BR112012014471A2 - método para o tratamento de cicatrizes e de distúrbios mediados por beta-catenina usando compostos nefopam - Google Patents

método para o tratamento de cicatrizes e de distúrbios mediados por beta-catenina usando compostos nefopam

Info

Publication number
BR112012014471A2
BR112012014471A2 BR112012014471A BR112012014471A BR112012014471A2 BR 112012014471 A2 BR112012014471 A2 BR 112012014471A2 BR 112012014471 A BR112012014471 A BR 112012014471A BR 112012014471 A BR112012014471 A BR 112012014471A BR 112012014471 A2 BR112012014471 A2 BR 112012014471A2
Authority
BR
Brazil
Prior art keywords
catenin
nefopam
disorders
cancer
compounds
Prior art date
Application number
BR112012014471A
Other languages
English (en)
Portuguese (pt)
Inventor
A Alman Benjamin
Hong Helen
Poon Raymond
Original Assignee
Hospital For Sick Children
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44166687&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112012014471(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hospital For Sick Children filed Critical Hospital For Sick Children
Publication of BR112012014471A2 publication Critical patent/BR112012014471A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/5545Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having eight-membered rings not containing additional condensed or non-condensed nitrogen-containing 3-7 membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/191Carboxylic acids, e.g. valproic acid having two or more hydroxy groups, e.g. gluconic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Emergency Medicine (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Inorganic Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Materials Engineering (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
BR112012014471A 2009-12-15 2010-12-15 método para o tratamento de cicatrizes e de distúrbios mediados por beta-catenina usando compostos nefopam BR112012014471A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US28663309P 2009-12-15 2009-12-15
PCT/CA2010/002014 WO2011072394A1 (en) 2009-12-15 2010-12-15 METHOD OF TREATING SCARS AND ß-CATENIN-MEDIATED DISORDERS USING NEFOPAM COMPOUNDS

Publications (1)

Publication Number Publication Date
BR112012014471A2 true BR112012014471A2 (pt) 2017-06-06

Family

ID=44166687

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012014471A BR112012014471A2 (pt) 2009-12-15 2010-12-15 método para o tratamento de cicatrizes e de distúrbios mediados por beta-catenina usando compostos nefopam

Country Status (10)

Country Link
US (4) US8957107B2 (enExample)
EP (1) EP2512468B1 (enExample)
JP (1) JP5792185B2 (enExample)
KR (1) KR101753439B1 (enExample)
CN (2) CN105687185B (enExample)
BR (1) BR112012014471A2 (enExample)
CA (1) CA2782472C (enExample)
DK (1) DK2512468T3 (enExample)
ES (1) ES2594900T3 (enExample)
WO (1) WO2011072394A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2512468B1 (en) * 2009-12-15 2016-08-24 The Hospital for Sick Children METHOD OF TREATING SCARS AND ß-CATENIN-MEDIATED DISORDERS USING NEFOPAM COMPOUNDS
US10736905B1 (en) 2016-09-09 2020-08-11 Shahin Fatholahi Nefopam dosage forms and methods of treatment
WO2018223023A1 (en) * 2017-06-02 2018-12-06 Beta Cat Pharmaceuticals, Inc. Methods for treatment of fibrotic diseases
US11446311B2 (en) 2017-09-08 2022-09-20 Shahin Fatholahi Methods for treating pain associated with sickle cell disease
US10736874B1 (en) 2017-09-08 2020-08-11 Shahin Fatholahi Methods for treating pain associated with sickle cell disease
US11266637B2 (en) * 2018-06-01 2022-03-08 Iterion Therapeutics, Inc. Formulations of tegavivint and related compounds
CN110638780A (zh) * 2019-09-11 2020-01-03 华益药业科技(安徽)有限公司 一种盐酸奈福泮片及其制备方法

