BR0110641A - Determinados carbonatos e éteres caprolactâmicos substituìdos, composições farmacêuticas contendo os mesmos e seu uso no tratamento de tumores - Google Patents

Determinados carbonatos e éteres caprolactâmicos substituìdos, composições farmacêuticas contendo os mesmos e seu uso no tratamento de tumores

Info

Publication number
BR0110641A
BR0110641A BR0110641-4A BR0110641A BR0110641A BR 0110641 A BR0110641 A BR 0110641A BR 0110641 A BR0110641 A BR 0110641A BR 0110641 A BR0110641 A BR 0110641A
Authority
BR
Brazil
Prior art keywords
pharmaceutical compositions
compositions containing
tumors
caprolactamic
carbonates
Prior art date
Application number
BR0110641-4A
Other languages
English (en)
Inventor
Frederick Ray Kinder Jr
Richard William Versace
Kenneth Walter Bair
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR0110641A publication Critical patent/BR0110641A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/02Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D223/06Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D223/12Nitrogen atoms not forming part of a nitro radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)

Abstract

"DETERMINADOS CARBONATOS E éTERES CAPROLACTâMICOS SUBSTITUìDOS, COMPOSIçõES FARMACêUTICAS CONTENDO OS MESMOS E SEU USO NO TRATAMENTO DE TUMORES". A presente invenção refere-se a certos compostos de carbonato e éter caprolactâmicos substituídos, a composições farmacêuticas que contêm os ditos compostos, ao uso dos ditos compostos no tratamento de tumores e a um processo para a produção dos ditos compostos.
BR0110641-4A 2000-05-11 2001-05-09 Determinados carbonatos e éteres caprolactâmicos substituìdos, composições farmacêuticas contendo os mesmos e seu uso no tratamento de tumores BR0110641A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US56866700A 2000-05-11 2000-05-11
PCT/EP2001/005263 WO2001085697A1 (en) 2000-05-11 2001-05-09 Substituted caprolactam carbonates and ethers and their use as anti-tumor agents

Publications (1)

Publication Number Publication Date
BR0110641A true BR0110641A (pt) 2003-03-18

Family

ID=24272224

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0110641-4A BR0110641A (pt) 2000-05-11 2001-05-09 Determinados carbonatos e éteres caprolactâmicos substituìdos, composições farmacêuticas contendo os mesmos e seu uso no tratamento de tumores

Country Status (11)

Country Link
EP (1) EP1282604B1 (pt)
JP (1) JP2003532711A (pt)
CN (1) CN1191237C (pt)
AT (1) ATE383341T1 (pt)
AU (1) AU2001295206A1 (pt)
BR (1) BR0110641A (pt)
CA (1) CA2405892C (pt)
DE (1) DE60132324T2 (pt)
ES (1) ES2299515T3 (pt)
PT (1) PT1282604E (pt)
WO (1) WO2001085697A1 (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2006528611A (ja) * 2003-07-25 2006-12-21 ノバルティス アクチエンゲゼルシャフト 置換ラクタムおよびそれらの抗がん剤としての使用
US7153846B2 (en) 2003-10-24 2006-12-26 Sanofi-Aventis Deutschland Gmbh Bengamide derivatives, process for preparing them, and their use
DE10349669B3 (de) * 2003-10-24 2005-05-25 Aventis Pharma Deutschland Gmbh Bengamide-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung
FR2878525B1 (fr) 2004-11-29 2007-02-23 Aventis Pharma Sa Bengamides possedant un cycle caprolactame substitue, procede de preparation, compositions les contenant et utilisation
FR2878528B1 (fr) * 2004-11-29 2008-05-16 Aventis Pharma Sa 2-alcoxy-3,4,5-trihydroxy-alkylamides, leur preparation, compositions les contenant et utilisation
FR2901556A1 (fr) 2006-05-24 2007-11-30 Sanofi Aventis Sa Derives de 2-alcoxy-3,4,5-trihydroxy-alkylamide, leur preparation, compositions les contenant et utilisation
FR2901555A1 (fr) * 2006-05-24 2007-11-30 Sanofi Aventis Sa 2-alcoxy-3,4,5-trihydroxy-alkylamide-benzothiazepine, leur preparation, compositions les contenant et utilisation
FR2901554B1 (fr) 2006-05-24 2011-04-01 Sanofi Aventis 2-alcoxy-3,4,5-trihydroxy-alkylamide-benzazepine, leur preparation, compositions les contenant et utilisation

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4831135A (en) * 1986-06-18 1989-05-16 The Regents Of The University Of California Bengamide anthelmintics
GB9411841D0 (en) * 1994-06-14 1994-08-03 Pharma Mar Sa New antitumoral compounds from jaspis sponge
CO5140099A1 (es) * 1998-11-17 2002-03-22 Novartis Ag Ciertas caprolactamas sustituidas, composiciones farmaceuticas que las contienen, y su uso en el tratamiento de tumores

Also Published As

Publication number Publication date
PT1282604E (pt) 2008-04-11
DE60132324D1 (de) 2008-02-21
ES2299515T3 (es) 2008-06-01
CA2405892A1 (en) 2001-11-15
CN1191237C (zh) 2005-03-02
DE60132324T2 (de) 2008-12-24
EP1282604A1 (en) 2003-02-12
EP1282604B1 (en) 2008-01-09
CN1429213A (zh) 2003-07-09
ATE383341T1 (de) 2008-01-15
JP2003532711A (ja) 2003-11-05
CA2405892C (en) 2009-07-07
WO2001085697A1 (en) 2001-11-15
AU2001295206A1 (en) 2001-11-20

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

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