BR0309930A - Derivados do ácido dihidroxihexanóico, seus intermediários e métodos de produção - Google Patents

Derivados do ácido dihidroxihexanóico, seus intermediários e métodos de produção

Info

Publication number
BR0309930A
BR0309930A BR0309930-0A BR0309930A BR0309930A BR 0309930 A BR0309930 A BR 0309930A BR 0309930 A BR0309930 A BR 0309930A BR 0309930 A BR0309930 A BR 0309930A
Authority
BR
Brazil
Prior art keywords
acid derivatives
intermediates
production methods
dihydroxyhexanoic acid
dihydroxyhexanoic
Prior art date
Application number
BR0309930-0A
Other languages
English (en)
Inventor
Frank John Urban
Vytautas John Jasys
Zhengong Bryan Li
John Charles Kath
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of BR0309930A publication Critical patent/BR0309930A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/26Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D307/30Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/32Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/26Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D307/30Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/32Oxygen atoms
    • C07D307/33Oxygen atoms in position 2, the oxygen atom being in its keto or unsubstituted enol form
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/36Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
    • C07D241/38Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
    • C07D241/40Benzopyrazines
    • C07D241/44Benzopyrazines with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Abstract

"DERIVADOS DO áCIDO DIHIDROXIHEXANóICO, SEUS INTERMEDIáRIOS E MéTODOS DE PRODUçãO". A presente invenção refere-se a derivados do ácido dihidroxihexanóico e seus intermediários, assim como métodos para preparação destes compostos. Adicionalmente, a presente invenção refere-se a remoção de um grupo protetor a partir de uma amina protegida onde o método compreende a reação de uma amina protegida com ácido fosfórico.
BR0309930-0A 2002-05-14 2003-05-05 Derivados do ácido dihidroxihexanóico, seus intermediários e métodos de produção BR0309930A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38069402P 2002-05-14 2002-05-14
US39713802P 2002-07-18 2002-07-18
PCT/IB2003/001840 WO2003095440A1 (en) 2002-05-14 2003-05-05 Dihydroxyhexanoic acid derivatives, their intermediates, and methods of making

Publications (1)

Publication Number Publication Date
BR0309930A true BR0309930A (pt) 2005-02-09

Family

ID=29423736

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0309930-0A BR0309930A (pt) 2002-05-14 2003-05-05 Derivados do ácido dihidroxihexanóico, seus intermediários e métodos de produção

Country Status (14)

Country Link
US (1) US6858744B2 (pt)
EP (1) EP1503999A1 (pt)
JP (1) JP2005530775A (pt)
KR (1) KR20050006256A (pt)
CN (1) CN1653056A (pt)
AR (1) AR039539A1 (pt)
AU (1) AU2003223052A1 (pt)
BR (1) BR0309930A (pt)
CA (1) CA2484860A1 (pt)
IL (1) IL164929A0 (pt)
PL (1) PL373961A1 (pt)
RU (1) RU2004133530A (pt)
TW (1) TW200306175A (pt)
WO (1) WO2003095440A1 (pt)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE640616A (pt) * 1962-12-19
US3492397A (en) * 1967-04-07 1970-01-27 Warner Lambert Pharmaceutical Sustained release dosage in the pellet form and process thereof
US4060598A (en) * 1967-06-28 1977-11-29 Boehringer Mannheim G.M.B.H. Tablets coated with aqueous resin dispersions
US3538214A (en) * 1969-04-22 1970-11-03 Merck & Co Inc Controlled release medicinal tablets
US4173626A (en) * 1978-12-11 1979-11-06 Merck & Co., Inc. Sustained release indomethacin
TR199902056T2 (xx) * 1997-02-26 2000-01-21 Pfizer Inc. Heteroaril-Heksanoik asit amid t�revleri.
BR9907655A (pt) * 1998-02-05 2000-10-24 Pfizer Prod Inc Derivados de ácido di-hidróxi-hexanóico

Also Published As

Publication number Publication date
CN1653056A (zh) 2005-08-10
US6858744B2 (en) 2005-02-22
EP1503999A1 (en) 2005-02-09
KR20050006256A (ko) 2005-01-15
PL373961A1 (en) 2005-09-19
CA2484860A1 (en) 2003-11-20
TW200306175A (en) 2003-11-16
RU2004133530A (ru) 2005-06-10
AU2003223052A1 (en) 2003-11-11
JP2005530775A (ja) 2005-10-13
IL164929A0 (en) 2005-12-18
AR039539A1 (es) 2005-02-23
WO2003095440A1 (en) 2003-11-20
US20040019217A1 (en) 2004-01-29

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]