BE787251A - Nouvelles benzodiazepines et leur preparation - Google Patents

Nouvelles benzodiazepines et leur preparation

Info

Publication number
BE787251A
BE787251A BE787251DA BE787251A BE 787251 A BE787251 A BE 787251A BE 787251D A BE787251D A BE 787251DA BE 787251 A BE787251 A BE 787251A
Authority
BE
Belgium
Prior art keywords
preparation
benzodiazepines
new
new benzodiazepines
Prior art date
Application number
Other languages
English (en)
French (fr)
Inventor
J B Hester Jr
A R Hanze
Pour Lequel Agit J W Hanze
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Publication date
Publication of BE787251A publication Critical patent/BE787251A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23K—FODDER
    • A23K20/00—Accessory food factors for animal feeding-stuffs
    • A23K20/10—Organic substances
    • A23K20/116—Heterocyclic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Polymers & Plastics (AREA)
  • Pain & Pain Management (AREA)
  • Food Science & Technology (AREA)
  • Zoology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Anesthesiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Animal Husbandry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE787251D 1971-08-04 Nouvelles benzodiazepines et leur preparation BE787251A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US16909171A 1971-08-04 1971-08-04

Publications (1)

Publication Number Publication Date
BE787251A true BE787251A (fr) 1973-02-05

Family

ID=22614230

Family Applications (1)

Application Number Title Priority Date Filing Date
BE787251D BE787251A (fr) 1971-08-04 Nouvelles benzodiazepines et leur preparation

Country Status (8)

Country Link
JP (3) JPS5714351B1 (enExample)
AU (1) AU461139B2 (enExample)
BE (1) BE787251A (enExample)
CH (3) CH591488A5 (enExample)
DE (1) DE2237592C2 (enExample)
FR (1) FR2150732B1 (enExample)
GB (4) GB1389434A (enExample)
ZA (1) ZA724880B (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3917627A (en) * 1971-08-04 1975-11-04 Upjohn Co 6-Substituted 4H-imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines and process for their production
FR2183716A1 (en) * 1972-05-05 1973-12-21 Centre Etd Ind Pharma Substd-6-phenyl-4h-imidazo (1,2-a)-1,4-benzo diazepines - - tranquillisers anxiolytics,sedatives and muscle-relaxants
ZA755418B (en) * 1974-09-11 1977-06-29 Hoffmann La Roche Diazepine derivatives
US3910946A (en) * 1974-09-12 1975-10-07 Upjohn Co 4H-Imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines
GB1484968A (en) * 1974-11-06 1977-09-08 Parke Davis & Co 4-aryl-imidazo(1,2-alpha)pyrazolo(4,3-f)(1,4)diazepines and their production
SE422580B (sv) * 1975-08-07 1982-03-15 Hoffmann La Roche Analogiforfarande for framstellning av imidazo (1,5-a)(1,4)diazepin-foreningar
US4118386A (en) * 1977-04-04 1978-10-03 Hoffmann-La Roche Inc. Synthesis of imidazo[1,5-a]diazepine-3-carboxylates
EP0763537A3 (en) * 1993-05-14 1997-10-22 Genentech Inc Non-peptides farnesyl transfer inhibitors
AU4382896A (en) * 1995-02-02 1996-08-21 F. Hoffmann-La Roche Ag Acetylimidazobenzodiazepines
EP3160969B1 (en) 2014-06-26 2023-09-13 The Johns Hopkins University Peripherally restricted gaba positive allosteric modulators for the treatment of irritable bowel syndrome and other ailments of the peripheral nervous system
WO2018083051A1 (en) * 2016-11-01 2018-05-11 F. Hoffmann-La Roche Ag 1,3-dihydro-1,4-benzodiazepine-2-thiones for the treatment of cns related diseases
CN113717176B (zh) * 2021-10-09 2022-07-05 上海再启生物技术有限公司 一种制备瑞马唑仑的方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3987052A (en) * 1969-03-17 1976-10-19 The Upjohn Company 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines

Also Published As

Publication number Publication date
JPS5726667A (en) 1982-02-12
GB1389436A (en) 1975-04-03
FR2150732B1 (enExample) 1976-04-16
JPS5734277B2 (enExample) 1982-07-22
JPS5547686A (en) 1980-04-04
DE2237592A1 (de) 1973-02-15
GB1389435A (en) 1975-04-03
CH574444A5 (enExample) 1976-04-15
GB1389437A (en) 1975-04-03
DE2237592C2 (de) 1985-08-14
GB1389434A (en) 1975-04-03
CH584206A5 (enExample) 1977-01-31
JPS5732066B2 (enExample) 1982-07-08
CH591488A5 (enExample) 1977-09-30
FR2150732A1 (enExample) 1973-04-13
AU4467372A (en) 1974-01-24
ZA724880B (en) 1973-06-27
AU461139B2 (en) 1975-05-15
JPS5714351B1 (enExample) 1982-03-24

Similar Documents

Publication Publication Date Title
BE783273A (fr) Nouvelles triazolobenzodiazepines et leur
BE810310A (fr) 4-phenylpiperidines et leur preparation
BE779390A (fr) Nouvelles pyridazinones et leur preparation
BE795907A (fr) 2-amino-4-arylthiazoles 5-substitues et leur preparation
BE808681A (fr) Nouvelles penicillines et leur preparation
BE820163A (fr) Triazolopyridazines et leur preparation
BE800781A (fr) Oxathiazinones et leur preparation
BE797101A (fr) Chlorothiazoles et leur preparation
FR2285891A1 (fr) Nouvelles benzodiazepines et leur preparation
BE787251A (fr) Nouvelles benzodiazepines et leur preparation
BE783272A (fr) Triazolobenzodiazepines et leur preparation
BE792906A (fr) Aryl-cetones et leur preparation
BE768401A (fr) Nouvelles aminophenyl-cycloamidines vermifuges et leur obtention
BE778484A (fr) Hydroxy-alcoyl-amino alcoylene-amides et leur
BE782680A (fr) Nouvelles benzodiazepines substituees et leur
BE785375A (fr) Thiolincosaminides et leur preparation
BE782848A (fr) Nouvelles triazolobenzodiazepines substituees et leur preparation
BE782849A (fr) Nouvelles triazolobenzodiazepines et leur preparation
BE761438A (fr) Alpha-halo-phenylacetamides et leur preparation
BE782846A (fr) Triazolobenzodiazepines substituees et leur preparation
BE784244A (fr) Nouvelles coumarines et leur preparation
BE764456A (fr) Amino-3-cardenolides et leur preparation
BE763671A (fr) Azidosulfonylcarbanilates et leur preparation
BE791087A (fr) Oxazoles 2,4,5-trisubstitues et leur preparation
BE820256A (fr) Nouvelles phenoxyalkylamines et leur preparation

Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: THE UPJOHN CY

Effective date: 19860831