BR0110641A - Determinados carbonatos e éteres caprolactâmicos substituìdos, composições farmacêuticas contendo os mesmos e seu uso no tratamento de tumores - Google Patents
Determinados carbonatos e éteres caprolactâmicos substituìdos, composições farmacêuticas contendo os mesmos e seu uso no tratamento de tumoresInfo
- Publication number
- BR0110641A BR0110641A BR0110641-4A BR0110641A BR0110641A BR 0110641 A BR0110641 A BR 0110641A BR 0110641 A BR0110641 A BR 0110641A BR 0110641 A BR0110641 A BR 0110641A
- Authority
- BR
- Brazil
- Prior art keywords
- pharmaceutical compositions
- compositions containing
- tumors
- caprolactamic
- carbonates
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D223/12—Nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
Abstract
"DETERMINADOS CARBONATOS E éTERES CAPROLACTâMICOS SUBSTITUìDOS, COMPOSIçõES FARMACêUTICAS CONTENDO OS MESMOS E SEU USO NO TRATAMENTO DE TUMORES". A presente invenção refere-se a certos compostos de carbonato e éter caprolactâmicos substituídos, a composições farmacêuticas que contêm os ditos compostos, ao uso dos ditos compostos no tratamento de tumores e a um processo para a produção dos ditos compostos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US56866700A | 2000-05-11 | 2000-05-11 | |
PCT/EP2001/005263 WO2001085697A1 (en) | 2000-05-11 | 2001-05-09 | Substituted caprolactam carbonates and ethers and their use as anti-tumor agents |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0110641A true BR0110641A (pt) | 2003-03-18 |
Family
ID=24272224
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0110641-4A BR0110641A (pt) | 2000-05-11 | 2001-05-09 | Determinados carbonatos e éteres caprolactâmicos substituìdos, composições farmacêuticas contendo os mesmos e seu uso no tratamento de tumores |
Country Status (11)
Country | Link |
---|---|
EP (1) | EP1282604B1 (pt) |
JP (1) | JP2003532711A (pt) |
CN (1) | CN1191237C (pt) |
AT (1) | ATE383341T1 (pt) |
AU (1) | AU2001295206A1 (pt) |
BR (1) | BR0110641A (pt) |
CA (1) | CA2405892C (pt) |
DE (1) | DE60132324T2 (pt) |
ES (1) | ES2299515T3 (pt) |
PT (1) | PT1282604E (pt) |
WO (1) | WO2001085697A1 (pt) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2006528611A (ja) * | 2003-07-25 | 2006-12-21 | ノバルティス アクチエンゲゼルシャフト | 置換ラクタムおよびそれらの抗がん剤としての使用 |
US7153846B2 (en) | 2003-10-24 | 2006-12-26 | Sanofi-Aventis Deutschland Gmbh | Bengamide derivatives, process for preparing them, and their use |
DE10349669B3 (de) * | 2003-10-24 | 2005-05-25 | Aventis Pharma Deutschland Gmbh | Bengamide-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung |
FR2878525B1 (fr) | 2004-11-29 | 2007-02-23 | Aventis Pharma Sa | Bengamides possedant un cycle caprolactame substitue, procede de preparation, compositions les contenant et utilisation |
FR2878528B1 (fr) * | 2004-11-29 | 2008-05-16 | Aventis Pharma Sa | 2-alcoxy-3,4,5-trihydroxy-alkylamides, leur preparation, compositions les contenant et utilisation |
FR2901556A1 (fr) | 2006-05-24 | 2007-11-30 | Sanofi Aventis Sa | Derives de 2-alcoxy-3,4,5-trihydroxy-alkylamide, leur preparation, compositions les contenant et utilisation |
FR2901555A1 (fr) * | 2006-05-24 | 2007-11-30 | Sanofi Aventis Sa | 2-alcoxy-3,4,5-trihydroxy-alkylamide-benzothiazepine, leur preparation, compositions les contenant et utilisation |
FR2901554B1 (fr) | 2006-05-24 | 2011-04-01 | Sanofi Aventis | 2-alcoxy-3,4,5-trihydroxy-alkylamide-benzazepine, leur preparation, compositions les contenant et utilisation |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4831135A (en) * | 1986-06-18 | 1989-05-16 | The Regents Of The University Of California | Bengamide anthelmintics |
GB9411841D0 (en) * | 1994-06-14 | 1994-08-03 | Pharma Mar Sa | New antitumoral compounds from jaspis sponge |
CO5140099A1 (es) * | 1998-11-17 | 2002-03-22 | Novartis Ag | Ciertas caprolactamas sustituidas, composiciones farmaceuticas que las contienen, y su uso en el tratamiento de tumores |
-
2001
- 2001-05-09 BR BR0110641-4A patent/BR0110641A/pt not_active Application Discontinuation
- 2001-05-09 AU AU2001295206A patent/AU2001295206A1/en not_active Abandoned
- 2001-05-09 CN CNB018093078A patent/CN1191237C/zh not_active Expired - Fee Related
- 2001-05-09 CA CA002405892A patent/CA2405892C/en not_active Expired - Fee Related
- 2001-05-09 PT PT01975824T patent/PT1282604E/pt unknown
- 2001-05-09 ES ES01975824T patent/ES2299515T3/es not_active Expired - Lifetime
- 2001-05-09 DE DE60132324T patent/DE60132324T2/de not_active Expired - Lifetime
- 2001-05-09 JP JP2001582298A patent/JP2003532711A/ja active Pending
- 2001-05-09 EP EP01975824A patent/EP1282604B1/en not_active Expired - Lifetime
- 2001-05-09 WO PCT/EP2001/005263 patent/WO2001085697A1/en active IP Right Grant
- 2001-05-09 AT AT01975824T patent/ATE383341T1/de not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
PT1282604E (pt) | 2008-04-11 |
DE60132324D1 (de) | 2008-02-21 |
ES2299515T3 (es) | 2008-06-01 |
CA2405892A1 (en) | 2001-11-15 |
CN1191237C (zh) | 2005-03-02 |
DE60132324T2 (de) | 2008-12-24 |
EP1282604A1 (en) | 2003-02-12 |
EP1282604B1 (en) | 2008-01-09 |
CN1429213A (zh) | 2003-07-09 |
ATE383341T1 (de) | 2008-01-15 |
JP2003532711A (ja) | 2003-11-05 |
CA2405892C (en) | 2009-07-07 |
WO2001085697A1 (en) | 2001-11-15 |
AU2001295206A1 (en) | 2001-11-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL. |