BR112014011336A2 - composições farmacêuticas que compreendem 7-(1h-imidazol-4-ilmetil)-5,6,7,8-tetra-hidro-quinolina para tratamento de doenças e condições de pele - Google Patents

composições farmacêuticas que compreendem 7-(1h-imidazol-4-ilmetil)-5,6,7,8-tetra-hidro-quinolina para tratamento de doenças e condições de pele

Info

Publication number
BR112014011336A2
BR112014011336A2 BR112014011336A BR112014011336A BR112014011336A2 BR 112014011336 A2 BR112014011336 A2 BR 112014011336A2 BR 112014011336 A BR112014011336 A BR 112014011336A BR 112014011336 A BR112014011336 A BR 112014011336A BR 112014011336 A2 BR112014011336 A2 BR 112014011336A2
Authority
BR
Brazil
Prior art keywords
conditions
imidazol
ylmethyl
tetrahydro
quinoline
Prior art date
Application number
BR112014011336A
Other languages
English (en)
Inventor
W Gil Daniel
C Hsia Edward
E Donello John
I Dibas Mohammed
Original Assignee
Allergan Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47178364&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112014011336(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Allergan Inc filed Critical Allergan Inc
Publication of BR112014011336A2 publication Critical patent/BR112014011336A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/14Decongestants or antiallergics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Cosmetics (AREA)

Abstract

resumo patente de invenção: "composições farmacêuticas que compreendem 7-(1h-imidazol-4-ilmetil)-5,6,7,8-tetra-hidro-quinolina para tratamento de doenças e condições de pele". a presente invenção refere-se a um método para o tratamento de doenças de pele e condições da pele em um paciente com necessidade do mesmo que compreende a administração de uma quantidade terapeuticamente eficaz de uma composição farmacêutica que compreende uma quantidade terapeuticamente eficaz de 7-(1h-imidazol-4-ilmetil)-5,6,7,8-tetra-hidro-quinolina, ou dos enantiômeros dos mesmos individuais ou os tautômeros dos mesmos ou um sal farmaceuticamente aceitável do mesmo. 21235160v1 1/1 21235160v1
BR112014011336A 2011-11-10 2012-11-08 composições farmacêuticas que compreendem 7-(1h-imidazol-4-ilmetil)-5,6,7,8-tetra-hidro-quinolina para tratamento de doenças e condições de pele BR112014011336A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161558104P 2011-11-10 2011-11-10
PCT/US2012/064075 WO2013070861A1 (en) 2011-11-10 2012-11-08 Pharmaceutical compositions comprising 7-(1h-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinoline for treating skin diseases and conditions

Publications (1)

Publication Number Publication Date
BR112014011336A2 true BR112014011336A2 (pt) 2017-05-02

Family

ID=47178364

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112014011336A BR112014011336A2 (pt) 2011-11-10 2012-11-08 composições farmacêuticas que compreendem 7-(1h-imidazol-4-ilmetil)-5,6,7,8-tetra-hidro-quinolina para tratamento de doenças e condições de pele

Country Status (21)

Country Link
US (4) US20130123303A1 (pt)
EP (3) EP2776034B1 (pt)
JP (2) JP6359456B2 (pt)
KR (1) KR102004563B1 (pt)
CN (1) CN104136029A (pt)
AR (1) AR088845A1 (pt)
AU (2) AU2012335803B2 (pt)
BR (1) BR112014011336A2 (pt)
CA (1) CA2855005C (pt)
CL (1) CL2014001242A1 (pt)
DK (1) DK2776034T3 (pt)
ES (1) ES2635421T3 (pt)
IL (3) IL232483B (pt)
MX (1) MX350662B (pt)
MY (1) MY182553A (pt)
RU (2) RU2667645C1 (pt)
SG (3) SG10201809506TA (pt)
TW (3) TWI708604B (pt)
UA (1) UA109359C2 (pt)
WO (1) WO2013070861A1 (pt)
ZA (1) ZA201403396B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9283217B2 (en) 2011-11-10 2016-03-15 Allergan, Inc. Pharmaceutical compositions comprising 7-(1 H-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinoline for treating skin diseases and conditions
CN105188691A (zh) * 2013-05-06 2015-12-23 阿勒根公司 用于治疗组织创伤的α-肾上腺素能激动剂
FR3061434B1 (fr) * 2017-01-04 2019-07-12 Pierre Fabre Dermo-Cosmetique Composition cosmetique comprenant une association d'huile de pongamia et de pentylene glycol 4-t-butylcyclohexanol pour lutter contre la rosacee
RU2727695C1 (ru) * 2020-02-13 2020-07-22 Мурад Умарович Магомедов Способ комплексного лечения ринофимы

