BE802596A - Carbazoles - Google Patents

Carbazoles

Info

Publication number
BE802596A
BE802596A BE133691A BE133691A BE802596A BE 802596 A BE802596 A BE 802596A BE 133691 A BE133691 A BE 133691A BE 133691 A BE133691 A BE 133691A BE 802596 A BE802596 A BE 802596A
Authority
BE
Belgium
Prior art keywords
carbazoles
Prior art date
Application number
BE133691A
Other languages
English (en)
French (fr)
Inventor
L Berger
A J Corraz
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BE802596A publication Critical patent/BE802596A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • C07D209/82Carbazoles; Hydrogenated carbazoles
    • C07D209/88Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • C07D209/82Carbazoles; Hydrogenated carbazoles
    • C07D209/86Carbazoles; Hydrogenated carbazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the ring system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE133691A 1972-07-24 1973-07-20 Carbazoles BE802596A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US27414272A 1972-07-24 1972-07-24

Publications (1)

Publication Number Publication Date
BE802596A true BE802596A (fr) 1974-01-21

Family

ID=23046965

Family Applications (1)

Application Number Title Priority Date Filing Date
BE133691A BE802596A (fr) 1972-07-24 1973-07-20 Carbazoles

Country Status (26)

Country Link
JP (1) JPS5740144B2 (en, 2012)
KR (1) KR780000289B1 (en, 2012)
AR (1) AR205331A1 (en, 2012)
AT (1) AT325607B (en, 2012)
AU (1) AU475534B2 (en, 2012)
BE (1) BE802596A (en, 2012)
CA (1) CA1026348A (en, 2012)
CH (1) CH587819A5 (en, 2012)
DD (1) DD107681A5 (en, 2012)
DE (1) DE2337340C2 (en, 2012)
DK (1) DK138537B (en, 2012)
FI (1) FI59244C (en, 2012)
FR (1) FR2193611B1 (en, 2012)
GB (1) GB1385620A (en, 2012)
HK (1) HK49878A (en, 2012)
HU (1) HU167611B (en, 2012)
IE (1) IE37942B1 (en, 2012)
IL (1) IL42799A (en, 2012)
KE (1) KE2847A (en, 2012)
LU (1) LU68071A1 (en, 2012)
MY (1) MY7800315A (en, 2012)
NL (1) NL169877C (en, 2012)
NO (1) NO142865C (en, 2012)
SE (2) SE402283B (en, 2012)
SU (1) SU509220A3 (en, 2012)
ZA (1) ZA734047B (en, 2012)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4146542A (en) * 1978-06-12 1979-03-27 Hoffmann-La Roche Inc. Dihydrocarbazole acetic acid and esters thereof
US4150031A (en) * 1978-06-26 1979-04-17 Hoffmann-La Roche Inc. Hydroxy methyl carbazole acetic acid and esters
US4158007A (en) * 1978-08-21 1979-06-12 Hoffmann-La Roche Inc. Carbazole methyl malonates
US4501908A (en) * 1981-03-12 1985-02-26 Hoffmann-La Roche Inc. 2,3-Isopropylidene ribonic acid, 1,4-lactones
JPS6040256U (ja) * 1983-08-25 1985-03-20 伊東 璋 容器類洗浄機
ATE61047T1 (de) * 1986-01-23 1991-03-15 Merck Frosst Canada Inc Tetrahydrocarbazol-1-alkansaeuren.
DE3786030T2 (de) 1986-03-27 1993-12-02 Merck Frosst Canada Inc Tetrahydrocarbazole Ester.
CA1326030C (en) * 1987-07-21 1994-01-11 John W. Gillard Cyclohept[b]indolealkanoic acids
EP0307077A1 (en) * 1987-07-21 1989-03-15 Merck Frosst Canada Inc. Tetrahydrocarbazoles for the improvement of cyclosporin therapy
PT95692A (pt) * 1989-10-27 1991-09-13 American Home Prod Processo para a preparacao de derivados de acidos indole-,indeno-,piranoindole- e tetra-hidrocarbazole-alcanoicos, ou quais sao uteis como inibidores de pla2 e da lipoxigenase
US6013808A (en) * 1998-06-16 2000-01-11 Pfizer Inc. Method of purifying carbazole ester precursors of 6-chloro-α-methyl-carbazole-2-acetic acid
JP2004010601A (ja) * 2002-06-11 2004-01-15 Nippon Steel Chem Co Ltd インドール誘導体の製造方法及びそのための有用な中間体
WO2004064771A2 (en) * 2003-01-14 2004-08-05 Merck & Co., Inc. Geminally di-substituted nsaid derivatives as abeta 42 lowering agents
EP2960204B1 (en) * 2003-05-06 2018-06-13 Air Products And Chemicals, Inc. Hydrogen storage by reversible hydrogenation of pi-conjugated substrates
EP1660450A4 (en) * 2003-08-15 2009-07-29 Univ Laval MONOMERS, OLIGOMERS AND POLYMERS OF 2-FUNCTIONALIZED AND 2,7-DIFUNCTIONAL CARBAZOLS
US7601856B2 (en) 2006-07-27 2009-10-13 Wyeth Benzofurans as potassium ion channel modulators
US7662831B2 (en) 2006-07-27 2010-02-16 Wyeth Llc Tetracyclic indoles as potassium channel modulators
RU2624446C9 (ru) * 2011-11-15 2018-04-04 Йиссум Ресерч Девелопмент Компани оф де Хебрю Юниверсити оф Джерусалем Лтд. Трициклические соединения, композиции, содержащие указанные соединения, и их применения
JP5940036B2 (ja) * 2013-10-08 2016-06-29 テックフィールズ バイオケム カンパニー リミテッド 非常に速い皮膚透過率を有するアリール−及びヘテロアリールプロピオン酸の正荷電水溶性プロドラッグ
CN114787130A (zh) * 2020-03-25 2022-07-22 捷恩智株式会社 化合物、液晶组合物及液晶显示元件

