BE862568A - Nouvelles piperazines disubstituees, leurs procedes de preparation et leur application en therapeutique - Google Patents

Nouvelles piperazines disubstituees, leurs procedes de preparation et leur application en therapeutique

Info

Publication number
BE862568A
BE862568A BE184051A BE184051A BE862568A BE 862568 A BE862568 A BE 862568A BE 184051 A BE184051 A BE 184051A BE 184051 A BE184051 A BE 184051A BE 862568 A BE862568 A BE 862568A
Authority
BE
Belgium
Prior art keywords
disubstitled
piperazines
therapeutics
preparation
new
Prior art date
Application number
BE184051A
Other languages
English (en)
French (fr)
Original Assignee
Science Union & Cie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Science Union & Cie filed Critical Science Union & Cie
Publication of BE862568A publication Critical patent/BE862568A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C07D271/071,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/101,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/14Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/081,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/121,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/1251,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C07D285/135Nitrogen atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
BE184051A 1976-12-31 1977-12-30 Nouvelles piperazines disubstituees, leurs procedes de preparation et leur application en therapeutique BE862568A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB54398/76A GB1560084A (en) 1976-12-31 1976-12-31 Disubstituted piperazines processes for their preparation and pharmaceutical mompositions containing them

Publications (1)

Publication Number Publication Date
BE862568A true BE862568A (fr) 1978-06-30

Family

ID=10470884

Family Applications (1)

Application Number Title Priority Date Filing Date
BE184051A BE862568A (fr) 1976-12-31 1977-12-30 Nouvelles piperazines disubstituees, leurs procedes de preparation et leur application en therapeutique

Country Status (24)

Country Link
US (1) US4177272A (da)
JP (1) JPS5384984A (da)
AR (3) AR216931A1 (da)
AT (1) AT358591B (da)
AU (1) AU513087B2 (da)
BE (1) BE862568A (da)
CA (1) CA1100968A (da)
DD (1) DD133802A5 (da)
DE (1) DE2758314A1 (da)
DK (1) DK572977A (da)
FR (1) FR2376148A1 (da)
GB (1) GB1560084A (da)
GR (1) GR62407B (da)
IE (1) IE46284B1 (da)
IL (1) IL53714A (da)
NL (1) NL7714628A (da)
NZ (1) NZ186158A (da)
OA (1) OA05840A (da)
PH (1) PH14321A (da)
PT (1) PT67486B (da)
SE (1) SE7714884L (da)
SU (2) SU703021A3 (da)
YU (1) YU304377A (da)
ZA (1) ZA777680B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2418798A1 (fr) * 1978-03-03 1979-09-28 Science Union & Cie Nouvelles piperazines disubstituees, leurs procedes de preparation et les compositions pharmaceutiques les renfermant
US4421753A (en) * 1982-01-15 1983-12-20 American Cyanamid Company 1-(5-Amino-4H-1,2,4-triazol-3-yl)-4-substituted-piperazines
FR2519986A1 (fr) * 1982-01-21 1983-07-22 Adir Nouveaux derives de benzodioxine, leurs procedes de preparation et les compositions pharmaceutiques les renfermant
FR2799464B1 (fr) * 1999-10-12 2001-12-28 Norchim Procede de fabrication de piperonyl piperazine par animation reductive
US10562869B2 (en) 2014-03-17 2020-02-18 Remynd Nv Oxadiazole compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1595923A1 (de) * 1965-02-20 1969-11-27 Merck Ag E 1-Aralkyl-4-(thiazolyl-2)-piperazine und Verfahren zu ihrer Herstellung
GB1307256A (en) * 1970-09-15 1973-02-14 Science Union & Cie Piperazine derivatives and a process for their preparation
GB1369379A (en) * 1972-04-07 1974-10-09 Science Union & Cie Benzodioxole derivatives and processes for preparing them
GB1407552A (en) * 1973-04-02 1975-09-24 Science Union & Cie Disubstituted piperazines processes for their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
FR2376148B1 (da) 1981-05-29
IL53714A0 (en) 1978-03-10
ATA927577A (de) 1980-02-15
CA1100968A (fr) 1981-05-12
AT358591B (de) 1980-09-25
JPS6149314B2 (da) 1986-10-29
JPS5384984A (en) 1978-07-26
DK572977A (da) 1978-07-01
DD133802A5 (de) 1979-01-24
GR62407B (en) 1979-04-11
AR217143A1 (es) 1980-02-29
GB1560084A (en) 1980-01-30
PT67486A (fr) 1978-01-01
OA05840A (fr) 1981-05-31
SU793397A3 (ru) 1980-12-30
PH14321A (en) 1981-05-27
IE46284L (en) 1978-06-30
AR217144A1 (es) 1980-02-29
AR216931A1 (es) 1980-02-15
AU3204577A (en) 1979-07-05
US4177272A (en) 1979-12-04
YU304377A (en) 1983-01-21
NZ186158A (en) 1980-03-05
AU513087B2 (en) 1980-11-13
SE7714884L (sv) 1978-07-02
DE2758314A1 (de) 1978-07-06
IL53714A (en) 1981-07-31
ZA777680B (en) 1978-10-25
FR2376148A1 (fr) 1978-07-28
IE46284B1 (en) 1983-04-20
SU703021A3 (ru) 1979-12-05
PT67486B (fr) 1979-05-30
NL7714628A (nl) 1978-07-04

