BR0112915A - Composição farmacêutica compreendendo metformina e um derivado do tipo 5-fenoxialquil-2,4-tiazolidinadiona - Google Patents

Composição farmacêutica compreendendo metformina e um derivado do tipo 5-fenoxialquil-2,4-tiazolidinadiona

Info

Publication number
BR0112915A
BR0112915A BR0112915-5A BR0112915A BR0112915A BR 0112915 A BR0112915 A BR 0112915A BR 0112915 A BR0112915 A BR 0112915A BR 0112915 A BR0112915 A BR 0112915A
Authority
BR
Brazil
Prior art keywords
phenoxyalkyl
pharmaceutical composition
metformin
thiazolidinedione derivative
type
Prior art date
Application number
BR0112915-5A
Other languages
English (en)
Inventor
Gerard Moinet
Gerard Botton
Didier Mesangeau
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of BR0112915A publication Critical patent/BR0112915A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12Antidiuretics, e.g. drugs for diabetes insipidus

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

"COMPOSIçãO FARMACêUTICA COMPREENDENDO METFORMINA E UM DERIVADO DO TIPO 5-FENOXIALQUIL-2,4-TIAZOLIDINADIONA". A presente invenção refere-se a uma composição farmacêutica compreendendo, como ingredientes ativos, metformina optativamente na forma de seus sais farmaceuticamente aceitáveis e uma derivado do tipo de 5-fenoxialquil-2,4-tiazolidinadiona.
BR0112915-5A 2000-08-04 2001-07-24 Composição farmacêutica compreendendo metformina e um derivado do tipo 5-fenoxialquil-2,4-tiazolidinadiona BR0112915A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0010362A FR2812547B1 (fr) 2000-08-04 2000-08-04 Composition pharmaceutique comprenant une association metformine et derive de thiazolidinedione et son utilisation pour la preparation de medicaments destines a traiter le diabete
PCT/EP2001/008512 WO2002011721A1 (en) 2000-08-04 2001-07-24 Pharmaceutical composition comprising metformin and a 5-phenoxyalkyl-2,4-thiazolidinedione-type derivative

Publications (1)

Publication Number Publication Date
BR0112915A true BR0112915A (pt) 2003-07-08

Family

ID=8853342

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0112915-5A BR0112915A (pt) 2000-08-04 2001-07-24 Composição farmacêutica compreendendo metformina e um derivado do tipo 5-fenoxialquil-2,4-tiazolidinadiona

Country Status (19)

Country Link
US (1) US20040014797A1 (pt)
EP (1) EP1305025A1 (pt)
JP (1) JP2004505915A (pt)
KR (1) KR20030019470A (pt)
CN (1) CN1446090A (pt)
AR (1) AR030309A1 (pt)
AU (1) AU2001282010A1 (pt)
BR (1) BR0112915A (pt)
CA (1) CA2417883A1 (pt)
CZ (1) CZ2003476A3 (pt)
EC (1) ECSP034463A (pt)
FR (1) FR2812547B1 (pt)
HU (1) HUP0303684A2 (pt)
MX (1) MXPA03000975A (pt)
NO (1) NO20030518D0 (pt)
PL (1) PL358791A1 (pt)
RU (1) RU2003105809A (pt)
SK (1) SK2082003A3 (pt)
WO (1) WO2002011721A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003105809A1 (en) 2002-06-17 2003-12-24 Themis Laboratories Private Limited Multilayer tablets containing thiazolidinedione and biguanides and methods for producing them
UA80991C2 (en) * 2002-10-07 2007-11-26 Solid preparation containing an insulin resistance improving drug and an active ingredient useful as a remedy for diabetes
WO2008016729A1 (en) * 2006-08-04 2008-02-07 Nastech Pharmaceutical Company Inc. Compositions for intranasal delivery of human insulin and uses thereof
KR100926417B1 (ko) 2007-01-29 2009-11-12 한올제약주식회사 N,n―디메틸 이미도디카르본이미딕 디아미드의 초산염,그의 제조방법 및 그를 포함하는 약제학적 조성물

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2749583B1 (fr) * 1996-06-07 1998-08-21 Lipha Nouveaux derives de thiazolidine -2,4- dione substitues, leurs procedes d'obtention et les compositions pharmaceutiques en renfermant
KR20060105005A (ko) * 1997-06-18 2006-10-09 스미스클라인비이참피이엘시이 티아졸리딘디온 및 메트포르민을 사용한 당뇨병의 치료
GB9715295D0 (en) * 1997-07-18 1997-09-24 Smithkline Beecham Plc Novel method of treatment

Also Published As

Publication number Publication date
KR20030019470A (ko) 2003-03-06
NO20030518L (no) 2003-02-03
SK2082003A3 (en) 2003-07-01
JP2004505915A (ja) 2004-02-26
FR2812547B1 (fr) 2002-10-31
CZ2003476A3 (cs) 2003-06-18
EP1305025A1 (en) 2003-05-02
AU2001282010A1 (en) 2002-02-18
FR2812547A1 (fr) 2002-02-08
AR030309A1 (es) 2003-08-20
PL358791A1 (en) 2004-08-23
HUP0303684A2 (hu) 2004-03-01
CA2417883A1 (en) 2002-02-14
RU2003105809A (ru) 2004-08-27
WO2002011721A1 (en) 2002-02-14
ECSP034463A (es) 2003-03-31
MXPA03000975A (es) 2003-06-09
CN1446090A (zh) 2003-10-01
NO20030518D0 (no) 2003-02-03
US20040014797A1 (en) 2004-01-22

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]