BR112012007701A2 - método para obter um composto, cassete para realizar o método, e, composto - Google Patents
método para obter um composto, cassete para realizar o método, e, compostoInfo
- Publication number
- BR112012007701A2 BR112012007701A2 BR112012007701A BR112012007701A BR112012007701A2 BR 112012007701 A2 BR112012007701 A2 BR 112012007701A2 BR 112012007701 A BR112012007701 A BR 112012007701A BR 112012007701 A BR112012007701 A BR 112012007701A BR 112012007701 A2 BR112012007701 A2 BR 112012007701A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- cassette
- perform
- compounds
- useful
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 8
- 150000001875 compounds Chemical class 0.000 title abstract 7
- 102000005915 GABA Receptors Human genes 0.000 abstract 1
- 108010005551 GABA Receptors Proteins 0.000 abstract 1
- 238000011503 in vivo imaging Methods 0.000 abstract 1
- 239000002243 precursor Substances 0.000 abstract 1
- 238000001308 synthesis method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Optics & Photonics (AREA)
- Physics & Mathematics (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0917611.6A GB0917611D0 (en) | 2009-10-08 | 2009-10-08 | Automated radiosynthesis |
| US25089209P | 2009-10-13 | 2009-10-13 | |
| PCT/EP2010/065077 WO2011042529A1 (en) | 2009-10-08 | 2010-10-08 | Automated radiosynthesis |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112012007701A2 true BR112012007701A2 (pt) | 2015-09-08 |
Family
ID=41402710
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112012007701A BR112012007701A2 (pt) | 2009-10-08 | 2010-10-08 | método para obter um composto, cassete para realizar o método, e, composto |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US8946410B2 (enExample) |
| EP (1) | EP2486040B1 (enExample) |
| JP (1) | JP5870031B2 (enExample) |
| KR (1) | KR20120095359A (enExample) |
| CN (1) | CN102548996B (enExample) |
| AU (1) | AU2010305355B2 (enExample) |
| BR (1) | BR112012007701A2 (enExample) |
| CA (1) | CA2774031A1 (enExample) |
| GB (1) | GB0917611D0 (enExample) |
| IL (1) | IL218454A0 (enExample) |
| IN (1) | IN2012DN02214A (enExample) |
| MX (1) | MX2012003994A (enExample) |
| NZ (1) | NZ598659A (enExample) |
| RU (1) | RU2012113138A (enExample) |
| WO (1) | WO2011042529A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201105445D0 (en) * | 2011-03-31 | 2011-05-18 | Ge Healthcare Ltd | Radiolabelled flumazenil derivatives |
| KR101441406B1 (ko) * | 2011-05-25 | 2014-11-04 | 주식회사 바이오이미징코리아 | 디아릴이오도늄 염 전구체를 이용한 플로오린-18이 표지된 플루마제닐의 제조 방법 |
| GB201209082D0 (en) * | 2012-05-24 | 2012-07-04 | Ge Healthcare Ltd | Purification method |
| CN112979658B (zh) * | 2021-02-22 | 2022-05-31 | 南湖实验室 | 一种氟马西尼的制备方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA806016B (en) * | 1979-10-04 | 1981-09-30 | Hoffmann La Roche | Imidazodiazepine derivatives |
| CA1184175A (en) * | 1981-02-27 | 1985-03-19 | Walter Hunkeler | Imidazodiazepines |
| GB8927928D0 (en) | 1989-12-11 | 1990-02-14 | Roussel Lab Ltd | Chemical compounds |
| JP3537914B2 (ja) * | 1995-05-18 | 2004-06-14 | 株式会社生体機能研究所 | [18f]フルオロ芳香族化合物の製造法 |
| FI101305B1 (fi) * | 1996-03-18 | 1998-05-29 | Map Medical Technologies Oy | Radiofarmaseuttisena aineena käyttökelpoiset radiojodatut bentsodiatsepiini-johdannaiset ja niiden käyttö diagnostiikassa |
| GB0407952D0 (en) * | 2004-04-08 | 2004-05-12 | Amersham Plc | Fluoridation method |
| WO2007141529A1 (en) * | 2006-06-09 | 2007-12-13 | Ge Healthcare Limited | Fluoridation method |
| GB0803729D0 (en) * | 2008-02-29 | 2008-04-09 | Ge Healthcare Ltd | Imaging the central nervous system |
-
2009
- 2009-10-08 GB GBGB0917611.6A patent/GB0917611D0/en not_active Ceased
-
2010
- 2010-10-08 CN CN201080045665.4A patent/CN102548996B/zh not_active Expired - Fee Related
- 2010-10-08 US US13/394,655 patent/US8946410B2/en not_active Expired - Fee Related
- 2010-10-08 NZ NZ598659A patent/NZ598659A/en not_active IP Right Cessation
- 2010-10-08 RU RU2012113138/04A patent/RU2012113138A/ru not_active Application Discontinuation
- 2010-10-08 CA CA2774031A patent/CA2774031A1/en not_active Abandoned
- 2010-10-08 KR KR1020127009090A patent/KR20120095359A/ko not_active Withdrawn
- 2010-10-08 WO PCT/EP2010/065077 patent/WO2011042529A1/en not_active Ceased
- 2010-10-08 JP JP2012532611A patent/JP5870031B2/ja not_active Expired - Fee Related
- 2010-10-08 AU AU2010305355A patent/AU2010305355B2/en not_active Ceased
- 2010-10-08 EP EP10762695.4A patent/EP2486040B1/en not_active Not-in-force
- 2010-10-08 BR BR112012007701A patent/BR112012007701A2/pt not_active IP Right Cessation
- 2010-10-08 MX MX2012003994A patent/MX2012003994A/es not_active Application Discontinuation
- 2010-10-08 IN IN2214DEN2012 patent/IN2012DN02214A/en unknown
-
2012
- 2012-03-04 IL IL218454A patent/IL218454A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011042529A1 (en) | 2011-04-14 |
| EP2486040A1 (en) | 2012-08-15 |
| JP2013507343A (ja) | 2013-03-04 |
| NZ598659A (en) | 2014-02-28 |
| RU2012113138A (ru) | 2013-11-20 |
| US8946410B2 (en) | 2015-02-03 |
| GB0917611D0 (en) | 2009-11-25 |
| US20120190843A1 (en) | 2012-07-26 |
| MX2012003994A (es) | 2012-04-30 |
| CA2774031A1 (en) | 2011-04-14 |
| AU2010305355B2 (en) | 2015-09-24 |
| CN102548996A (zh) | 2012-07-04 |
| AU2010305355A1 (en) | 2012-04-05 |
| EP2486040B1 (en) | 2017-06-21 |
| JP5870031B2 (ja) | 2016-02-24 |
| KR20120095359A (ko) | 2012-08-28 |
| IN2012DN02214A (enExample) | 2015-08-21 |
| CN102548996B (zh) | 2016-06-01 |
| IL218454A0 (en) | 2012-04-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 6A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2384 DE 13-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |