ko) 2021-05-18
MX2015005486A (es) 2015-11-13
EP2916856A4 (en) 2016-06-22
PH12015500915A1 (en) 2015-06-29
AU2013337341B2 (en) 2018-02-22
CA2890081A1 (en) 2014-05-08
DK2916856T3 (en) 2019-01-14
NZ707246A (en) 2019-03-29
MX362610B (es) 2019-01-28
EP2916856A2 (en) 2015-09-16
AU2013337341A1 (en) 2015-05-07
FI2916856T4 (fi) 2024-01-15
DK2916856T4 (da) 2024-01-22
HK1211227A1 (en) 2016-05-20
EA032959B9 (ru) 2019-11-27
ES2701444T5 (es) 2024-05-21
ES2701444T3 (es) 2019-02-22
EA201590760A1 (ru) 2015-10-30
WO2014071339A3 (en) 2014-06-12
UA118656C2 (uk) 2019-02-25
GEP20196947B (en) 2019-02-11
WO2014071339A2 (en) 2014-05-08
ZA201503128B (en) 2016-11-30
EP2916856B2 (en) 2023-10-18
PL2916856T5 (pl) 2024-01-29
US9352013B2 (en) 2016-05-31
MY179755A (en) 2020-11-12
JP6567971B2 (ja) 2019-08-28
PH12015500915B1 (en) 2015-06-29
EP2916856B1 (en) 2018-09-19
CN104755094A (zh) 2015-07-01
US9700592B2 (en) 2017-07-11
BR112015009936A2 (pt) 2017-07-11
KR20150081345A (ko) 2015-07-13
US20150231196A1 (en) 2015-08-20
IL238276A0 (en) 2015-06-30
IL238276B (en) 2020-04-30
US20210060120A1 (en) 2021-03-04
JP2016503406A (ja) 2016-02-04
EA032959B1 (ru) 2019-08-30
US10286034B2 (en) 2019-05-14
US20180085425A1 (en) 2018-03-29
SG11201502949QA (en) 2015-06-29
PL2916856T3 (pl) 2019-02-28
US20190216888A1 (en) 2019-07-18
US20140378392A1 (en) 2014-12-25
CN117860866A (zh) 2024-04-12

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B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.