BR112014030288A2 - composição farmacêutica - Google Patents

composição farmacêutica

Info

Publication number
BR112014030288A2
BR112014030288A2 BR112014030288A BR112014030288A BR112014030288A2 BR 112014030288 A2 BR112014030288 A2 BR 112014030288A2 BR 112014030288 A BR112014030288 A BR 112014030288A BR 112014030288 A BR112014030288 A BR 112014030288A BR 112014030288 A2 BR112014030288 A2 BR 112014030288A2
Authority
BR
Brazil
Prior art keywords
pharmaceutical composition
pharmaceutically acceptable
solvate
directed
acceptable salt
Prior art date
Application number
BR112014030288A
Other languages
English (en)
Other versions
BR112014030288A8 (pt
Inventor
M Bresse David
s jones Gerald
P St Laurent Joseph
Original Assignee
Olatec Ind Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Olatec Ind Llc filed Critical Olatec Ind Llc
Publication of BR112014030288A2 publication Critical patent/BR112014030288A2/pt
Publication of BR112014030288A8 publication Critical patent/BR112014030288A8/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/095Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A61K31/10Sulfides; Sulfoxides; Sulfones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/06Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physiology (AREA)
  • Pulmonology (AREA)
  • Nutrition Science (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

1 / 1 resumo. “composiã‡ãƒo farmacãšutica” a presente invenã§ã£o ã© dirigida a uma composiã§ã£o farmacãªutica, que compreende um carreador farmaceuticamente aceitã¡vel e um composto metanossulfonilalquilnitrila, ou um sal farmaceuticamente aceitã¡vel do mesmo ou um solvato do mesmo. a presente invenã§ã£o ã© tambã©m dirigida a um mã©todo para o tratamento de inflamaã§ã£o, distãºrbios relacionados inflamatã³rios, ou dor, atravã©s da administraã§ã£o de um composto metanossulfonilalquilnitrila ou de um sal farmaceuticamente aceitã¡vel do mesmo ou um solvato do mesmo, a um paciente que esteja em necessidade do mesmo.
BR112014030288A 2012-06-05 2013-06-04 composição farmacêutica, uso da mesma, e, uso de metanossulfonilacetonitrila BR112014030288A8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261655891P 2012-06-05 2012-06-05
PCT/US2013/044149 WO2013184703A1 (en) 2012-06-05 2013-06-04 Pharmaceutical composition for treating inflammation and pain

Publications (2)

Publication Number Publication Date
BR112014030288A2 true BR112014030288A2 (pt) 2017-06-27
BR112014030288A8 BR112014030288A8 (pt) 2021-06-22

Family

ID=49671008

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112014030288A BR112014030288A8 (pt) 2012-06-05 2013-06-04 composição farmacêutica, uso da mesma, e, uso de metanossulfonilacetonitrila

Country Status (10)

Country Link
US (4) US20130324603A1 (pt)
EP (1) EP2854786B1 (pt)
JP (1) JP6178412B2 (pt)
KR (1) KR102134046B1 (pt)
CN (1) CN104334165B (pt)
AU (1) AU2013271773B2 (pt)
BR (1) BR112014030288A8 (pt)
CA (1) CA2875053C (pt)
MX (1) MX366309B (pt)
WO (1) WO2013184703A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9522878B2 (en) 2013-10-07 2016-12-20 Olatec Therapeutics Llc 4-methylsulfonyl-2-butenenitrile and its pharmaceutical use
CA2896038C (en) * 2015-07-03 2022-08-09 Glycobiosciences Inc. Polymer matrix compositions comprising a high concentration of bio-fermented sodium hyaluronate and uses thereof
EP3565540B1 (en) * 2017-01-06 2023-12-06 Olatec Therapeutics LLC A pharmaceutical composition for use in treating cardiovascular diseases
JP7229565B2 (ja) * 2018-03-21 2023-02-28 オラテック セラピューティクス リミティド ライアビリティ カンパニー メラノーマを治療するための方法

Family Cites Families (22)

