BE883390A - Derives de l'acide penicillanique utiles comme medicaments, compositions therapeutiques les contenant et procedes de leur preparation - Google Patents
Derives de l'acide penicillanique utiles comme medicaments, compositions therapeutiques les contenant et procedes de leur preparation Download PDFInfo
- Publication number
- BE883390A BE883390A BE0/200687A BE200687A BE883390A BE 883390 A BE883390 A BE 883390A BE 0/200687 A BE0/200687 A BE 0/200687A BE 200687 A BE200687 A BE 200687A BE 883390 A BE883390 A BE 883390A
- Authority
- BE
- Belgium
- Prior art keywords
- emi
- salt
- acid
- penicillanate
- mixture
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB7917665 | 1979-05-21 | ||
GB7930819 | 1979-09-05 | ||
GB7941252 | 1979-11-29 | ||
GB8006681 | 1980-02-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE883390A true BE883390A (fr) | 1980-11-20 |
Family
ID=27449123
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE0/200687A BE883390A (fr) | 1979-05-21 | 1980-05-20 | Derives de l'acide penicillanique utiles comme medicaments, compositions therapeutiques les contenant et procedes de leur preparation |
Country Status (19)
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4432970A (en) * | 1979-11-23 | 1984-02-21 | Pfizer Inc. | 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IE51846B1 (en) * | 1980-11-17 | 1987-04-15 | Leo Pharm Prod Ltd | Pharmaceutical preparation for veterinary use and an appliance containing it |
US4521533A (en) * | 1984-07-12 | 1985-06-04 | Pfizer Inc. | Salts of 6-alpha-(aminomethyl)penicillanic acid 1,1-dioxide esters and beta-lactam antibiotics |
GB8522156D0 (en) * | 1985-09-06 | 1985-10-09 | Leo Pharm Prod Ltd | Producing chemical compounds |
US5589354A (en) * | 1994-12-20 | 1996-12-31 | Biopure Corporation | Halogenation of cephalexin with haloperoxidase from Rathayibacter biopuresis |
US5695951A (en) * | 1994-12-20 | 1997-12-09 | Biopure Corporation | Chlorination of cephalexin with chloroperoxidase from Rathayibacter biopuresis |
DK0971690T4 (en) | 1996-12-18 | 2015-07-13 | Bimeda Res & Dev Ltd | Anti-infective intramammary veterinary composition. |
US20020035107A1 (en) * | 2000-06-20 | 2002-03-21 | Stefan Henke | Highly concentrated stable meloxicam solutions |
CA2501395C (en) * | 2002-10-25 | 2011-05-24 | Akzo Nobel Nv | Prolonged release pharmaceutical composition |
EP1568369A1 (en) | 2004-02-23 | 2005-08-31 | Boehringer Ingelheim Vetmedica Gmbh | Use of meloxicam for the treatment of respiratory diseases in pigs |
DE102004025324A1 (de) * | 2004-05-19 | 2005-12-08 | Boehringer Ingelheim Vetmedica Gmbh | Flüssige Zubereitung für die Veterinärmedizin, Verfahren zu deren Herstellung und deren Verwendung |
WO2014014364A1 (en) * | 2012-07-17 | 2014-01-23 | Bayer New Zealand Limited | Injectable antibiotic formulations and their methods of use |
MY172561A (en) * | 2012-07-17 | 2019-12-03 | Bayer New Zealand Ltd | Injectable antibiotic formulations and their methods of use |
BR112015014963B1 (pt) * | 2012-12-20 | 2022-04-12 | Alleva Animal Health Limited | Formulação de suspensão injetável veterinária |
EP4265241A1 (en) * | 2022-04-20 | 2023-10-25 | Bilim Ilac Sanayii Ve Ticaret A.S. | Tablet formulations for the treatment of urinary system infections and method for the preparation of such formulations |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1089385B (de) | 1954-06-21 | 1960-09-22 | Biochemie Gmbh | Verfahren zur Herstellung von in Wasser schwer loeslichen, besonders fuer die Oraltherapie geeigneten Salzen des Penicillins mit organischen Basen |
DE1031795B (de) | 1955-09-29 | 1958-06-12 | Chimiotherapie Lab Franc | Verfahren zur Herstellung eines Salzes aus Penicillin und einer Piperazinbase |
US3206469A (en) * | 1961-08-15 | 1965-09-14 | Lepetit Spa | 6-halopenicillanic acid |