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6294350B1 (en) 1997-06-05 2001-09-25 Dalhousie University Methods for treating fibroproliferative diseases
US6630142B2 (en) 1999-05-03 2003-10-07 Zymogenetics, Inc. Method of treating fibroproliferative disorders
US6638981B2 (en) * 2001-08-17 2003-10-28 Epicept Corporation Topical compositions and methods for treating pain
US20030190308A1 (en) * 2002-03-19 2003-10-09 Braun Ralph P. Adjuvant
GB0213869D0 (en) * 2002-06-17 2002-07-31 Arakis Ltd The treatment of pain
US20060019940A1 (en) 2002-12-20 2006-01-26 Baxter Andrew D Novel benzoxazocines and their therapeutic use
BR0317467A (pt) 2002-12-20 2005-11-16 Arakis Ltd Benzoxazocinas e seu uso como inibidores de reassimilação de monoaminas
GB0330049D0 (en) 2003-12-24 2004-02-04 Arakis Ltd The treatment of neuropathic pain conditions
JP2007533718A (ja) 2004-04-21 2007-11-22 ソセイ・アール・アンド・ディー・リミテッド ベンゾオキサゾシン類およびそれらのモノアミン再取込み阻害剤としての治療的使用
GB2413322A (en) 2004-04-21 2005-10-26 Arakis Ltd Nefopam analogues
CN1569004A (zh) * 2004-05-13 2005-01-26 南昌弘益科技有限公司 盐酸奈福泮滴丸及其制备方法
FR2880275B1 (fr) 2005-01-06 2007-04-13 Biocodex Utilisation de composes pharmacologiques pour la prevention ou le traitement de la tolerance aigue aux morphiniques
GB0506835D0 (en) * 2005-04-04 2005-05-11 Arakis Ltd Therapeutic use of nefopam
GB0515703D0 (en) 2005-07-29 2005-09-07 Arakis Ltd Therapeutic use of nefopam
CN101002756A (zh) 2007-01-19 2007-07-25 陶燃 盐酸奈福泮的透皮贴片制剂
GB0721013D0 (en) 2007-10-25 2007-12-05 Sosei R & D Ltd New Salts
US8158367B2 (en) 2008-06-16 2012-04-17 Academia Sinica Cancer diagnosis based on levels of antibodies against Globo H and its fragments
GB2461874B (en) 2008-07-14 2012-11-21 Caltec Ltd Separation system and method
FR2940911B1 (fr) * 2009-01-13 2012-09-21 Philippe Perovitch Formulation pour l'administration par voie trans-muqueuse buccale de molecules antalgiques et/ou anti-spasmodiques
EP2512468B1 (en) * 2009-12-15 2016-08-24 The Hospital for Sick Children METHOD OF TREATING SCARS AND ß-CATENIN-MEDIATED DISORDERS USING NEFOPAM COMPOUNDS

Also Published As

Publication number Publication date
US20170172980A1 (en) 2017-06-22
KR20120110117A (ko) 2012-10-09
US20170281594A1 (en) 2017-10-05
EP2512468B1 (en) 2016-08-24
HK1174565A1 (zh) 2013-06-14
US8957107B2 (en) 2015-02-17
KR101753439B1 (ko) 2017-07-19
US20150105363A1 (en) 2015-04-16
ES2594900T3 (es) 2016-12-23
CN102781442A (zh) 2012-11-14
US20120294928A1 (en) 2012-11-22
HK1224224A1 (zh) 2017-08-18
WO2011072394A1 (en) 2011-06-23
US9566263B2 (en) 2017-02-14
CN105687185B (zh) 2019-07-09
JP2013513625A (ja) 2013-04-22
CN105687185A (zh) 2016-06-22
US10722493B2 (en) 2020-07-28
CA2782472C (en) 2019-04-16
CN102781442B (zh) 2016-02-17
DK2512468T3 (en) 2016-11-14
CA2782472A1 (en) 2011-06-23
EP2512468A1 (en) 2012-10-24
JP5792185B2 (ja) 2015-10-07
EP2512468A4 (en) 2013-08-07

Similar Documents

Publication Publication Date Title
BR112012014471A2 (pt) método para o tratamento de cicatrizes e de distúrbios mediados por beta-catenina usando compostos nefopam
CY1124197T1 (el) Antinohmatika πολυνουκλεοτιδια για να διεγειρεται παραλειψη εξονιου και μεθοδοι θεραπειας δυστροφιων
BR112015022998A2 (pt) composições melhoradas para o tratamento de distrofia muscular
CY1121357T1 (el) Νεος ανοσοτροποποιητης και αντιφλεγμονωδεις ενωσεις
PH12017502141A1 (en) Compounds and their methods of use
MY192633A (en) 1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase
BR112015023038A2 (pt) composições para salto de exon para o tratamento da distrofia muscular
GEP20146138B (en) Method for treating androgen receptor positive cancers
ECSP14013223A (es) Métodos para tratar el cáncer por el uso de antagonistas de unión al eje pd-1 e inhibidores de mek
SA515360657B1 (ar) مثبطات ديميثيلاز هيستون
BR112015023001A2 (pt) composição de salto de exon para tratamento de distrofia muscular
EA201100879A1 (ru) Производные пиридопиримидина в качестве ингибиторов аутотаксина
MX352672B (es) Compuestos heterocíclicos como inhibidores de mdm2 para el tratamiento del cáncer.
MX377405B (es) Compuestos para el tratamiento de cáncer.
UA107783C2 (en) Isoindoline compounds for use in treating cancer
MX394676B (es) Métodos para tratar el cáncer.
PH12015502414A1 (en) Enhancer of zeste homolog 2 inhibitors
WO2012006181A3 (en) Compositions and methods for inhibiting oncogenic micrornas and treatment of cancer
MX391013B (es) Compuestos y metodos para tratar influenza.
PH12016501048A1 (en) Piperidine derivatives as mdm2 inhibitors for the treatment of cancer
EA201390015A1 (ru) Композиции и способы ингибирования пути jak
GEP20156372B (en) Pyridazinone compounds and their use as daao inhibitors
MY161473A (en) Compositions, synthesis, and methods of utilizing arylpiperazine derivatives
BR112012008546A2 (pt) derivados de sulfóxido para o tratamento de tumor
UA107455C2 (uk) Похідні індолу як протиракові агенти

Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law
B06F Objections, documents and/or translations needed after an examination request according art. 34 industrial property law
B07E Notice of approval relating to section 229 industrial property law

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06U Preliminary requirement: requests with searches performed by other patent offices: suspension of the patent application procedure
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements