BE862213A - Derives de 5-fluoro-uracile et leur application en therapeutique - Google Patents

Derives de 5-fluoro-uracile et leur application en therapeutique

Info

Publication number
BE862213A
BE862213A BE183769A BE183769A BE862213A BE 862213 A BE862213 A BE 862213A BE 183769 A BE183769 A BE 183769A BE 183769 A BE183769 A BE 183769A BE 862213 A BE862213 A BE 862213A
Authority
BE
Belgium
Prior art keywords
uracil
therapeutics
fluoro
derivatives
application
Prior art date
Application number
BE183769A
Other languages
English (en)
French (fr)
Original Assignee
Eisai Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai Co Ltd filed Critical Eisai Co Ltd
Publication of BE862213A publication Critical patent/BE862213A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE183769A 1976-12-24 1977-12-22 Derives de 5-fluoro-uracile et leur application en therapeutique BE862213A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP51154941A JPS6052708B2 (ja) 1976-12-24 1976-12-24 5−フルオロウラシル系化合物およびそれを含有する抗腫瘍剤

Publications (1)

Publication Number Publication Date
BE862213A true BE862213A (fr) 1978-04-14

Family

ID=15595270

Family Applications (1)

Application Number Title Priority Date Filing Date
BE183769A BE862213A (fr) 1976-12-24 1977-12-22 Derives de 5-fluoro-uracile et leur application en therapeutique

Country Status (14)

Country Link
US (1) US4130648A (de)
JP (1) JPS6052708B2 (de)
AU (1) AU519524B2 (de)
BE (1) BE862213A (de)
CA (1) CA1077483A (de)
CH (1) CH636874A5 (de)
DE (1) DE2757431A1 (de)
ES (1) ES465406A1 (de)
FR (1) FR2378779A1 (de)
GB (1) GB1594840A (de)
NL (1) NL7714205A (de)
PH (1) PH12700A (de)
SE (1) SE436208B (de)
SU (2) SU827489A1 (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU1235864A1 (ru) * 1983-03-11 1986-06-07 Отделение ордена Ленина института химической физики АН СССР Нитроксильные производные 5-фторурацила,обладающие противоопухолевой активностью
US4727077A (en) * 1985-02-20 1988-02-23 Ishihara Sangyo Kaisha Ltd. Benzoyl urea compounds, process for their production, and antitumorous compositions containing them
DK197486A (da) * 1986-04-30 1987-10-31 Ferring Farma Lab 5-fluoruracilprodug
WO2018129533A1 (en) 2017-01-09 2018-07-12 Shuttle Pharmaceuticals, Llc Selective histone deacetylase inhibitors for the treatment of human disease
US11584733B2 (en) 2017-01-09 2023-02-21 Shuttle Pharmaceuticals, Inc. Selective histone deacetylase inhibitors for the treatment of human disease
WO2019139921A1 (en) 2018-01-09 2019-07-18 Shuttle Pharmaceuticals, Inc. Selective histone deacetylase inhibitors for the treatment of human disease

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5324951B2 (de) * 1973-11-28 1978-07-24

Also Published As

Publication number Publication date
SE7714670L (sv) 1978-06-25
AU519524B2 (en) 1981-12-10
JPS5379880A (en) 1978-07-14
FR2378779A1 (fr) 1978-08-25
SU827489A1 (ru) 1981-05-07
JPS6052708B2 (ja) 1985-11-20
CA1077483A (en) 1980-05-13
ES465406A1 (es) 1978-09-16
DE2757431A1 (de) 1978-06-29
PH12700A (en) 1979-07-20
NL7714205A (nl) 1978-06-27
CH636874A5 (de) 1983-06-30
AU3182577A (en) 1979-06-28
GB1594840A (en) 1981-08-05
SU795469A3 (ru) 1981-01-07
SE436208B (sv) 1984-11-19
FR2378779B1 (de) 1980-08-22
US4130648A (en) 1978-12-19

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: EISAI CO. LTD

Effective date: 19871231