BR112013020520A2 - derivados de isoxazolina, composição para o controle de parasitas os compreendendo e uso dos mesmos - Google Patents

derivados de isoxazolina, composição para o controle de parasitas os compreendendo e uso dos mesmos

Info

Publication number
BR112013020520A2
BR112013020520A2 BR112013020520A BR112013020520A BR112013020520A2 BR 112013020520 A2 BR112013020520 A2 BR 112013020520A2 BR 112013020520 A BR112013020520 A BR 112013020520A BR 112013020520 A BR112013020520 A BR 112013020520A BR 112013020520 A2 BR112013020520 A2 BR 112013020520A2
Authority
BR
Brazil
Prior art keywords
parasites
composition
control
isoxazoline derivatives
isoxazoline
Prior art date
Application number
BR112013020520A
Other languages
English (en)
Inventor
Noëlle Gauvry
Steve Nanchen
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR112013020520A2 publication Critical patent/BR112013020520A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/84—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms six-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,4
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/24—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing the groups, or; Thio analogues thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Abstract

derivados de isoxazolina para o controle de pragas de invertebrados a invenção relaciona-se a novos compostos isoxazolina de fórmula (i), em que as variáveis possuem o significado como indicado nas reivindicações; em forma livre e em forma de sal; e opcionalmente os enantiômeros e isômeros geométricos desses. os compostos de fórmula (i) são úteis no controle de parasitas, em particular ectoparasitas, em animais de sangue quente.
BR112013020520A 2011-02-10 2012-02-09 derivados de isoxazolina, composição para o controle de parasitas os compreendendo e uso dos mesmos BR112013020520A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH2472011 2011-02-10
PCT/EP2012/052241 WO2012107533A1 (en) 2011-02-10 2012-02-09 Isoxazoline derivatives for controlling invertebrate pests

Publications (1)

Publication Number Publication Date
BR112013020520A2 true BR112013020520A2 (pt) 2016-07-12

Family

ID=45607737

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112013020520A BR112013020520A2 (pt) 2011-02-10 2012-02-09 derivados de isoxazolina, composição para o controle de parasitas os compreendendo e uso dos mesmos

Country Status (15)

Country Link
US (2) US20130324538A1 (pt)
EP (1) EP2673273A1 (pt)
JP (1) JP2014505089A (pt)
CN (1) CN103347880B (pt)
AR (1) AR085354A1 (pt)
AU (1) AU2012215440B2 (pt)
BR (1) BR112013020520A2 (pt)
CA (1) CA2826067A1 (pt)
CL (1) CL2013002296A1 (pt)
CO (1) CO6731114A2 (pt)
MX (1) MX2013009211A (pt)
RU (1) RU2013141413A (pt)
TW (1) TWI511966B (pt)
WO (1) WO2012107533A1 (pt)
ZA (1) ZA201305226B (pt)

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US11883530B2 (en) 2013-12-20 2024-01-30 Intervet Inc. Isoxazoline compositions and use thereof in the prevention or treatment of parasite infestations in animals