* Cited by examiner, † Cited by third party
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US3427387A (en) * 1964-01-09 1969-02-11 Norwich Pharma Co Antibacterial composition containing 5-nitro-2-furyl-1,2,4-triazoles
DE3041155A1 (de) 1980-10-31 1982-06-09 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von 2,3-dichlor-sulfonyl-acrylnitrilen
GB2116964B (en) 1981-10-16 1985-07-17 Abbott Lab (1-(2-benzoxazolyl)hydrazinojalkyl nitrile derivatives
US5175192A (en) * 1984-03-19 1992-12-29 The Rockefeller University Inhibitors of the advanced glycosylation of proteins and methods of use therefor
US5218001A (en) * 1984-03-19 1993-06-08 The Rockefeller University Inhibitors of the advanced glycosylation of proteins and methods of use therefor
EP0355049A3 (en) 1988-08-18 1990-06-13 Zeneca Limited Heterocyclic compounds
JPH05310565A (ja) * 1990-04-03 1993-11-22 Univ Rockefeller 蛋白質の高度グリコシル化抑制組成物及び抑制方法
KR910018021A (ko) * 1990-04-03 1991-11-30 더 록펠러 유니버시티 단백질의 글리코실화 진행 억제제 및 그 이용 방법
US5348838A (en) 1991-07-31 1994-09-20 Kabushiki Kaisha Toshiba Photosensitive composition comprising alkali soluble binder and photoacid generator having sulfonyl group
US6362205B2 (en) * 1998-11-05 2002-03-26 Novo Nordisk A/S Substituted 3,3-diamino-2-propenenitriles, their preparation and use
US6551615B1 (en) 2001-10-18 2003-04-22 M/S. Strides Arcolab Limited Dexibuprofen-containing soft gelatin capsules and process for preparing the same
US7423064B2 (en) * 2004-09-24 2008-09-09 Olatec Industries, Llc Composition for treating bacterial, viral, fungal diseases, inflammation and pain
US20060217347A1 (en) * 2005-03-24 2006-09-28 David Perry Topical formulations of borinic acid antibiotics and their methods of use
ES2728455T3 (es) 2006-02-16 2019-10-24 Anacor Pharmaceuticals Inc Moléculas pequeñas que contienen boro como agentes antiinflamatorios
WO2007103273A2 (en) * 2006-03-03 2007-09-13 Trustees Of Boston University Thioredoxin and thioredoxin reductase inhibitors
US20100221336A1 (en) * 2007-02-14 2010-09-02 Logical Therapeutics, Inc. Method of treating arthritis, pain or inflammation with naproxen 2(methanesulfonyl)ethyl ester and a proton pump inhibitor
ES2830024T3 (es) * 2007-10-19 2021-06-02 Novartis Ag Composiciones y métodos para el tratamiento del edema macular
KR101672511B1 (ko) 2008-03-06 2016-11-03 아나코르 파마슈티칼스 인코포레이티드 소염제로써 붕소가 함유된 소분자
WO2010018814A1 (ja) 2008-08-12 2010-02-18 宇部興産株式会社 非水電解液及びそれを用いたリチウム電池
CN102438983A (zh) * 2009-03-18 2012-05-02 欧拉泰克工业有限责任公司 用于治疗炎症和疼痛的化合物
JP5932830B2 (ja) * 2010-12-15 2016-06-08 オラテック セラピューティクス リミティド ライアビリティ カンパニー 炎症及び疼痛を処置するための3‐メタンスルホニルプロピオニトリル
CN103071020B (zh) * 2012-12-30 2014-08-20 慧广世纪医疗技术(天津)有限公司 用于小儿气管-支气管炎、肺炎治疗的外敷软膏及其制法

Also Published As

Publication number Publication date
CA2875053A1 (en) 2013-12-12
AU2013271773B2 (en) 2018-03-08
JP6178412B2 (ja) 2017-08-09
US10751316B2 (en) 2020-08-25
US20130324603A1 (en) 2013-12-05
US20180353459A1 (en) 2018-12-13
CA2875053C (en) 2020-07-14
KR102134046B1 (ko) 2020-07-14
CN104334165B (zh) 2017-09-05
BR112014030288A8 (pt) 2021-06-22
MX366309B (es) 2019-07-04
EP2854786A4 (en) 2015-11-11
MX2014014814A (es) 2015-02-12
EP2854786B1 (en) 2017-03-29
EP2854786A1 (en) 2015-04-08
JP2015523987A (ja) 2015-08-20
WO2013184703A1 (en) 2013-12-12
US20230372279A1 (en) 2023-11-23
CN104334165A (zh) 2015-02-04
AU2013271773A1 (en) 2015-01-22
US20210059971A1 (en) 2021-03-04
KR20150018852A (ko) 2015-02-24

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06I Publication of requirement cancelled [chapter 6.9 patent gazette]

Free format text: ANULADA A PUBLICACAO CODIGO 6.6.1 NA RPI NO 2462 DE 13/03/2018 POR TER SIDO INDEVIDA.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]