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* Cited by examiner, † Cited by third party
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PT1676579E (pt) * 1998-05-08 2009-03-24 Univ Miami Utilização de tetraciclinas sub-antimicrobianas para o tratamento de rosácea ocular
US6242442B1 (en) * 1998-12-17 2001-06-05 Alcon Laboratories, Inc. Brinzolamide and brimonidine for treating ocular conditions
US20010049369A1 (en) * 2000-02-10 2001-12-06 Jablonski Monica M. Brimonidine compositions and methods for retinal degeneration
US6468989B1 (en) 2000-07-13 2002-10-22 Dow Pharmaceutical Sciences Gel compositions containing metronidazole
US6387383B1 (en) 2000-08-03 2002-05-14 Dow Pharmaceutical Sciences Topical low-viscosity gel composition
US20020198209A1 (en) 2001-05-03 2002-12-26 Allergan Sales Inc. Compositions having enhanced pharmacokinetic characteristics
US6680062B2 (en) 2001-10-05 2004-01-20 Color Access, Inc. Anti-irritating rosacea treatment
US7030149B2 (en) * 2002-04-19 2006-04-18 Allergan, Inc. Combination of brimonidine timolol for topical ophthalmic use
US20040146539A1 (en) * 2003-01-24 2004-07-29 Gupta Shyam K. Topical Nutraceutical Compositions with Selective Body Slimming and Tone Firming Antiaging Benefits
US7439241B2 (en) * 2003-05-27 2008-10-21 Galderma Laboratories, Inc. Compounds, formulations, and methods for treating or preventing rosacea
US20050020600A1 (en) * 2003-07-23 2005-01-27 Scherer Warren J. Methods of treating cutaneous flushing using selective alpha-2-adrenergic receptor agonists
CN100558360C (zh) * 2003-11-20 2009-11-11 奥特拉控股公司 羟胺组合物在制备缓解黄斑变性和其他眼科疾病的药物中的用途
US7812049B2 (en) 2004-01-22 2010-10-12 Vicept Therapeutics, Inc. Method and therapeutic/cosmetic topical compositions for the treatment of rosacea and skin erythema using α1-adrenoceptor agonists
MXPA06013649A (es) * 2004-05-25 2007-07-09 Sansrosa Pharmaceutical Dev In Compuestos, formulaciones, y metodos para tratar o prevenir desordenes inflamatorios de la piel.
US20070203144A1 (en) * 2006-01-17 2007-08-30 Allergan, Inc. Use of Memantine and Brimonidine to Attenuate Vitreoretinal Vascular Endothelial Growth Factor (VEGF) Protein Levels in Animals
US7323477B2 (en) 2006-02-02 2008-01-29 Allergan, Inc. 7-((1H-imidazol-4-yl)methyl)-5,6,7,8-tetrahydroquinoline
RU2321399C1 (ru) * 2006-06-01 2008-04-10 Федеральное государственное учреждение "Нижегородский научно-исследовательский кожно-венерологический институт Федерального агентства по здравоохранению и социальному развитию" Способ лечения больных розацеа
WO2008124151A2 (en) * 2007-04-09 2008-10-16 Avicena Group, Inc. Use of creatine compounds for the treatment of eye disorders
US20090061020A1 (en) * 2007-08-31 2009-03-05 Theobald Klaus P Brimonidine Compositions for Treating Erythema
WO2009052073A2 (en) * 2007-10-18 2009-04-23 Allergan, Inc. Method of treating sensorimotor disorders with alpha-2 adrenergic receptor agonists
US20100203165A1 (en) * 2008-08-01 2010-08-12 Gerald Horn Compositions and methods for treatment of disorders or conditions of the eye
SI2320911T1 (sl) * 2008-08-01 2014-12-31 Eye Therapies Llc Vazokonstrikcijski sestavki in metode uporabe
FR2942138A1 (fr) 2009-02-16 2010-08-20 Galderma Res & Dev Association de composes pour le traitement ou la prevention des affections dermatologiques
KR20120125230A (ko) * 2009-10-26 2012-11-14 갈더마파마 에스.아. 급성 홍반 치료 또는 예방 방법
US8394800B2 (en) * 2009-11-19 2013-03-12 Galderma Laboratories, L.P. Method for treating psoriasis
WO2011117378A2 (en) * 2010-03-26 2011-09-29 Galderma Research & Development Improved methods and compositions for safe and effective treatment of telangiectasia
WO2011117377A2 (en) * 2010-03-26 2011-09-29 Galderma Research & Development Improved methods and compositions for safe and effective treatment of erythema
EP2600832A1 (en) * 2010-08-06 2013-06-12 Galderma Research & Development Combination of compounds for treating or preventing skin diseases

