BG62003B1 - Производни на 1-(2-флуороциклопропил)-хинолон- инафтиридон- карбонови киселини - Google Patents

Производни на 1-(2-флуороциклопропил)-хинолон- инафтиридон- карбонови киселини Download PDF

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Publication number
BG62003B1
BG62003B1 BG99179A BG9917994A BG62003B1 BG 62003 B1 BG62003 B1 BG 62003B1 BG 99179 A BG99179 A BG 99179A BG 9917994 A BG9917994 A BG 9917994A BG 62003 B1 BG62003 B1 BG 62003B1
Authority
BG
Bulgaria
Prior art keywords
oxo
dihydro
fluorocyclopropyl
acid
quinolinecarboxylic acid
Prior art date
Application number
BG99179A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG99179A (en
Inventor
Uwe Petersen
Thomas Schenke
Stefan Boehm
Rolf Grosser
Klaus Bremm
Rainer Endermann
Karl Metzger
Original Assignee
Bayer Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft
Publication of BG99179A publication Critical patent/BG99179A/bg
Publication of BG62003B1 publication Critical patent/BG62003B1/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
BG99179A 1993-11-16 1994-11-14 Производни на 1-(2-флуороциклопропил)-хинолон- инафтиридон- карбонови киселини BG62003B1 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4339134A DE4339134A1 (de) 1993-11-16 1993-11-16 1-(2-Fluorcyclopropyl)-chinolon- und -naphthyridoncarbonsäure-Derivate

Publications (2)

Publication Number Publication Date
BG99179A BG99179A (en) 1995-07-28
BG62003B1 true BG62003B1 (bg) 1998-12-30

Family

ID=6502741

Family Applications (1)

Application Number Title Priority Date Filing Date
BG99179A BG62003B1 (bg) 1993-11-16 1994-11-14 Производни на 1-(2-флуороциклопропил)-хинолон- инафтиридон- карбонови киселини

Country Status (27)

Country Link
US (1) US5545642A (no)
EP (1) EP0653425A1 (no)
JP (1) JPH07188230A (no)
KR (1) KR950014114A (no)
CN (1) CN1106412A (no)
AU (2) AU681703B2 (no)
BG (1) BG62003B1 (no)
CA (1) CA2135548A1 (no)
CO (1) CO4180605A1 (no)
CZ (1) CZ280594A3 (no)
DE (1) DE4339134A1 (no)
EE (1) EE9400240A (no)
FI (1) FI945360A (no)
HR (1) HRP940833A2 (no)
HU (1) HUT70175A (no)
IL (1) IL111624A0 (no)
LV (1) LV11328B (no)
NO (1) NO302367B1 (no)
NZ (1) NZ264905A (no)
PE (1) PE32395A1 (no)
PL (1) PL305862A1 (no)
RU (1) RU94040885A (no)
SK (1) SK137194A3 (no)
SV (1) SV1994000064A (no)
TW (1) TW273547B (no)
YU (1) YU65494A (no)
ZA (1) ZA949052B (no)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0664288A1 (en) * 1992-10-09 1995-07-26 Chugai Seiyaku Kabushiki Kaisha Fluoroquinoline derivative
JP3468244B2 (ja) * 1995-12-22 2003-11-17 ナガセケムテックス株式会社 抗ヘリコバクターピロリ剤
WO1998058928A1 (fr) * 1997-06-23 1998-12-30 Yoshitomi Pharmaceutical Industries, Ltd. Agent prophylactique ou therapeutique contre des maladies attribuables a une infection par des helicobacters
DE10108750A1 (de) 2001-02-23 2002-09-05 Bayer Ag Verbessertes Verfahren zur Herstellung von Fluorchinoloncarbonsäuren
JP4675234B2 (ja) * 2003-06-06 2011-04-20 第一三共株式会社 光学活性なキノロンカルボン酸誘導体の製造中間体およびその製造法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5274167A (en) * 1989-01-26 1993-12-28 Bayer Aktiengesellschaft Polymeriable optically active (meth) acrylic acid derivatives
DE3910663A1 (de) * 1989-04-03 1990-10-04 Bayer Ag 5-alkylchinoloncarbonsaeuren
KR910009330B1 (ko) * 1989-10-23 1991-11-11 재단법인 한국화학연구소 항균작용을 갖는 퀴놀린계 화합물과 그의 제조방법
KR910009331B1 (ko) * 1989-10-23 1991-11-11 재단법인 한국화학연구소 디아자비시클로아민 화합물과 그의 제조방법
KR910009333B1 (ko) * 1989-10-23 1991-11-11 재단법인 한국화학연구소 항균작용을 갖는 퀴놀린계 화합물과 그의 제조방법
DE69231422T2 (de) * 1991-05-28 2001-03-29 Daiichi Pharmaceutical Co., Ltd. Pyridoncarbonsäurederivate
DE4121214A1 (de) * 1991-06-27 1993-01-14 Bayer Ag 7-azaisoindolinyl-chinolon- und -naphthyridoncarbonsaeure-derivate
EP0550016A1 (en) * 1991-12-31 1993-07-07 Korea Research Institute Of Chemical Technology Novel quinolone carboxylic acid derivatives and processes for preparing same
AU4272793A (en) * 1993-04-24 1994-11-21 Korea Research Institute Of Chemical Technology Novel quinolone carboxylic acid derivatives and process for preparing the same

Also Published As

Publication number Publication date
CZ280594A3 (en) 1995-08-16
JPH07188230A (ja) 1995-07-25
HU9403288D0 (en) 1995-01-30
LV11328B (en) 1996-12-20
US5545642A (en) 1996-08-13
HUT70175A (en) 1995-09-28
IL111624A0 (en) 1995-01-24
SK137194A3 (en) 1995-06-07
RU94040885A (ru) 1996-11-20
KR950014114A (ko) 1995-06-15
AU2559997A (en) 1997-09-04
CA2135548A1 (en) 1995-05-17
FI945360A (fi) 1995-05-17
NO944365D0 (no) 1994-11-15
NO944365L (no) 1995-05-18
FI945360A0 (fi) 1994-11-14
NZ264905A (en) 1995-11-27
AU681703B2 (en) 1997-09-04
CO4180605A1 (es) 1995-06-07
NO302367B1 (no) 1998-02-23
BG99179A (en) 1995-07-28
AU7773094A (en) 1995-05-25
EP0653425A1 (de) 1995-05-17
TW273547B (no) 1996-04-01
LV11328A (lv) 1996-06-20
EE9400240A (et) 1996-02-15
PE32395A1 (es) 1995-12-15
SV1994000064A (es) 1995-05-25
HRP940833A2 (en) 1996-12-31
CN1106412A (zh) 1995-08-09
ZA949052B (en) 1995-07-19
PL305862A1 (en) 1995-05-29
DE4339134A1 (de) 1995-05-18
YU65494A (sh) 1997-09-30

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