Similar Documents

Publication Publication Date Title
BE887800A (fr) Derives de carbostyrile, leurs procedes de preparation et leur application en therapeutique
BE809041A (fr) Nouvelles arylpiperazines et leurs procedes de preparation
BE865990A (fr) Nouvelles cinnamoyles piperazines et homopiperazines, leur procede de preparation et leur application en therapeutique
BE839615A (fr) Nouvelles amidinourees, leur preparation et leur emploi
BE851893A (fr) Nouvelles aryl-3 oxazolidinones-2, leur procede de preparation et leur application en therapeutique
BE827323A (fr) Nouvelles diaryl-1,1 oxadiazole-1 alkylamines, leur procede de preparation et leur utilisation therapeutique
BE856636A (fr) Nouvelles 7-b-oxyiminoacylcephalosporines, leurs procedes de preparation et leurs applications en therapeutique
FR2348907A1 (fr) Derives polyprenyliques,leur procede de preparation et leur application en therapeutique
BE856784A (fr) Nouvelles quinazolinones, leurs procedes d'obtention et leur application a la therapeutique
BE843152A (fr) Nouvelles cephalosporimes, leur preparation et leur emploi
BE829807A (fr) Nouvelles 1,4-dihydropyridines et leurs procedes de preparation
FR2345439A1 (fr) Dihydrooxadiazinones et leurs procedes de preparation
FR2342290A1 (fr) Aminoalkylpyrrolobenzoxo-aza-alcanes, leur preparation et leurs applications
BE862568A (fr) Nouvelles piperazines disubstituees, leurs procedes de preparation et leur application en therapeutique
FR2352804A1 (fr) 4-quinazolinyl-guanidines, leur preparation et leur application en therapeutique
BE869352A (fr) Nouvelles nitrosourees et leur application
BE884602R (fr) Nouvelles cinnamoyles piperazines et homopiperazines leur procede de preparation et leur application en therapeutique
FR2302102A1 (fr) Nouvelles substances antibiotiques derivees de l'antibiotique 67-694 et leurs procedes de preparation
FR2283689A1 (fr) Nouvelles cephamycines, leur preparation et leur application
BE871857A (fr) Nouvelles piperazines disubstituees, leur procedes de preparation et les compositions pharmaceutiques les renfermant
FR2321284A1 (fr) Nouvelles o-(arylsulfonamido) alkylamine, leur procede de preparation et leur application en therapeutique
FR2352783A1 (fr) Derives polyprenyl-carboxyliques, leur procede de preparation et leur application en therapeutique
BE838630A (fr) Aminocyclitols antibiotiques et leurs procedes de preparation
FR2301511A1 (fr) Pentafluorsethylarylamines et leurs procedes de preparation
FR2343746A1 (fr) Nouvelles cephalosporines, leur procede de preparation et leur application en therapeutique