BG26531A4 - Метод за получаване на бензоксазолови производни - Google Patents

Метод за получаване на бензоксазолови производни

Info

Publication number
BG26531A4
BG26531A4 BG032026A BG3202674A BG26531A4 BG 26531 A4 BG26531 A4 BG 26531A4 BG 032026 A BG032026 A BG 032026A BG 3202674 A BG3202674 A BG 3202674A BG 26531 A4 BG26531 A4 BG 26531A4
Authority
BG
Bulgaria
Prior art keywords
obtaining
benzoxazole derivatives
benzoxazole
derivatives
obtaining benzoxazole
Prior art date
Application number
BG032026A
Other languages
Bulgarian (bg)
English (en)
Inventor
John Saunders
William Williamson
Original Assignee
Неизвестен
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Неизвестен filed Critical Неизвестен
Publication of BG26531A4 publication Critical patent/BG26531A4/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D263/57Aryl or substituted aryl radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46Friedel-Crafts reactions
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BG032026A 1973-10-23 1974-10-23 Метод за получаване на бензоксазолови производни BG26531A4 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB49259/73A GB1488003A (en) 1973-10-23 1973-10-23 1,2-benzisoxazole derivatives processes for their preparation and their use as pharmaceuticals

Publications (1)

Publication Number Publication Date
BG26531A4 true BG26531A4 (bg) 1979-04-12

Family

ID=10451720

Family Applications (2)

Application Number Title Priority Date Filing Date
BG032026A BG26531A4 (bg) 1973-10-23 1974-10-23 Метод за получаване на бензоксазолови производни
BG028023A BG25991A3 (bg) 1973-10-23 1974-10-23 Метод за получаване на 1,2-бензизоксазолови производни

Family Applications After (1)

Application Number Title Priority Date Filing Date
BG028023A BG25991A3 (bg) 1973-10-23 1974-10-23 Метод за получаване на 1,2-бензизоксазолови производни

Country Status (27)

Country Link
US (1) US3951999A (cs)
JP (2) JPS5912671B2 (cs)
AR (3) AR209755A1 (cs)
AT (1) AT341520B (cs)
AU (1) AU510909B2 (cs)
BE (1) BE821406A (cs)
BG (2) BG26531A4 (cs)
CA (1) CA1042005A (cs)
CH (2) CH605864A5 (cs)
CS (1) CS189671B2 (cs)
DD (1) DD116830A5 (cs)
DE (1) DE2450053A1 (cs)
DK (1) DK552674A (cs)
ES (3) ES431247A1 (cs)
FR (3) FR2248041B1 (cs)
GB (1) GB1488003A (cs)
HU (1) HU171613B (cs)
IE (1) IE40078B1 (cs)
IL (3) IL45880A (cs)
NL (1) NL7413848A (cs)
NZ (1) NZ175780A (cs)
PH (1) PH11022A (cs)
RO (2) RO78465A (cs)
SE (3) SE424324B (cs)
SU (3) SU604491A3 (cs)
YU (1) YU282474A (cs)
ZA (1) ZA746594B (cs)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1590587A (en) * 1977-06-28 1981-06-03 Lilly Industries Ltd Benoxaprofen
US4728662A (en) * 1977-11-21 1988-03-01 Hoechst-Roussel Pharmaceuticals Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4673746A (en) * 1978-10-06 1987-06-16 Hoechst-Roussel Pharmaceuticals, Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
NZ189705A (en) * 1978-03-01 1981-07-13 Boots Co Ltd Benzophenone-hydrazone derivatives and pesticidal compositions intermediates
US4337261A (en) * 1980-07-28 1982-06-29 Hoechst-Roussel Pharmaceuticals Inc. (1,2-Benzisoxazol)phenoxyacetic acids as diuretics
US4894461A (en) * 1981-04-27 1990-01-16 Hoechst-Roussel Pharmaceuticals, Inc. 3-(γ-chloropropyl)-6-fluoro-1,2-benzisoxazole
US4396770A (en) * 1982-04-09 1983-08-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-hydroxy-4-phenylpiperidines
US4536578A (en) * 1982-04-09 1985-08-20 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines
US4374245A (en) * 1982-04-09 1983-02-15 Hoechst-Roussel Pharmaceuticals Inc. 8-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
US4390544A (en) * 1982-04-09 1983-06-28 Hoechst-Roussel Pharmaceuticals Inc. {1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(2-oxo-1-benzimidazolinyl}p
US4610988A (en) * 1982-04-09 1986-09-09 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines useful for alleviating pain
US4609658A (en) * 1982-04-09 1986-09-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted) piperazines useful for reducing blood pressure
US4458075A (en) * 1982-04-09 1984-07-03 Hoechst-Roussel Pharmaceuticals Inc. 6-Fluoro-3-[3-(1-heterocyclo)propyl]-1,2-benzisoxazoles
US4420485A (en) * 1982-09-29 1983-12-13 Hoechst-Roussel Pharmaceuticals Inc. 1'-[3-(1,2-Benzisoxazol-3-yl) proply]spiro[benzofuran-2(3H),3' or 4'-piperidines or 3'-pyrrolidines]
FR2540107B1 (fr) * 1983-01-28 1986-10-17 Inst Rech Chim Biolog Nouveaux derives d'halogenobenzophenone-oxime, utilisation en therapeutique et procede de preparation
FI92189C (fi) * 1986-03-17 1994-10-10 Eisai Co Ltd Menetelmä lääkeaineina käyttökelpoisen difenyylimetaanijohdannaisen valmistamiseksi
US4898874A (en) * 1986-09-15 1990-02-06 A. H. Robins Company, Inc. Acetic acid derivatives of 3-aryl-2,1-benzisoxazole and esters and amides thereof
JPH037961U (cs) * 1989-06-14 1991-01-25
US5114960A (en) * 1989-07-20 1992-05-19 Hoffmann-La Roche Inc. Substituted isoxazole derivatives
PL1986633T3 (pl) * 2006-02-10 2015-01-30 Summit Oxford Ltd Leczenie dystrofii mięśniowej Duchenne'a
EP2755961A1 (en) * 2011-09-16 2014-07-23 Pfizer Inc Solid forms of a transthyretin dissociation inhibitor

