AU7950382A - Aromatic amino keto esters, pharmaceutical use - Google Patents

Aromatic amino keto esters, pharmaceutical use

Info

Publication number
AU7950382A
AU7950382A AU79503/82A AU7950382A AU7950382A AU 7950382 A AU7950382 A AU 7950382A AU 79503/82 A AU79503/82 A AU 79503/82A AU 7950382 A AU7950382 A AU 7950382A AU 7950382 A AU7950382 A AU 7950382A
Authority
AU
Australia
Prior art keywords
aromatic amino
pharmaceutical use
keto esters
amino keto
esters
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU79503/82A
Other languages
English (en)
Inventor
Dwight Allen Shamblee
David Allan Walsh
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AH Robins Co Inc
Original Assignee
AH Robins Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by AH Robins Co Inc filed Critical AH Robins Co Inc
Publication of AU7950382A publication Critical patent/AU7950382A/en
Abandoned legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/12Ketones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/222Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin with compounds having aromatic groups, e.g. dipivefrine, ibopamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • A61K31/24Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group having an amino or nitro group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C1/00Preparation of hydrocarbons from one or more compounds, none of them being a hydrocarbon
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/40Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/42Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton with carboxyl groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by saturated carbon chains
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76Ketones containing a keto group bound to a six-membered aromatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/30Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/30Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing six-membered aromatic rings
    • C07C57/32Phenylacetic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/46Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing six-membered aromatic rings and other rings, e.g. cyclohexylphenylacetic acid

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Indole Compounds (AREA)
AU79503/82A 1981-02-17 1982-01-14 Aromatic amino keto esters, pharmaceutical use Abandoned AU7950382A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23453181A 1981-02-17 1981-02-17
US234531 1981-02-17

Publications (1)

Publication Number Publication Date
AU7950382A true AU7950382A (en) 1982-08-26

Family

ID=22881752

Family Applications (1)

Application Number Title Priority Date Filing Date
AU79503/82A Abandoned AU7950382A (en) 1981-02-17 1982-01-14 Aromatic amino keto esters, pharmaceutical use

Country Status (32)

Country Link
JP (1) JPS57149256A (fr)
KR (1) KR880002289B1 (fr)
AT (1) AT387213B (fr)
AU (1) AU7950382A (fr)
BE (1) BE892156A (fr)
CA (1) CA1173852A (fr)
CH (1) CH651294A5 (fr)
DE (1) DE3204854C2 (fr)
DK (1) DK155936C (fr)
EG (1) EG15798A (fr)
ES (1) ES509622A0 (fr)
FI (1) FI73970C (fr)
FR (1) FR2499981B1 (fr)
GB (1) GB2093027B (fr)
GR (1) GR76516B (fr)
HK (1) HK90384A (fr)
HU (1) HU187644B (fr)
IE (1) IE52289B1 (fr)
IL (1) IL64724A0 (fr)
IT (1) IT1157001B (fr)
KE (1) KE3454A (fr)
LU (1) LU83928A1 (fr)
MY (1) MY8500908A (fr)
NL (1) NL8200607A (fr)
NO (1) NO160133C (fr)
NZ (1) NZ199745A (fr)
PL (1) PL139815B1 (fr)
PT (1) PT74441B (fr)
SE (1) SE453387B (fr)
SG (1) SG68584G (fr)
YU (1) YU44333B (fr)
ZA (1) ZA82697B (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4683242A (en) * 1985-10-28 1987-07-28 A. H. Robins Company, Incorporated Transdermal treatment for pain and inflammation with 2-amino-3-aroylbenzeneacetic acids, salts and esters
US5475034A (en) * 1994-06-06 1995-12-12 Alcon Laboratories, Inc. Topically administrable compositions containing 3-benzoylphenylacetic acid derivatives for treatment of ophthalmic inflammatory disorders
US6034266A (en) * 1996-03-11 2000-03-07 Fundacao Oswaldo Cruz-Fiocruz Gem-difluoro derivative of phenylacetamide and phenylacetic acid and their pharmaceutical uses
BR9600975A (pt) * 1996-03-11 1997-12-30 Fundacao Oswaldo Cruz Derivados do ácido gem-difluorfenilacético e de gem-difluorfenilacetamida processo de sua preparação e suas aplicações farmacêuticas
AR030345A1 (es) * 2000-08-14 2003-08-20 Alcon Inc Metodo de tratamiento de desordenes relacionados con angiogenesis
AR030346A1 (es) * 2000-08-14 2003-08-20 Alcon Inc Metodo de tratamiento de desordenes neurodegenerativos de la retina y cabeza de nervio optico
AU2002247284A1 (en) 2001-04-02 2002-10-15 Alcon, Inc. Method of treating ocular inflammatory and angiogenesis-related disorders using an amide derivative of flubiprofen or ketorolac
TWI358290B (en) 2004-12-02 2012-02-21 Alcon Inc Topical nepafenac formulations

