BR0313161A - Composto, composição farmacêutica, e, uso de uma quantidade eficaz de hemiidrato de (r)-(6-(1-((4-fluorobenzil)metilamino]etilidenoamino)-2 (r)-hidroxiindan-1-il) amida do ácido bifenil-4-carboxìlico - Google Patents

Composto, composição farmacêutica, e, uso de uma quantidade eficaz de hemiidrato de (r)-(6-(1-((4-fluorobenzil)metilamino]etilidenoamino)-2 (r)-hidroxiindan-1-il) amida do ácido bifenil-4-carboxìlico

Info

Publication number
BR0313161A
BR0313161A BR0313161-0A BR0313161A BR0313161A BR 0313161 A BR0313161 A BR 0313161A BR 0313161 A BR0313161 A BR 0313161A BR 0313161 A BR0313161 A BR 0313161A
Authority
BR
Brazil
Prior art keywords
fluorobenzyl
biphenyl
ethylidenoamino
hydroxyindan
methylamino
Prior art date
Application number
BR0313161-0A
Other languages
English (en)
Portuguese (pt)
Inventor
Julie Kay Bush
Perry Clark Heath
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of BR0313161A publication Critical patent/BR0313161A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C257/00Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines
    • C07C257/10Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines
    • C07C257/14Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines having carbon atoms of amidino groups bound to acyclic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00Systems containing two condensed rings
    • C07C2602/02Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04One of the condensed rings being a six-membered aromatic ring
    • C07C2602/08One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BR0313161-0A 2002-08-22 2003-08-12 Composto, composição farmacêutica, e, uso de uma quantidade eficaz de hemiidrato de (r)-(6-(1-((4-fluorobenzil)metilamino]etilidenoamino)-2 (r)-hidroxiindan-1-il) amida do ácido bifenil-4-carboxìlico BR0313161A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40544302P 2002-08-22 2002-08-22
PCT/US2003/023260 WO2004018411A1 (en) 2002-08-22 2003-08-12 Muscarinic agonists

Publications (1)

Publication Number Publication Date
BR0313161A true BR0313161A (pt) 2005-06-14

Family

ID=31946873

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0313161-0A BR0313161A (pt) 2002-08-22 2003-08-12 Composto, composição farmacêutica, e, uso de uma quantidade eficaz de hemiidrato de (r)-(6-(1-((4-fluorobenzil)metilamino]etilidenoamino)-2 (r)-hidroxiindan-1-il) amida do ácido bifenil-4-carboxìlico

Country Status (19)

Country Link
US (1) US7160922B2 (https=)
EP (1) EP1534667B1 (https=)
JP (1) JP4469280B2 (https=)
CN (1) CN100554247C (https=)
AR (1) AR040889A1 (https=)
AT (1) ATE491683T1 (https=)
AU (1) AU2003256791B2 (https=)
BR (1) BR0313161A (https=)
CA (1) CA2493958C (https=)
CY (1) CY1111115T1 (https=)
DE (1) DE60335380D1 (https=)
DK (1) DK1534667T3 (https=)
ES (1) ES2355213T3 (https=)
MX (1) MXPA05002080A (https=)
PE (1) PE20040894A1 (https=)
PT (1) PT1534667E (https=)
SI (1) SI1534667T1 (https=)
TW (1) TW200410922A (https=)
WO (1) WO2004018411A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2275095A3 (en) * 2005-08-26 2011-08-17 Braincells, Inc. Neurogenesis by muscarinic receptor modulation
JP2013523679A (ja) 2010-03-29 2013-06-17 ビーエーエスエフ ソシエタス・ヨーロピア 殺菌性イミノ誘導体

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA76492C2 (en) * 2001-09-21 2006-08-15 Lilly Co Eli Muscarinic agonists, a pharmaceutical composition on their basis

Also Published As

Publication number Publication date
CA2493958A1 (en) 2004-03-04
WO2004018411A1 (en) 2004-03-04
CN1675173A (zh) 2005-09-28
ES2355213T3 (es) 2011-03-23
CY1111115T1 (el) 2015-06-11
JP2005536549A (ja) 2005-12-02
MXPA05002080A (es) 2005-08-18
PE20040894A1 (es) 2004-11-25
CN100554247C (zh) 2009-10-28
AR040889A1 (es) 2005-04-20
DK1534667T3 (da) 2011-02-14
DE60335380D1 (de) 2011-01-27
US7160922B2 (en) 2007-01-09
TW200410922A (en) 2004-07-01
EP1534667B1 (en) 2010-12-15
JP4469280B2 (ja) 2010-05-26
EP1534667A1 (en) 2005-06-01
AU2003256791A1 (en) 2004-03-11
ATE491683T1 (de) 2011-01-15
AU2003256791B2 (en) 2008-12-11
US20060122280A1 (en) 2006-06-08
CA2493958C (en) 2010-11-09
SI1534667T1 (sl) 2011-02-28
PT1534667E (pt) 2011-01-19

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Legal Events

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B15I Others concerning applications: loss of priority

Free format text: PERDA DA PRIORIDADE REIVINDICADA (US 60/405,443), POR NAO ESTAR EM CONFORMIDADE COM O PREVISTO NOS 6O E 7O DO ART.16 DA LPI/96.

B150 Others concerning applications: publication cancelled [chapter 15.30 patent gazette]

Free format text: ANULADO O DESPACHO (15.9) DA RPI 2017, POR TER SIDO REALIZADO INDEVIDAMENTE.

B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 11A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2266 DE 10/06/2014.