Also Published As

Publication number Publication date
KR102004563B1 (ko) 2019-07-26
IL232483B (en) 2018-10-31
ZA201403396B (en) 2015-07-29
EP2776034B1 (en) 2017-03-22
JP2017149767A (ja) 2017-08-31
JP6526737B2 (ja) 2019-06-05
TW201713338A (zh) 2017-04-16
AU2016216627A1 (en) 2016-09-08
CA2855005C (en) 2016-11-22
MY182553A (en) 2021-01-25
US9308201B2 (en) 2016-04-12
ES2635421T3 (es) 2017-10-03
SG11201402246RA (en) 2014-06-27
JP6359456B2 (ja) 2018-07-18
RU2630978C2 (ru) 2017-09-15
CL2014001242A1 (es) 2014-11-14
NZ624771A (en) 2016-11-25
US20170095466A1 (en) 2017-04-06
JP2014533271A (ja) 2014-12-11
MX2014005640A (es) 2014-09-22
IL268757A (en) 2019-10-31
US20160051534A1 (en) 2016-02-25
TW202014189A (zh) 2020-04-16
TWI580424B (zh) 2017-05-01
US20150231128A1 (en) 2015-08-20
DK2776034T3 (en) 2017-07-10
KR20140107237A (ko) 2014-09-04
CA2855005A1 (en) 2013-05-16
IL261269A (en) 2018-10-31
TW201328694A (zh) 2013-07-16
AU2012335803A1 (en) 2014-05-29
SG10201609145PA (en) 2016-12-29
EP3184110A1 (en) 2017-06-28
UA109359C2 (xx) 2015-08-10
AU2012335803B2 (en) 2016-05-26
RU2667645C1 (ru) 2018-09-21
AR088845A1 (es) 2014-07-10
RU2014122758A (ru) 2015-12-20
MX350662B (es) 2017-09-13
EP3763370A1 (en) 2021-01-13
EP2776034A1 (en) 2014-09-17
TWI708604B (zh) 2020-11-01
US20130123303A1 (en) 2013-05-16
AU2016216627B2 (en) 2017-10-19
IL232483A0 (en) 2014-06-30
SG10201809506TA (en) 2018-11-29
CN104136029A (zh) 2014-11-05
WO2013070861A1 (en) 2013-05-16
EP3184110B1 (en) 2020-10-07

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]
B350 Update of information on the portal [chapter 15.35 patent gazette]