GB1297555A (US07579456-20090825-P00002.png) * | 1970-09-22 | 1972-11-22 | ||
GB1377817A (en) * | 1971-06-09 | 1974-12-18 | Beecham Group Ltd | Penicillins and cephalosporins |
US4234579A (en) * | 1977-06-07 | 1980-11-18 | Pfizer Inc. | Penicillanic acid 1,1-dioxides as β-lactamase inhibitors |
IN149747B (US07579456-20090825-P00002.png) * | 1977-06-07 | 1982-04-03 | Pfizer | |
US4180506A (en) * | 1978-01-18 | 1979-12-25 | Rex Pratt | 6β-Bromo penicillanic acid |
CA1158639A (en) | 1978-12-11 | 1983-12-13 | Eric M. Gordon | 6-bromopenicillanic acid sulfone |
US4203992A (en) * | 1978-12-11 | 1980-05-20 | E. R. Squibb & Sons, Inc. | β-Bromopenicillanic acid sulfone |
IL59081A0 (en) * | 1979-01-10 | 1980-05-30 | Schering Corp | 2-penem compounds and a method for preparing them |
DE3068390D1 (en) * | 1979-01-10 | 1984-08-09 | Beecham Group Plc | Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds |
US4518530A (en) * | 1979-03-05 | 1985-05-21 | Pfizer Inc. | 6-β-Substituted penicillanic acids as β-lactamase inhibitors |
US4397783A (en) * | 1979-03-05 | 1983-08-09 | Pfizer Inc. | Process for converting 6,6-disubstituted penicillanic acid derivatives to the 6-β-congeners |
US4287181A (en) * | 1979-10-22 | 1981-09-01 | Pfizer Inc. | Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors |
US4432970A (en) * | 1979-11-23 | 1984-02-21 | Pfizer Inc. | 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors |
-
1980
- 1980-04-29 IE IE2559/84A patent/IE49770B1/en unknown
- 1980-04-29 IE IE868/80A patent/IE49768B1/en not_active IP Right Cessation
- 1980-04-29 IL IL59948A patent/IL59948A0/xx unknown
- 1980-05-01 NZ NZ193597A patent/NZ193597A/en unknown
- 1980-05-05 PH PH23982A patent/PH17959A/en unknown
- 1980-05-12 GR GR61906A patent/GR68372B/el unknown
- 1980-05-19 SE SE8003722A patent/SE452465B/sv not_active IP Right Cessation
- 1980-05-20 JP JP6768580A patent/JPS55154977A/ja active Granted
- 1980-05-20 BE BE0/200687A patent/BE883390A/fr not_active IP Right Cessation
- 1980-05-20 NL NL8002911A patent/NL8002911A/nl not_active Application Discontinuation
- 1980-05-20 DE DE19803051038 patent/DE3051038C2/de not_active Expired
- 1980-05-20 DE DE19803051037 patent/DE3051037C2/de not_active Expired
- 1980-05-20 DK DK218580A patent/DK158669C/da not_active IP Right Cessation
- 1980-05-20 FR FR8011263A patent/FR2457294A1/fr active Granted
- 1980-05-20 IT IT67790/80A patent/IT1133091B/it active
- 1980-05-20 CA CA000352237A patent/CA1265787A/en not_active Expired - Fee Related
- 1980-05-20 PT PT71273A patent/PT71273A/pt unknown
- 1980-05-20 DE DE19803019244 patent/DE3019244A1/de active Granted
- 1980-05-20 LU LU82468A patent/LU82468A1/fr unknown
- 1980-05-20 FI FI801618A patent/FI801618A/fi not_active Application Discontinuation
- 1980-05-20 AU AU58584/80A patent/AU534754B2/en not_active Ceased
- 1980-11-17 US US06/207,614 patent/US4446144A/en not_active Expired - Lifetime
-
1982
- 1982-03-04 FR FR8203636A patent/FR2499575A1/fr active Granted
-
1983
- 1983-08-26 AU AU18487/83A patent/AU541323B2/en not_active Ceased
- 1983-08-26 PH PH29453A patent/PH19005A/en unknown
- 1983-08-26 AU AU18486/83A patent/AU541322B2/en not_active Ceased
- 1983-12-23 US US06/564,901 patent/US4594246A/en not_active Expired - Fee Related
-
1984
- 1984-12-06 SE SE8406201A patent/SE462096B/sv not_active IP Right Cessation
- 1984-12-06 SE SE8406202A patent/SE462097B/sv not_active IP Right Cessation
-
1986
- 1986-03-31 US US06/845,941 patent/US4672114A/en not_active Expired - Fee Related
-
1989
- 1989-11-10 DK DK562589A patent/DK158670C/da not_active IP Right Cessation
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4432970A (en) * | 1979-11-23 | 1984-02-21 | Pfizer Inc. | 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors |
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: LEO PHARMACEUTICAL PRODUCTS LTD A/S (LOVENS KEMIS Effective date: 19950531 |