BR112013008362A2 - combinações - Google Patents

combinações

Info

Publication number
BR112013008362A2
BR112013008362A2 BR112013008362A BR112013008362A BR112013008362A2 BR 112013008362 A2 BR112013008362 A2 BR 112013008362A2 BR 112013008362 A BR112013008362 A BR 112013008362A BR 112013008362 A BR112013008362 A BR 112013008362A BR 112013008362 A2 BR112013008362 A2 BR 112013008362A2
Authority
BR
Brazil
Prior art keywords
agonist
inhibitor
receptor
combinations
antagonist
Prior art date
Application number
BR112013008362A
Other languages
English (en)
Inventor
Frank Burkamp
Peter Robert Hansen
Svetlana Ivanova
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BR112013008362A2 publication Critical patent/BR112013008362A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/007—Pulmonary tract; Aromatherapy
    • A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Otolaryngology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

combinações. a invenção refere-se a um produto farmacêutico que compreende, em combinação, (1) um denominado agonista e receptor de glicorticosteroide e (2) um agonista de adrenorreceptor <225>2, um agonista duplo de adrenorreceptor <225>2/antagonista do receptor m3, um antagonista muscarínico, um inibidor da p38 quinase, um inibidor da elastase do neutrófilo, um inibidor da fosfodiesterase pde4, um inibidor de ikk2 quinase ou um agonista do receptor de glicorticoide não esteroidal e o uso do dito produto no tratamento de doenças respiratórias.
BR112013008362A 2010-10-07 2011-10-05 combinações BR112013008362A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB1016912.6A GB201016912D0 (en) 2010-10-07 2010-10-07 Novel combination
PCT/GB2011/051898 WO2012046050A1 (en) 2010-10-07 2011-10-05 Novel combinations

Publications (1)

Publication Number Publication Date
BR112013008362A2 true BR112013008362A2 (pt) 2016-06-14

Family

ID=43304217

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112013008362A BR112013008362A2 (pt) 2010-10-07 2011-10-05 combinações

Country Status (14)

Country Link
EP (1) EP2624838A1 (pt)
JP (1) JP2013538867A (pt)
KR (1) KR20130126595A (pt)
CN (1) CN103249418A (pt)
AU (1) AU2011311310A1 (pt)
BR (1) BR112013008362A2 (pt)
CA (1) CA2813684A1 (pt)
GB (1) GB201016912D0 (pt)
IL (1) IL225312A0 (pt)
IN (1) IN2013MN00567A (pt)
MX (1) MX2013003816A (pt)
RU (1) RU2013115103A (pt)
SG (1) SG188575A1 (pt)
WO (1) WO2012046050A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20150027922A (ko) * 2013-09-04 2015-03-13 주식회사 대웅제약 신규한 항진균성 피리디닐하이드라자이드 유도체
KR101657678B1 (ko) * 2013-11-05 2016-09-20 주식회사 대웅제약 신규한 화합물, 이의 제조방법 및 이를 포함하는 항진균제 조성물
PL3377500T3 (pl) * 2015-11-16 2023-01-23 Esteve Pharmaceuticals, S.A. Związki oksadiazaspiro do leczenia nadużywania i uzależnienia od narkotyków/leków
WO2018059537A1 (zh) * 2016-09-30 2018-04-05 四川海思科制药有限公司 一种二氮杂螺[5.5]十一碳烷衍生物及其用途

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Also Published As

Publication number Publication date
CN103249418A (zh) 2013-08-14
IL225312A0 (en) 2013-06-27
MX2013003816A (es) 2013-05-01
IN2013MN00567A (pt) 2015-10-09
JP2013538867A (ja) 2013-10-17
AU2011311310A1 (en) 2013-04-11
EP2624838A1 (en) 2013-08-14
KR20130126595A (ko) 2013-11-20
RU2013115103A (ru) 2014-11-20
SG188575A1 (en) 2013-04-30
WO2012046050A1 (en) 2012-04-12
GB201016912D0 (en) 2010-11-24
CA2813684A1 (en) 2012-04-12

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Legal Events

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B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

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B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]