FR2352804A1 - 4-quinazolinyl-guanidines, leur preparation et leur application en therapeutique - Google Patents

4-quinazolinyl-guanidines, leur preparation et leur application en therapeutique

Info

Publication number
FR2352804A1
FR2352804A1 FR7716549A FR7716549A FR2352804A1 FR 2352804 A1 FR2352804 A1 FR 2352804A1 FR 7716549 A FR7716549 A FR 7716549A FR 7716549 A FR7716549 A FR 7716549A FR 2352804 A1 FR2352804 A1 FR 2352804A1
Authority
FR
France
Prior art keywords
guanidines
quinazolinyl
therapeutics
preparation
application
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
FR7716549A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hoechst AG
Original Assignee
Hoechst AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst AG filed Critical Hoechst AG
Publication of FR2352804A1 publication Critical patent/FR2352804A1/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
    • C07D295/215Radicals derived from nitrogen analogues of carbonic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR7716549A 1976-05-28 1977-05-31 4-quinazolinyl-guanidines, leur preparation et leur application en therapeutique Withdrawn FR2352804A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19762623846 DE2623846A1 (de) 1976-05-28 1976-05-28 4-chinazolinyl-guanidine und verfahren zu ihrer herstellung

Publications (1)

Publication Number Publication Date
FR2352804A1 true FR2352804A1 (fr) 1977-12-23

Family

ID=5979166

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7716549A Withdrawn FR2352804A1 (fr) 1976-05-28 1977-05-31 4-quinazolinyl-guanidines, leur preparation et leur application en therapeutique

Country Status (4)

Country Link
US (1) US4128643A (fr)
JP (1) JPS52148085A (fr)
DE (1) DE2623846A1 (fr)
FR (1) FR2352804A1 (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5793977A (en) * 1980-11-26 1982-06-11 Sankyo Co Ltd Acylaminoquinazoline derivative and its preparation
DZ3415A1 (fr) * 2000-08-31 2002-03-07 Chiron Corp Guanidinobenzamides comme mc4-r agonistes.
EP1385823B1 (fr) * 2001-04-09 2006-12-13 Chiron Corporation Composes guanidino comme agonistes du recepteur 4 de la melanocortine (mc4-r)
EP1487474A4 (fr) * 2002-02-25 2006-11-29 Chiron Corp Administration intranasale d'agonistes de mc4-r
PT1551834E (pt) 2002-05-23 2010-09-30 Novartis Vaccines & Diagnostic Compostos de quinazolinona substituídos
WO2004112793A1 (fr) * 2003-05-23 2004-12-29 Chiron Corporation Composes de quinazoline substitues par guanidino constituant des agonistes de mc4-r
KR20060105785A (ko) * 2003-11-19 2006-10-11 카이론 코포레이션 감소된 생체축적을 갖는 퀴나졸리논 화합물
JP5739820B2 (ja) 2008-12-30 2015-06-24 アークル インコーポレイテッド 置換5,6−ジヒドロ−6−フェニルベンゾ[f]イソキノリン−2−アミン化合物

Also Published As

Publication number Publication date
DE2623846A1 (de) 1977-12-15
US4128643A (en) 1978-12-05
JPS52148085A (en) 1977-12-08

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Legal Events

Date Code Title Description
ST Notification of lapse