SE424325B - Forfarande for framstellning av 1,2-bensisoxazoler - Google Patents

Forfarande for framstellning av 1,2-bensisoxazoler

Info

Publication number
SE424325B
SE424325B SE7710599A SE7710599A SE424325B SE 424325 B SE424325 B SE 424325B SE 7710599 A SE7710599 A SE 7710599A SE 7710599 A SE7710599 A SE 7710599A SE 424325 B SE424325 B SE 424325B
Authority
SE
Sweden
Prior art keywords
benzisoxazoles
preparing
Prior art date
Application number
SE7710599A
Other languages
English (en)
Swedish (sv)
Other versions
SE7710599L (sv
Inventor
J C Saunders
W R N Williamson
Original Assignee
Lilly Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd
Publication of SE7710599L publication Critical patent/SE7710599L/xx
Publication of SE424325B publication Critical patent/SE424325B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D263/57—Aryl or substituted aryl radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46—Friedel-Crafts reactions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SE7710599A 1973-10-23 1977-09-21 Forfarande for framstellning av 1,2-bensisoxazoler SE424325B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB49259/73A GB1488003A (en) 1973-10-23 1973-10-23 1,2-benzisoxazole derivatives processes for their preparation and their use as pharmaceuticals

Publications (2)

Publication Number Publication Date
SE7710599L SE7710599L (sv) 1977-09-21
SE424325B true SE424325B (sv) 1982-07-12

Family

ID=10451720

Family Applications (3)

Application Number Title Priority Date Filing Date
SE7413237A SE424324B (sv) 1973-10-23 1974-10-21 Analogiforfarande for framstellning av 1,2-benzisoxazolderivat
SE7710600A SE435713B (sv) 1973-10-23 1977-09-21 Forfarande for framstellning av 1,3-bensoxazoler
SE7710599A SE424325B (sv) 1973-10-23 1977-09-21 Forfarande for framstellning av 1,2-bensisoxazoler

Family Applications Before (2)

Application Number Title Priority Date Filing Date
SE7413237A SE424324B (sv) 1973-10-23 1974-10-21 Analogiforfarande for framstellning av 1,2-benzisoxazolderivat
SE7710600A SE435713B (sv) 1973-10-23 1977-09-21 Forfarande for framstellning av 1,3-bensoxazoler

Country Status (27)