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UY33403A (es) * 2010-06-17 2011-12-30 Novartis Ag Compuestos orgánicos con novedosas isoxazolinas, sus n-óxidos, s-óxidos y sales
AR086113A1 (es) 2011-04-30 2013-11-20 Abbott Lab Isoxazolinas como agentes terapeuticos
WO2012155352A1 (en) * 2011-05-19 2012-11-22 Eli Lilly And Company Dihydroisoxazole compounds, parasiticidal uses and formulations thereof
RU2660346C1 (ru) 2012-02-06 2018-07-05 Мериал, Инк. Паразитицидные пероральные ветеринарные композиции, включающие системно действующие активные агенты, способы и применение этих композиций и способов
JO3626B1 (ar) 2012-02-23 2020-08-27 Merial Inc تركيبات موضعية تحتوي على فيبرونيل و بيرميثرين و طرق استخدامها
SI2953942T1 (en) 2013-02-06 2018-03-30 Bayer Cropscience Ag Halogen-substituted pyrazole derivatives such as pesticides
US10533002B2 (en) 2013-06-24 2020-01-14 Boehringer Ingelheim Animal Health USA Inc. Thiophene- or furan-substituted isothiazoline compounds as pesticides
EP3063144B1 (en) 2013-11-01 2021-09-08 Boehringer Ingelheim Animal Health USA Inc. Antiparasitic and pesticidal isoxazoline compounds
CN110839641A (zh) * 2013-12-20 2020-02-28 英特维特国际股份有限公司 异噁唑啉衍生物用于治疗或预防家禽中的节肢动物侵袭的用途
RU2016131792A (ru) 2014-01-03 2018-02-06 Байер Энимэл Хельс ГмбХ Новые пиразолил-гетероариламиды в качестве средств для борьбы с вредителями
US10857121B2 (en) 2014-04-17 2020-12-08 Merial Inc. Use of malononitrile compounds for protecting animals from parasites
US10208015B2 (en) 2014-07-15 2019-02-19 Bayer Animal Health Gmbh Aryl-triazolyl pyridines as pest control agents
EP3018129A1 (en) * 2014-11-10 2016-05-11 Novartis Tiergesundheit AG Diaryl isoxazoline compound
UY36570A (es) * 2015-02-26 2016-10-31 Merial Inc Formulaciones inyectables de acción prolongada que comprenden un agente activo isoxazolina, métodos y usos de las mismas
EA036272B1 (ru) * 2015-04-08 2020-10-21 БЁРИНГЕР ИНГЕЛЬХАЙМ ЭНИМАЛ ХЕЛТ ЮЭсЭй ИНК. Инъецируемые препараты замедленного высвобождения, содержащие изоксазолиновое действующее вещество, способы и применение
CN107835818B (zh) 2015-05-20 2022-04-29 勃林格殷格翰动物保健美国公司 驱虫缩酚酸肽化合物
UY37137A (es) * 2016-02-24 2017-09-29 Merial Inc Compuestos antiparasitarios de isoxazolina, formulaciones inyectables de acción prolongada que los comprenden, métodos y usos de los mismos
CN109843878A (zh) * 2016-08-10 2019-06-04 拜耳作物科学股份公司 用作害虫防治剂的取代的2-杂环基咪唑基甲酰胺
US10653144B2 (en) 2016-10-14 2020-05-19 Boehringer Ingelheim Animal Health USA Inc. Pesticidal and parasiticidal vinyl isoxazoline compounds
CN110167921A (zh) 2016-11-16 2019-08-23 勃林格殷格翰动物保健美国公司 驱蠕虫缩肽化合物
WO2018166855A1 (en) 2017-03-16 2018-09-20 Basf Se Heterobicyclic substituted dihydroisoxazoles
JP2020530850A (ja) 2017-08-14 2020-10-29 ベーリンガー インゲルハイム アニマル ヘルス ユーエスエイ インコーポレイテッド 殺有害生物および殺寄生生物ピラゾール−イソキサゾリン化合物
IL307992A (en) 2017-12-15 2023-12-01 Tarsus Pharmaceuticals Inc Parasitic formulations containing isoxazoline and methods for treating blepharitis
TWI812673B (zh) * 2018-02-12 2023-08-21 美商富曼西公司 用於防治無脊椎害蟲之萘異噁唑啉化合物
AU2019301510A1 (en) 2018-07-09 2021-03-04 Boehringer Ingelheim Pharma Gmbh & Co. Kg Anthelminthic heterocyclic compounds
CN113260419A (zh) 2018-11-20 2021-08-13 勃林格殷格翰动物保健美国公司 吲唑基氰基乙基氨基化合物、其组合物、其制备方法和其使用方法
EP3941587A1 (en) 2019-03-19 2022-01-26 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic aza-benzothiophene and aza-benzofuran compounds
CN114269324A (zh) * 2019-06-19 2022-04-01 塔苏斯制药有限公司 用于治疗睑炎的异恶唑啉驱虫剂制剂和方法
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US11883530B2 (en) 2013-12-20 2024-01-30 Intervet Inc. Isoxazoline compositions and use thereof in the prevention or treatment of parasite infestations in animals

Also Published As

Publication number Publication date
NZ613191A (en) 2015-06-26
WO2012107533A1 (en) 2012-08-16
AR085354A1 (es) 2013-09-25
CL2013002296A1 (es) 2014-03-14
TWI511966B (zh) 2015-12-11
US20160024062A1 (en) 2016-01-28
TW201309683A (zh) 2013-03-01
AU2012215440A1 (en) 2013-08-01
ZA201305226B (en) 2014-03-26
CO6731114A2 (es) 2013-08-15
CN103347880B (zh) 2015-11-25
RU2013141413A (ru) 2015-03-20
CN103347880A (zh) 2013-10-09
JP2014505089A (ja) 2014-02-27
EP2673273A1 (en) 2013-12-18
US20130324538A1 (en) 2013-12-05
AU2012215440B2 (en) 2015-08-27
MX2013009211A (es) 2013-08-29
CA2826067A1 (en) 2012-08-16

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