BE868594A - Derives alpha-acetyleniques d'amines utiles notamment comme inhibiteurs de certaines decarboxylases et leur procede de preparation - Google Patents
Derives alpha-acetyleniques d'amines utiles notamment comme inhibiteurs de certaines decarboxylases et leur procede de preparationInfo
- Publication number
- BE868594A BE868594A BE188954A BE188954A BE868594A BE 868594 A BE868594 A BE 868594A BE 188954 A BE188954 A BE 188954A BE 188954 A BE188954 A BE 188954A BE 868594 A BE868594 A BE 868594A
- Authority
- BE
- Belgium
- Prior art keywords
- decarboxylases
- inhibitors
- alpha
- certain
- preparation process
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
- C07C279/04—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton
- C07C279/12—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton being further substituted by nitrogen atoms not being part of nitro or nitroso groups
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Communicable Diseases (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Dermatology (AREA)
- Hematology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Oncology (AREA)
- Immunology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Saccharide Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/812,265 US4139563A (en) | 1977-07-01 | 1977-07-01 | α-ACETYLENIC DERIVATIVES OF AMINES |
Publications (1)
Publication Number | Publication Date |
---|---|
BE868594A true BE868594A (fr) | 1978-10-16 |
Family
ID=25209053
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE188954A BE868594A (fr) | 1977-07-01 | 1978-06-29 | Derives alpha-acetyleniques d'amines utiles notamment comme inhibiteurs de certaines decarboxylases et leur procede de preparation |
Country Status (14)
Country | Link |
---|---|
US (1) | US4139563A (ja) |
JP (1) | JPS5481206A (ja) |
AU (1) | AU517458B2 (ja) |
BE (1) | BE868594A (ja) |
CA (1) | CA1090790A (ja) |
CH (1) | CH640820A5 (ja) |
DE (1) | DE2827907A1 (ja) |
ES (1) | ES471269A1 (ja) |
FR (1) | FR2395990A1 (ja) |
GB (1) | GB2001058B (ja) |
IT (1) | IT1105054B (ja) |
NL (1) | NL190115C (ja) |
NZ (1) | NZ187543A (ja) |
ZA (1) | ZA783355B (ja) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4182891A (en) * | 1977-07-01 | 1980-01-08 | Merrell Toraude Et Compagnie | α-Acetylenic derivatives of α-amino acids |
US4456619A (en) * | 1978-09-18 | 1984-06-26 | Sandoz, Inc. | Amides of 2-alkynoic acids and use for inhibiting accumulation of cholesterol ester in arterial walls |
US4414395A (en) * | 1980-03-13 | 1983-11-08 | Ciba-Geigy Corporation | Process for the manufacture of hydrazono-isoindolines |
ZA811555B (en) * | 1980-03-25 | 1982-03-31 | Merrell Toraude & Co | Substituted deoxyadenosine derivatives |
PH16634A (en) * | 1980-06-16 | 1983-12-05 | Merrell Dow Pharma | Method of inhibiting the growth of protozoa |
US4437873A (en) | 1981-03-23 | 1984-03-20 | Merrell Dow Pharmaceuticals Inc. | Method of inhibiting algae |
IE54304B1 (en) * | 1981-08-19 | 1989-08-16 | Merrell Dow France | Fluorinated diamino-heptene and -heptyne derivatives |
US4376116A (en) * | 1981-09-01 | 1983-03-08 | Research Corporation | Polyamine biosynthesis inhibitors |
US4421768A (en) | 1982-08-11 | 1983-12-20 | Merrell Toraude Et Compagnie | Fluorinated diamino-heptene and-heptyne derivatives |
US4720489A (en) * | 1984-10-15 | 1988-01-19 | Douglas Shander | Hair growth modification with ornithine decarboxylase inhibitors |
US5196450A (en) * | 1985-12-19 | 1993-03-23 | Merrell Dow Pharmaceuticals Inc. | Method of inhibiting protozoal growth |
JPS62148462A (ja) * | 1985-12-19 | 1987-07-02 | メレルダウフア−マス−テイカルズ インコ−ポレ−テツド | 原生動物の生長を抑制する新規な方法 |
US4707498A (en) * | 1986-01-14 | 1987-11-17 | Merrell Dow Pharmaceuticals Inc. | Fluorinated diaminoalkyne derivatives |