Country Link
US (1) US3951999A (xx)
JP (2) JPS5912671B2 (xx)
AR (3) AR209755A1 (xx)
AT (1) AT341520B (xx)
AU (1) AU510909B2 (xx)
BE (1) BE821406A (xx)
BG (2) BG26531A4 (xx)
CA (1) CA1042005A (xx)
CH (2) CH595360A5 (xx)
CS (1) CS189671B2 (xx)
DD (1) DD116830A5 (xx)
DE (1) DE2450053A1 (xx)
DK (1) DK552674A (xx)
ES (3) ES431247A1 (xx)
FR (3) FR2248041B1 (xx)
GB (1) GB1488003A (xx)
HU (1) HU171613B (xx)
IE (1) IE40078B1 (xx)
IL (3) IL45880A (xx)
NL (1) NL7413848A (xx)
NZ (1) NZ175780A (xx)
PH (1) PH11022A (xx)
RO (2) RO78465A (xx)
SE (3) SE424324B (xx)
SU (3) SU604491A3 (xx)
YU (1) YU282474A (xx)
ZA (1) ZA746594B (xx)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1590587A (en) * 1977-06-28 1981-06-03 Lilly Industries Ltd Benoxaprofen
US4728662A (en) * 1977-11-21 1988-03-01 Hoechst-Roussel Pharmaceuticals Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4673746A (en) * 1978-10-06 1987-06-16 Hoechst-Roussel Pharmaceuticals, Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
NZ189705A (en) * 1978-03-01 1981-07-13 Boots Co Ltd Benzophenone-hydrazone derivatives and pesticidal compositions intermediates
US4337261A (en) * 1980-07-28 1982-06-29 Hoechst-Roussel Pharmaceuticals Inc. (1,2-Benzisoxazol)phenoxyacetic acids as diuretics
US4894461A (en) * 1981-04-27 1990-01-16 Hoechst-Roussel Pharmaceuticals, Inc. 3-(γ-chloropropyl)-6-fluoro-1,2-benzisoxazole
US4396770A (en) * 1982-04-09 1983-08-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-hydroxy-4-phenylpiperidines
US4374245A (en) * 1982-04-09 1983-02-15 Hoechst-Roussel Pharmaceuticals Inc. 8-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
US4390544A (en) * 1982-04-09 1983-06-28 Hoechst-Roussel Pharmaceuticals Inc. {1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(2-oxo-1-benzimidazolinyl}p
US4609658A (en) * 1982-04-09 1986-09-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted) piperazines useful for reducing blood pressure
US4536578A (en) * 1982-04-09 1985-08-20 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines
US4610988A (en) * 1982-04-09 1986-09-09 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines useful for alleviating pain
US4458075A (en) * 1982-04-09 1984-07-03 Hoechst-Roussel Pharmaceuticals Inc. 6-Fluoro-3-[3-(1-heterocyclo)propyl]-1,2-benzisoxazoles
US4420485A (en) * 1982-09-29 1983-12-13 Hoechst-Roussel Pharmaceuticals Inc. 1'-[3-(1,2-Benzisoxazol-3-yl) proply]spiro[benzofuran-2(3H),3' or 4'-piperidines or 3'-pyrrolidines]
FR2540107B1 (fr) * 1983-01-28 1986-10-17 Inst Rech Chim Biolog Nouveaux derives d'halogenobenzophenone-oxime, utilisation en therapeutique et procede de preparation
FI92189C (fi) * 1986-03-17 1994-10-10 Eisai Co Ltd Menetelmä lääkeaineina käyttökelpoisen difenyylimetaanijohdannaisen valmistamiseksi
US4898874A (en) * 1986-09-15 1990-02-06 A. H. Robins Company, Inc. Acetic acid derivatives of 3-aryl-2,1-benzisoxazole and esters and amides thereof
JPH037961U (xx) * 1989-06-14 1991-01-25
US5114960A (en) * 1989-07-20 1992-05-19 Hoffmann-La Roche Inc. Substituted isoxazole derivatives
EP1986633B1 (en) * 2006-02-10 2014-07-30 Summit Corporation Plc Treatment of duchenne muscular dystrophy
AU2012310157B2 (en) * 2011-09-16 2015-11-12 Pfizer Inc. Solid forms of a transthyretin dissociation inhibitor

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH503463A (de) * 1969-07-17 1971-02-28 Ciba Geigy Ag Verwendung von 2-Hydroxybenzophenonen zur Bekämpfung schädlicher Mikroorganismen ausserhalb der Textilindustrie
FR2093173A5 (en) * 1970-06-04 1972-01-28 Gen Mills Inc Substituted 2-hydroxybenzophenoximes for - copper extraction

Also Published As

Publication number Publication date
AR209755A1 (es) 1977-05-31
FR2361359B1 (xx) 1979-07-20
CH605864A5 (xx) 1978-10-13
IE40078L (en) 1975-04-23
AR213086A1 (es) 1978-12-15
SE435713B (sv) 1984-10-15
DK552674A (xx) 1975-06-16
SU608476A3 (ru) 1978-05-25
DE2450053A1 (de) 1975-04-24
CH595360A5 (xx) 1978-02-15
FR2361359A1 (fr) 1978-03-10
BG26531A4 (xx) 1979-04-12
ATA852374A (de) 1977-06-15
NZ175780A (en) 1978-04-03
DD116830A5 (xx) 1975-12-12
AU510909B2 (en) 1980-07-17
JPS57154174A (en) 1982-09-22
CS189671B2 (en) 1979-04-30
IL45880A (en) 1979-09-30
BG25991A3 (xx) 1979-01-12
BE821406A (fr) 1975-04-23
ES449655A1 (es) 1977-07-01
JPS5912671B2 (ja) 1984-03-24
AR221321A1 (es) 1981-01-30
IL52180A0 (en) 1977-07-31
IE40078B1 (en) 1979-03-14
FR2248041A1 (xx) 1975-05-16
ES449654A1 (es) 1977-07-01
ZA746594B (en) 1976-06-30
AU2880177A (en) 1979-03-15
SU604491A3 (ru) 1978-04-25
RO78465A (ro) 1982-02-26
IL45880A0 (en) 1974-12-31
JPS636066B2 (xx) 1988-02-08
NL7413848A (nl) 1975-04-25
FR2361328A1 (fr) 1978-03-10
AU7454774A (en) 1976-04-29
IL52179A0 (en) 1977-07-31
FR2361328B1 (xx) 1979-07-13
SE7710599L (sv) 1977-09-21
RO74031A (ro) 1982-02-01
SE7710600L (sv) 1977-09-21
FR2248041B1 (xx) 1978-09-08
PH11022A (en) 1977-10-25
US3951999A (en) 1976-04-20
ES431247A1 (es) 1977-02-16
SE7413237L (xx) 1975-04-24
HU171613B (hu) 1978-02-28
SU795459A3 (ru) 1981-01-07
GB1488003A (en) 1977-10-05
AT341520B (de) 1978-02-10
CA1042005A (en) 1978-11-07
JPS5077364A (xx) 1975-06-24
SE424324B (sv) 1982-07-12
YU282474A (en) 1982-02-28