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1226344A (fr) * 1967-07-31 1971-03-24
US3997368A (en) * 1975-06-24 1976-12-14 Bell Telephone Laboratories, Incorporated Elimination of stacking faults in silicon devices: a gettering process
CH577461A5 (fr) * 1975-08-13 1976-07-15 Robins Co Inc A H
FR2366015A1 (fr) * 1975-11-05 1978-04-28 Robins Co Inc A H Nouveaux acides amino-2 benzoyl-3 (5 et 6) phenylacetiques et leurs esters et sels de metaux alcalins, utiles notamment comme anti-inflammatoires, et leur procede de preparation
IL61945A (en) * 1980-02-19 1984-09-30 Robins Co Inc A H 2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
ATA43382A (de) 1988-05-15
FR2499981A1 (fr) 1982-08-20
IT8267152A0 (it) 1982-02-10
ES8301895A1 (es) 1982-12-16
DK155936B (da) 1989-06-05
NL8200607A (nl) 1982-09-16
CH651294A5 (fr) 1985-09-13
JPH0365338B2 (fr) 1991-10-11
FI73970C (fi) 1987-12-10
IL64724A0 (en) 1982-03-31
GB2093027A (en) 1982-08-25
SG68584G (en) 1985-03-15
CA1173852A (fr) 1984-09-04
DK67382A (da) 1982-08-18
SE8200891L (sv) 1982-08-18
IE820310L (en) 1982-08-17
YU44333B (en) 1990-06-30
PT74441A (en) 1982-03-01
NZ199745A (en) 1985-07-12
FR2499981B1 (fr) 1986-05-23
IE52289B1 (en) 1987-09-02
GB2093027B (en) 1984-07-04
JPS57149256A (en) 1982-09-14
ES509622A0 (es) 1982-12-16
ZA82697B (en) 1983-01-26
DE3204854C2 (de) 1994-06-16
LU83928A1 (fr) 1983-06-07
PL235095A1 (fr) 1982-11-08
HK90384A (en) 1984-11-23
DK155936C (da) 1989-11-06
KR880002289B1 (ko) 1988-10-22
DE3204854A1 (de) 1982-09-09
KE3454A (en) 1984-10-12
NO160133B (no) 1988-12-05
NO820468L (no) 1982-08-18
FI820392L (fi) 1982-08-18
EG15798A (en) 1986-06-30
IT1157001B (it) 1987-02-11
AT387213B (de) 1988-12-27
MY8500908A (en) 1985-12-31
SE453387B (sv) 1988-02-01
BE892156A (fr) 1982-06-16
KR830008990A (ko) 1983-12-16
PL139815B1 (en) 1987-02-28
GR76516B (fr) 1984-08-10
NO160133C (no) 1989-03-15
YU32582A (en) 1985-06-30
HU187644B (en) 1986-02-28
FI73970B (fi) 1987-08-31
PT74441B (pt) 1983-08-24

Similar Documents

Publication Publication Date Title
AU566510B2 (en) Pharmaceutical 1,4-benzodiazepine-2-ones
AU8171282A (en) 5 oxo-thiazolo(3,2-a)azepine-3-carboxylic acids
AU4243289A (en) Pharmaceutical formulations
AU554377B2 (en) Sustained release pharmaceutical preparations
AU1392783A (en) 1,8-naphthyridine and 1,5,8-azanaphthyridine derivatives
AU557693B2 (en) Pharmaceutical sustained release compounds
AU556373B2 (en) Stable pharmaceutical tablet
AU587925B2 (en) Hanky delivery system
AU562216B2 (en) Coated pharmaceutical preparations
AU2227483A (en) Pharmaceutical dihydropyridines
AU2201888A (en) Pharmaceutical combination
AU8148782A (en) 1alpha, 25-dihydroxy-2beta-fluorovitamin d3
AU4918790A (en) Medicament
AU561449B2 (en) Pharmaceutical 3-aryl-7-chloro-9-oxo-3,4-dihyroacridines
AU7950382A (en) Aromatic amino keto esters, pharmaceutical use
AU2345988A (en) Pharmaceutical composition for piperidinoalkanol-decongestant combination
AU563979B2 (en) Pharmaceutical azolylmethylcycloalkanes
AU587255B2 (en) Pharmaceutical tablet
AU584547B2 (en) Pharmaceutical `` -aminoalkyl- `` -alkylphenylacetonitriles
AU7984487A (en) Pharmaceutical combination
AU2065588A (en) Pharmaceutical preparations for external use
AU553100B2 (en) Caerulein-containing psychotropic drugs
AU584266B2 (en) Azoniaspironortropanol esters, processes for the preparation thereof and pharmaceutical compositions containing them
AU3298589A (en) New pharmaceutical composition
AU8559582A (en) Titanium