BE794597A - Nouveaux alpha-aryl-piperidinoalcanols dont le groupe piperidino est substitue en 4 et leur procede de preparation - Google Patents

Nouveaux alpha-aryl-piperidinoalcanols dont le groupe piperidino est substitue en 4 et leur procede de preparation

Info

Publication number
BE794597A
BE794597A BE794597DA BE794597A BE 794597 A BE794597 A BE 794597A BE 794597D A BE794597D A BE 794597DA BE 794597 A BE794597 A BE 794597A
Authority
BE
Belgium
Prior art keywords
piperidinoalcanols
aryl
substituted
preparation process
piperidino group
Prior art date
Application number
Other languages
English (en)
French (fr)
Inventor
A A Carr
C R Kinsolving
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22829539&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BE794597(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of BE794597A publication Critical patent/BE794597A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
    • C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BE794597D 1972-01-28 1973-01-26 Nouveaux alpha-aryl-piperidinoalcanols dont le groupe piperidino est substitue en 4 et leur procede de preparation BE794597A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US22182172A 1972-01-28 1972-01-28

Publications (1)

Publication Number Publication Date
BE794597A true BE794597A (fr) 1973-05-16

Family

ID=22829539

Family Applications (1)

Application Number Title Priority Date Filing Date
BE794597D BE794597A (fr) 1972-01-28 1973-01-26 Nouveaux alpha-aryl-piperidinoalcanols dont le groupe piperidino est substitue en 4 et leur procede de preparation

Country Status (26)

Country Link
JP (1) JPS5115035B2 (da)
AR (1) AR195314A1 (da)
AT (2) AT321917B (da)
AU (1) AU467361B2 (da)
BE (1) BE794597A (da)
CA (1) CA978946A (da)
CH (2) CH587820A5 (da)
CS (1) CS177834B2 (da)
DD (1) DD103239A5 (da)
DE (1) DE2303306C3 (da)
DK (1) DK136713B (da)
ES (1) ES410731A1 (da)
FR (1) FR2181690B1 (da)
GB (1) GB1413138A (da)
HU (1) HU166477B (da)
IE (1) IE36983B1 (da)
IL (1) IL41060A (da)
LU (1) LU66916A1 (da)
NL (1) NL175410C (da)
NO (1) NO140057C (da)
PH (1) PH10264A (da)
PL (1) PL89095B1 (da)
SE (1) SE382058B (da)
SU (1) SU464997A3 (da)
YU (1) YU36013B (da)
ZA (1) ZA728544B (da)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3941795A (en) 1974-02-08 1976-03-02 Richardson-Merrell Inc. α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4254129A (en) * 1979-04-10 1981-03-03 Richardson-Merrell Inc. Piperidine derivatives
US4254130A (en) * 1979-04-10 1981-03-03 Richardson-Merrell Inc. Piperidine derivatives
IT1200123B (it) * 1985-09-27 1989-01-05 Ind Chimica Srl Procedimento per la preparazione di alfa-(p-terbutilfenil)-4-(idrossidifenilmetil)-1-piperidinobutanolo
US4742175A (en) * 1986-05-07 1988-05-03 Merrell Dow Pharmaceuticals Inc. Preparation of polymorphically pure terfenadine
JPS63101760U (da) * 1986-12-19 1988-07-02
IT1205685B (it) * 1987-05-26 1989-03-31 Erregierre Spa Processo per la preparazione di alfa-(alchilfenil)-4-(idrossi difenilmetil)-1-piperidina butanolo
ZA901360B (en) * 1989-02-28 1990-11-28 Merrell Dow Pharma Preparation of the low-melting polymorphic form of terfenadine
ZA903145B (en) * 1989-05-01 1991-02-27 Merrell Dow Pharma Process for the preparation of the high melting polymorphic form of terfenadine
DE3917241A1 (de) * 1989-05-26 1990-11-29 Schaper & Bruemmer Gmbh 4-(hydroxydiphenylmethyl)-1-piperidyl-phenylalkan-derivate
WO1993003025A1 (fr) * 1991-08-09 1993-02-18 Yoshitomi Pharmaceutical Industries, Ltd. Compose de thiophene
AU705427B2 (en) * 1995-05-08 1999-05-20 Aventisub Ii Inc. Alpha-(substituted alkylphenyl) -4-(hydroxydiphenylmethyl)-1-piperidine butanol derivatives, their preparation and their use as anti-histamines, anti-allergy agents and bronchodilators
DE59810863D1 (de) * 1997-03-11 2004-04-08 Aventis Pharma Inc Verfahren zur Herstellung von 4-(4-(4-(Hydroxydiphenyl)-1-piperidinyl)-1-hydroxybutyl)-alpha,alpha-dimenthylphenylessigsäure und phosphorylierter Derivate
US7498345B2 (en) * 2004-09-17 2009-03-03 Albany Molecular Research, Inc. Process for production of piperidine derivatives
WO2006043691A1 (ja) * 2004-10-18 2006-04-27 Reverse Proteomics Research Institute Co., Ltd. 創薬標的タンパク質及び標的遺伝子、並びにスクリーニング方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3081303A (en) * 1961-10-13 1963-03-12 Searle & Co 1-aminoalkyl-alpha, alpha-diphenylpiperidine-methanols
GB1242169A (en) * 1969-04-09 1971-08-11 Ucb Sa Piperidine derivatives

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3941795A (en) 1974-02-08 1976-03-02 Richardson-Merrell Inc. α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES

Also Published As

Publication number Publication date
YU3473A (en) 1981-02-28
YU36013B (en) 1981-11-13
DE2303306A1 (de) 1973-08-02
DK136713B (da) 1977-11-14
IE36983B1 (en) 1977-04-13
LU66916A1 (da) 1973-07-27
PH10264A (en) 1976-10-20
AU467361B2 (en) 1975-11-27
ES410731A1 (es) 1976-04-01
NL7300873A (da) 1973-07-31
PL89095B1 (da) 1976-10-30
GB1413138A (en) 1975-11-05
SU464997A3 (ru) 1975-03-25
NO140057C (no) 1979-07-04
NL175410C (nl) 1984-11-01
DE2303306C3 (de) 1979-05-31
AU4989372A (en) 1974-06-13
CH593259A5 (da) 1977-11-30
AR195314A1 (es) 1973-09-28
DK136713C (da) 1978-05-01
CH587820A5 (da) 1977-05-13
DD103239A5 (da) 1974-01-12
CS177834B2 (da) 1977-08-31
ZA728544B (en) 1974-02-27
SE382058B (sv) 1976-01-12
JPS5115035B2 (da) 1976-05-13
HU166477B (da) 1975-03-28
IL41060A0 (en) 1973-02-28
IL41060A (en) 1975-06-25
CA978946A (en) 1975-12-02
AT323742B (de) 1975-07-25
AT321917B (de) 1975-04-25
NL175410B (nl) 1984-06-01
DE2303306B2 (de) 1978-09-28
FR2181690A1 (da) 1973-12-07
IE36983L (en) 1973-07-28
JPS4885578A (da) 1973-11-13
NO140057B (no) 1979-03-19
FR2181690B1 (da) 1976-05-14

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Legal Events

Date Code Title Description
RE20 Patent expired

Owner name: MERRELL DOW PHARMACEUTICALS INC.

Effective date: 19930126