BR0111531A - Nucleosìdeos de pirido[2,3-d]pirimidina e pirimido[4,5-d]pirimidina - Google Patents

Nucleosìdeos de pirido[2,3-d]pirimidina e pirimido[4,5-d]pirimidina

Info

Publication number
BR0111531A
BR0111531A BR0111531-6A BR0111531A BR0111531A BR 0111531 A BR0111531 A BR 0111531A BR 0111531 A BR0111531 A BR 0111531A BR 0111531 A BR0111531 A BR 0111531A
Authority
BR
Brazil
Prior art keywords
pyrimidine
pyrimido
pyrido
nucleosides
purine nucleoside
Prior art date
Application number
BR0111531-6A
Other languages
English (en)
Portuguese (pt)
Inventor
Guangyi Wang
Jean-Luc Girardet
Esmir Gunic
Johnson Lau
Zbigniew Pietrzkoeski
Zhi Hong
Original Assignee
Ribapharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ribapharm Inc filed Critical Ribapharm Inc
Publication of BR0111531A publication Critical patent/BR0111531A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BR0111531-6A 2000-07-06 2001-07-03 Nucleosìdeos de pirido[2,3-d]pirimidina e pirimido[4,5-d]pirimidina BR0111531A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US21641800P 2000-07-06 2000-07-06
PCT/US2001/041242 WO2002003997A1 (en) 2000-07-06 2001-07-03 Pyrido[2,3-d]pyrimidine and pyrimido[4,5-d]pyrimidine nucleosides

Publications (1)

Publication Number Publication Date
BR0111531A true BR0111531A (pt) 2004-07-06

Family

ID=22806989

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0111531-6A BR0111531A (pt) 2000-07-06 2001-07-03 Nucleosìdeos de pirido[2,3-d]pirimidina e pirimido[4,5-d]pirimidina

Country Status (19)

Country Link
US (1) US7081449B2 (https=)
EP (1) EP1303282A4 (https=)
JP (1) JP2004522694A (https=)
KR (1) KR20030032944A (https=)
CN (1) CN1440292A (https=)
AU (2) AU2001273670B2 (https=)
BR (1) BR0111531A (https=)
CA (1) CA2405798A1 (https=)
CZ (1) CZ20024052A3 (https=)
HU (1) HUP0301614A3 (https=)
IL (1) IL151849A0 (https=)
MX (1) MXPA02012156A (https=)
NO (1) NO20030033L (https=)
NZ (1) NZ521457A (https=)
PL (1) PL359559A1 (https=)
SK (1) SK112003A3 (https=)
UA (1) UA72612C2 (https=)
WO (1) WO2002003997A1 (https=)
ZA (1) ZA200208010B (https=)

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Also Published As

Publication number Publication date
NO20030033D0 (no) 2003-01-03
NO20030033L (no) 2003-01-03
CA2405798A1 (en) 2002-01-17
CZ20024052A3 (cs) 2003-03-12
AU7367001A (en) 2002-01-21
SK112003A3 (en) 2003-04-01
HUP0301614A3 (en) 2005-02-28
PL359559A1 (en) 2004-08-23
AU2001273670B2 (en) 2005-07-14
WO2002003997A1 (en) 2002-01-17
MXPA02012156A (es) 2004-08-19
NZ521457A (en) 2005-03-24
ZA200208010B (en) 2004-04-28
EP1303282A4 (en) 2004-04-07
JP2004522694A (ja) 2004-07-29
KR20030032944A (ko) 2003-04-26
IL151849A0 (en) 2003-04-10
EP1303282A1 (en) 2003-04-23
HUP0301614A2 (hu) 2003-09-29
UA72612C2 (en) 2005-03-15
US20030144502A1 (en) 2003-07-31
CN1440292A (zh) 2003-09-03
US7081449B2 (en) 2006-07-25

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Legal Events

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B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 5A, 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO PUBLICADO NA RPI 1963 DE 19.08.2008.