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DD70880A (en, 2012) *
US3580926A (en) * 1969-11-10 1971-05-25 Parke Davis & Co Carbazole-4-alkanoic acids and tetrahydrocarbazole-4-alkanoic acids
ZA715217B (en) * 1970-08-20 1972-04-26 Org Nv Anti-inflammatory preparations

Also Published As

Publication number Publication date
SE7605813L (sv) 1976-05-21
FR2193611B1 (en, 2012) 1976-05-14
SU509220A3 (ru) 1976-03-30
JPS4943973A (en, 2012) 1974-04-25
NO142865C (no) 1980-11-05
GB1385620A (en) 1975-02-26
NL7310275A (en, 2012) 1974-01-28
DK138537C (en, 2012) 1979-03-05
ZA734047B (en) 1974-03-27
AR205331A1 (es) 1976-04-30
SE402283B (sv) 1978-06-26
NL169877C (nl) 1982-09-01
CH587819A5 (en, 2012) 1977-05-13
AU475534B2 (en) 1976-08-26
IL42799A0 (en) 1973-10-25
FI59244C (fi) 1981-07-10
AT325607B (de) 1975-10-27
ATA649773A (de) 1975-01-15
KR780000289B1 (en) 1978-08-10
DK138537B (da) 1978-09-25
NL169877B (nl) 1982-04-01
FI59244B (fi) 1981-03-31
MY7800315A (en) 1978-12-31
IE37942B1 (en) 1977-11-23
FR2193611A1 (en, 2012) 1974-02-22
LU68071A1 (en, 2012) 1975-04-11
IE37942L (en) 1974-01-24
AU5839073A (en) 1975-01-23
IL42799A (en) 1977-03-31
NO142865B (no) 1980-07-28
JPS5740144B2 (en, 2012) 1982-08-25
HU167611B (en, 2012) 1975-11-28
CA1026348A (en) 1978-02-14
DE2337340A1 (de) 1974-02-14
DE2337340C2 (de) 1985-05-02
HK49878A (en) 1978-09-08
KE2847A (en) 1978-06-30
DD107681A5 (en, 2012) 1974-08-12

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Legal Events

Date Code Title Description
RE20 Patent expired

Owner name: F. HOFFMANN-LA ROCHE A.G.

Effective date: 19930720