US5366971A (en) * | 1987-11-09 | 1994-11-22 | Sandoz Ltd. | Use of 11,28-dioxa-4-azatricyclo[22.3.1.04,9 ]octacos-18-ene derivatives and pharmaceutical compositions containing them |
DK175235B1 (da) * | 1987-11-09 | 2004-07-19 | Novartis Ag | Ny anvendelse af azatricycloderivater og farmaceutiske præparater med indhold deraf |
US5013719A (en) * | 1988-05-13 | 1991-05-07 | Merrell Dow Pharmaceuticals Inc. | Method of effecting immunosuppression |
WO2001095897A1 (en) | 2000-06-15 | 2001-12-20 | University Of Kentucky Research Foundation | Agmatine and agmatine analogs in the treatment of epilepsy, seizure, and electroconvulsive disorders |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2766285A (en) * | 1952-10-20 | 1956-10-09 | Lilly Co Eli | Substituted aminopropynes and process for their preparation |
US3024190A (en) * | 1958-10-03 | 1962-03-06 | Commercial Solvents Corp | Process for the control of bacteria in a flooding process for the recovery of petroleum oil |
US3160664A (en) * | 1959-04-10 | 1964-12-08 | Miles Lab | Acetylenic omega-haloalkylamines |
GB1041987A (en) * | 1964-09-03 | 1966-09-07 | Beecham Group Ltd | Acetylenic compounds |
US3291683A (en) * | 1965-05-24 | 1966-12-13 | American Cyanamid Co | Controlling fungi and bacteria with alkoxy or alkylthio alkylamine ethers |
FR1481067A (fr) * | 1965-12-29 | 1967-05-19 | Soc Ind Fab Antibiotiques Sifa | Nouvelles nu-propynyl méthylamines et leurs sels et procédé de préparation |
GB1161915A (en) * | 1966-06-03 | 1969-08-20 | Ciba Ltd | Pharmaceutical Preparations comprising Sulphur-Containing Amino-Compounds for the Treatment of Depressive Conditions |
US3960927A (en) * | 1975-03-18 | 1976-06-01 | Richardson-Merrell Inc. | Olefinic derivatives of amino acids |
FR2354100A2 (fr) * | 1976-06-08 | 1978-01-06 | Anvar | Medicament a base de 5' thioethers de l'adenosine |
-
1977
- 1977-07-01 US US05/812,265 patent/US4139563A/en not_active Expired - Lifetime
-
1978
- 1978-06-06 CA CA304,897A patent/CA1090790A/en not_active Expired
- 1978-06-12 ZA ZA00783355A patent/ZA783355B/xx unknown
- 1978-06-13 NZ NZ187543A patent/NZ187543A/xx unknown
- 1978-06-21 AU AU37320/78A patent/AU517458B2/en not_active Expired
- 1978-06-24 DE DE19782827907 patent/DE2827907A1/de active Granted
- 1978-06-27 GB GB7827970A patent/GB2001058B/en not_active Expired
- 1978-06-28 FR FR7819353A patent/FR2395990A1/fr active Granted
- 1978-06-28 IT IT7850078A patent/IT1105054B/it active
- 1978-06-29 BE BE188954A patent/BE868594A/xx not_active IP Right Cessation
- 1978-06-29 ES ES471269A patent/ES471269A1/es not_active Expired
- 1978-06-29 CH CH710778A patent/CH640820A5/de not_active IP Right Cessation
- 1978-06-30 NL NLAANVRAGE7807090,A patent/NL190115C/xx not_active IP Right Cessation
- 1978-07-01 JP JP7927378A patent/JPS5481206A/ja active Granted
Also Published As
Publication number | Publication date |
---|---|
ZA783355B (en) | 1979-06-27 |
NL190115B (nl) | 1993-06-01 |
NL7807090A (nl) | 1979-01-03 |
NL190115C (nl) | 1993-11-01 |
FR2395990B1 (ja) | 1980-07-18 |
IT7850078A0 (it) | 1978-06-28 |
JPS6216941B2 (ja) | 1987-04-15 |
ES471269A1 (es) | 1979-10-01 |
NZ187543A (en) | 1982-03-30 |
FR2395990A1 (fr) | 1979-01-26 |
CH640820A5 (de) | 1984-01-31 |
JPS5481206A (en) | 1979-06-28 |
IT1105054B (it) | 1985-10-28 |
CA1090790A (en) | 1980-12-02 |
AU517458B2 (en) | 1981-07-30 |
US4139563A (en) | 1979-02-13 |
AU3732078A (en) | 1980-01-03 |
GB2001058A (en) | 1979-01-24 |
DE2827907C2 (ja) | 1987-10-01 |
DE2827907A1 (de) | 1979-01-11 |
GB2001058B (en) | 1982-02-03 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE20 | Patent expired |
Owner name: MERRELL TORAUDE ET CIE Effective date: 19980629 |