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH503463A (de) * 1969-07-17 1971-02-28 Ciba Geigy Ag Verwendung von 2-Hydroxybenzophenonen zur Bekämpfung schädlicher Mikroorganismen ausserhalb der Textilindustrie
FR2093173A5 (en) * 1970-06-04 1972-01-28 Gen Mills Inc Substituted 2-hydroxybenzophenoximes for - copper extraction

Also Published As

Publication number Publication date
AR213086A1 (es) 1978-12-15
AT341520B (de) 1978-02-10
FR2361328B1 (cs) 1979-07-13
FR2361328A1 (fr) 1978-03-10
AU2880177A (en) 1979-03-15
CS189671B2 (en) 1979-04-30
FR2248041B1 (cs) 1978-09-08
IL52179A0 (en) 1977-07-31
SU604491A3 (ru) 1978-04-25
JPS636066B2 (cs) 1988-02-08
FR2248041A1 (cs) 1975-05-16
AU7454774A (en) 1976-04-29
JPS57154174A (en) 1982-09-22
ATA852374A (de) 1977-06-15
NL7413848A (nl) 1975-04-25
IE40078B1 (en) 1979-03-14
YU282474A (en) 1982-02-28
CH595360A5 (cs) 1978-02-15
ZA746594B (en) 1976-06-30
AR209755A1 (es) 1977-05-31
CH605864A5 (cs) 1978-10-13
SE7413237L (cs) 1975-04-24
DK552674A (cs) 1975-06-16
SE7710600L (sv) 1977-09-21
AR221321A1 (es) 1981-01-30
ES449655A1 (es) 1977-07-01
IL45880A (en) 1979-09-30
SU795459A3 (ru) 1981-01-07
JPS5077364A (cs) 1975-06-24
ES449654A1 (es) 1977-07-01
BE821406A (fr) 1975-04-23
RO78465A (ro) 1982-02-26
SE435713B (sv) 1984-10-15
IE40078L (en) 1975-04-23
AU510909B2 (en) 1980-07-17
SU608476A3 (ru) 1978-05-25
GB1488003A (en) 1977-10-05
IL45880A0 (en) 1974-12-31
SE424324B (sv) 1982-07-12
FR2361359B1 (cs) 1979-07-20
BG25991A3 (bg) 1979-01-12
IL52180A0 (en) 1977-07-31
HU171613B (hu) 1978-02-28
NZ175780A (en) 1978-04-03
SE7710599L (sv) 1977-09-21
ES431247A1 (es) 1977-02-16
RO74031A (ro) 1982-02-01
FR2361359A1 (fr) 1978-03-10
JPS5912671B2 (ja) 1984-03-24
US3951999A (en) 1976-04-20
SE424325B (sv) 1982-07-12
DE2450053A1 (de) 1975-04-24
PH11022A (en) 1977-10-25
CA1042005A (en) 1978-11-07
DD116830A5 (cs) 1975-12-12

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