Similar Documents

Publication Publication Date Title
RO69615A (ro) Procedeu pentru prepararea unor 2,4,6-triiod-izo-ftaloilamide
SE424325B (sv) Forfarande for framstellning av 1,2-bensisoxazoler
SE420720B (sv) Forfarande for framstellning av 2,6-disubstuerade fenylaminoguanidinforeningar
SE419750B (sv) Forfarande for framstellning av 6-acyl-2,4-dialkyl-2-hydroxicyklohexan-1,35-trion
NO740670L (no) Analogifremgangsmåte for fremstilling av nye 1-aryloksy-2-hydroksy-3-alkynylaminopropanforbindelser.
SE420491B (sv) Forfarande for framstellning av 1,1-diaryl-1-oxadiazol-alkylaminer
NO741886L (no) Fremgangsmåte for fremstilling av et veterinærpreparat.
SE403478B (sv) Sett att framstella 2,2,6,6-tetrametyl-4-oxopiperidin
NO741223L (no) Fremgangsmåte for fremstilling av 6-deoksytetracykliner.
AR206807A1 (es) Proceso para preparar derivados de 1,1-difenil-2-hidroxi-3aminopropano
SE387341B (sv) Forfarande for framstellning av 1-aryl-n-dialkyl-aminoalkyl-3,4-dihydro2(h)-isokinolinkarboxamider
NO740841L (no) Fremgangsmåte for fremstilling av 1-beta-D-ribofuranosyl-1, 2, 4-triazol-3-karboksamid.
RO69264A (ro) Procedeu pentru prepararea alfa-amino-alcoolilor
NO741133L (no) Fremgangsmåte for fremstilling av metyl-3-(2-kinoksalinylmetylen)-karbazat-N1.N4-dioksyd.
SE417092B (sv) Forfarande for framstellning av 1,2,3,4-tetrahydroisokinoliner
SE415475B (sv) Forfarande for framstellning av 4,5-didehydro-pgf?711alfa
SE420600B (sv) Forfarande for framstellning av 1,2,3,4-tetrahydroisokinoliner
SE401833B (sv) Forfarande for framstellnig av vissa angivna 1,2,4-friazolderivat
RO65994A (ro) Procedeu pentru prepararea unor diaminobenzofenone
SE423992B (sv) Forfarande for framstellning av 9, 11, 15-trihydroxi-13, 14-dehydroprostaglandiner
NO740820L (no) Fremgangsmåte for fremstilling av benzylaminer.
TR18199A (tr) Yeni 3, 4-dihidro-1, 2, 4-triazinlerin hazirlanmasina mahsus usul
SE396751B (sv) Sett att framstella s?72iv-benso-1,2,4-tiadiaziner
SU502900A1 (ru) "Способ получени производных -алкилоксаазафосфоринанов-1,3,2
NO740744L (no) Fremgangsmåte til fremstilling av oksiranforbindelser.