BE843840A - Nouvelles guanidines et thiourees, leur procede de preparation et leur utilisations - Google Patents

Nouvelles guanidines et thiourees, leur procede de preparation et leur utilisations

Info

Publication number
BE843840A
BE843840A BE168682A BE168682A BE843840A BE 843840 A BE843840 A BE 843840A BE 168682 A BE168682 A BE 168682A BE 168682 A BE168682 A BE 168682A BE 843840 A BE843840 A BE 843840A
Authority
BE
Belgium
Prior art keywords
thiourees
preparation process
guanidines
new
new guanidines
Prior art date
Application number
BE168682A
Other languages
English (en)
French (fr)
Inventor
G R White
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE843840A publication Critical patent/BE843840A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BE168682A 1975-07-31 1976-07-06 Nouvelles guanidines et thiourees, leur procede de preparation et leur utilisations BE843840A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB31968/75A GB1565647A (en) 1975-07-31 1975-07-31 Pharmacologically active compounds 4-substituted-imidazole-5-methanols

Publications (1)

Publication Number Publication Date
BE843840A true BE843840A (fr) 1977-01-06

Family

ID=10331071

Family Applications (1)

Application Number Title Priority Date Filing Date
BE168682A BE843840A (fr) 1975-07-31 1976-07-06 Nouvelles guanidines et thiourees, leur procede de preparation et leur utilisations

Country Status (28)

Country Link
JP (1) JPS5219663A (xx)
AR (1) AR213100A1 (xx)
AT (1) AT356668B (xx)
AU (1) AU508262B2 (xx)
BE (1) BE843840A (xx)
CA (1) CA1075702A (xx)
CS (1) CS203054B2 (xx)
DD (1) DD125205A5 (xx)
DE (1) DE2634430A1 (xx)
DK (1) DK316376A (xx)
ES (1) ES450309A1 (xx)
FI (1) FI762191A (xx)
FR (1) FR2319341A1 (xx)
GB (1) GB1565647A (xx)
GR (1) GR61114B (xx)
HU (1) HU174068B (xx)
IL (1) IL50006A0 (xx)
LU (1) LU75495A1 (xx)
NL (1) NL7608505A (xx)
NO (1) NO762659L (xx)
OA (1) OA05405A (xx)
PH (1) PH13417A (xx)
PT (1) PT65377B (xx)
RO (1) RO72312B (xx)
SE (1) SE7608478L (xx)
SU (1) SU655310A3 (xx)
ZA (1) ZA763686B (xx)
ZM (1) ZM9676A1 (xx)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4112234A (en) 1977-08-22 1978-09-05 Bristol-Myers Company Imidazolylmethylthioethyl alkynyl guanidines
US4165378A (en) 1977-04-20 1979-08-21 Ici Americas Inc. Guanidine derivatives of imidazoles and thiazoles
US4165377A (en) 1977-04-20 1979-08-21 Ici Americas Inc. Guanidino imidazoles and thiazoles
US4200760A (en) * 1978-09-26 1980-04-29 Bristol-Myers Company Imidazolylalkylthioalkylamino-ethylene derivatives
US4233302A (en) 1977-12-23 1980-11-11 Glaxo Group Limited Amine derivatives and pharmaceutical compositions containing them
USRE31588E (en) * 1977-06-03 1984-05-22 Bristol-Myers Company Imidazolylmethylthioethyl alkynyl guanidines

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0008596A1 (fr) * 1978-09-04 1980-03-19 DEVINTER Europe S.A. Société anonyme dite: Procédé de préparation de dérivés du type 4-hydroxyméthyl imidazole à partir d'esters d'acides 4-imidazole carboxyliques correspondants
JPS5914460B2 (ja) * 1978-12-27 1984-04-04 相互薬工株式会社 H↓2受容体「きつ」抗剤シメチジンの製造法
CN103288742A (zh) * 2013-06-04 2013-09-11 四川百利药业有限责任公司 一种高纯度英加韦林原料的制备方法
US20230349922A1 (en) 2020-08-11 2023-11-02 Université De Strasbourg H2 Blockers Targeting Liver Macrophages for the Prevention and Treatment of Liver Disease and Cancer

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA938556A (en) * 1970-06-25 1973-12-18 Smith Kline And French Laboratories Limited Pharmaceutical compositions containing thiourea derivatives

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4165378A (en) 1977-04-20 1979-08-21 Ici Americas Inc. Guanidine derivatives of imidazoles and thiazoles
US4165377A (en) 1977-04-20 1979-08-21 Ici Americas Inc. Guanidino imidazoles and thiazoles
US4234735A (en) 1977-04-20 1980-11-18 Imperial Chemical Industries Limited Guanidino imidazoles and thiazoles
US4262126A (en) 1977-04-20 1981-04-14 Imperial Chemical Industries Limited Guanidine derivatives of imidazoles and thiazoles
USRE31588E (en) * 1977-06-03 1984-05-22 Bristol-Myers Company Imidazolylmethylthioethyl alkynyl guanidines
US4112234A (en) 1977-08-22 1978-09-05 Bristol-Myers Company Imidazolylmethylthioethyl alkynyl guanidines
US4233302A (en) 1977-12-23 1980-11-11 Glaxo Group Limited Amine derivatives and pharmaceutical compositions containing them
US4200760A (en) * 1978-09-26 1980-04-29 Bristol-Myers Company Imidazolylalkylthioalkylamino-ethylene derivatives

Also Published As

Publication number Publication date
SU655310A3 (ru) 1979-03-30
OA05405A (fr) 1981-02-28
JPS5219663A (en) 1977-02-15
AU1644776A (en) 1978-02-02
ES450309A1 (es) 1977-12-01
PH13417A (en) 1980-03-30
NO762659L (xx) 1977-02-01
AU508262B2 (en) 1980-03-13
DE2634430A1 (de) 1977-02-10
NL7608505A (nl) 1977-02-02
ATA552376A (de) 1979-10-15
DK316376A (da) 1977-02-01
IL50006A0 (en) 1976-09-30
FR2319341B1 (xx) 1979-01-12
AR213100A1 (es) 1978-12-15
AT356668B (de) 1980-05-12
RO72312A (ro) 1984-03-15
CA1075702A (en) 1980-04-15
PT65377A (en) 1976-08-01
LU75495A1 (xx) 1977-03-03
GR61114B (en) 1978-09-13
RO72312B (ro) 1984-03-31
FI762191A (xx) 1977-02-01
FR2319341A1 (fr) 1977-02-25
ZA763686B (en) 1977-05-25
DD125205A5 (xx) 1977-04-06
HU174068B (hu) 1979-10-28
CS203054B2 (en) 1981-02-27
GB1565647A (en) 1980-04-23
PT65377B (en) 1978-01-19
SE7608478L (sv) 1977-02-01
ZM9676A1 (en) 1977-07-21

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: SMITH KLINE + FRENCH LABORATORIES LTD

Effective date: 19840706