AU772575B2 - Procollagen C-proteinase inhibitors - Google Patents
Procollagen C-proteinase inhibitors Download PDFInfo
- Publication number
- AU772575B2 AU772575B2 AU25375/00A AU2537500A AU772575B2 AU 772575 B2 AU772575 B2 AU 772575B2 AU 25375/00 A AU25375/00 A AU 25375/00A AU 2537500 A AU2537500 A AU 2537500A AU 772575 B2 AU772575 B2 AU 772575B2
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- Australia
- Prior art keywords
- compound
- alkyl
- resin
- aralkyl
- heteroaralkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Classifications
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- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Zoology (AREA)
- Toxicology (AREA)
- Physical Education & Sports Medicine (AREA)
- Urology & Nephrology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Transplantation (AREA)
- Vascular Medicine (AREA)
- Dermatology (AREA)
- Biomedical Technology (AREA)
- Rheumatology (AREA)
- Neurology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US11166198P | 1998-12-10 | 1998-12-10 | |
| US60/111661 | 1998-12-10 | ||
| PCT/EP1999/009519 WO2000034313A1 (fr) | 1998-12-10 | 1999-12-06 | Inhibiteurs de la c-proteinase de procollagene |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2537500A AU2537500A (en) | 2000-06-26 |
| AU772575B2 true AU772575B2 (en) | 2004-04-29 |
Family
ID=22339762
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU25375/00A Ceased AU772575B2 (en) | 1998-12-10 | 1999-12-06 | Procollagen C-proteinase inhibitors |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US6426402B1 (fr) |
| EP (1) | EP1137661A1 (fr) |
| JP (1) | JP2002531576A (fr) |
| KR (1) | KR20010080709A (fr) |
| CN (1) | CN1330661A (fr) |
| AR (1) | AR021596A1 (fr) |
| AU (1) | AU772575B2 (fr) |
| BR (1) | BR9916004A (fr) |
| CA (1) | CA2352740A1 (fr) |
| TR (1) | TR200101663T2 (fr) |
| WO (1) | WO2000034313A1 (fr) |
| ZA (1) | ZA200104672B (fr) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6777217B1 (en) | 1996-03-26 | 2004-08-17 | President And Fellows Of Harvard College | Histone deacetylases, and uses related thereto |
| US20030129724A1 (en) | 2000-03-03 | 2003-07-10 | Grozinger Christina M. | Class II human histone deacetylases, and uses related thereto |
| US7244853B2 (en) | 2001-05-09 | 2007-07-17 | President And Fellows Of Harvard College | Dioxanes and uses thereof |
| US7153822B2 (en) * | 2002-01-29 | 2006-12-26 | Wyeth | Compositions and methods for modulating connexin hemichannels |
| FR2840897B1 (fr) | 2002-06-14 | 2004-09-10 | Fournier Lab Sa | Nouveaux derives d'arylsulfonamides et leur utilisation en therapeutique |
| WO2004076386A2 (fr) | 2003-02-25 | 2004-09-10 | Topotarget Uk Limited | Composes d'acide carbamique comprenant un groupe heteroaryle bicyclique utilises en tant qu'inhibiteurs de hdac |
| US20040213758A1 (en) * | 2003-04-23 | 2004-10-28 | Rimon Therapeutics Ltd. | Hydroxyamate-containing materials for the inhibition of matrix metalloproteinases |
| US20070160655A1 (en) * | 2003-04-23 | 2007-07-12 | Sefton Michael V | Hydroxyamate-containing materials for the inhibition of matrix metalloproteinases |
| US7317019B2 (en) | 2003-08-21 | 2008-01-08 | Bristol Myers Squibb Co. | N-alkylated diaminopropane derivatives as modulators of chemokine receptor activity |
| KR100629712B1 (ko) * | 2003-08-26 | 2006-09-29 | (주)아모레퍼시픽 | 항노화 효과를 나타내는 히드록삼산 유도체 및 이의제조방법 |
| CA2601706C (fr) | 2005-03-22 | 2016-09-20 | Dana-Farber Cancer Institute, Inc. | Traitement de troubles lies a la degradation de proteines |
| MX2008010462A (es) * | 2006-02-14 | 2009-04-17 | Harvard College | Inhibidores de histona desacetilasa. |
| CN101400362B (zh) | 2006-02-14 | 2016-10-12 | 哈佛大学校长及研究员协会 | 双官能组蛋白去乙酰化酶抑制剂 |
| WO2007130429A2 (fr) | 2006-05-03 | 2007-11-15 | The President And Fellows Of Harvard College | Inhibiteurs d'histone désacétylases et de tubuline désacétylases |
| WO2009097893A1 (fr) * | 2008-02-04 | 2009-08-13 | Proyecto De Biomedicina Cima, S.L. | Procédés de traitement d'une maladie cardiaque associée à une fibrose myocardique à l'aide d'un inhibiteur de pcp |
| CA2716347C (fr) * | 2008-02-21 | 2017-06-20 | Sequoia Pharmaceuticals, Inc. | Inhibiteurs aminoacides du cytochrome p450 |
| AU2009274549B2 (en) | 2008-07-23 | 2014-05-01 | Dana-Farber Cancer Institute, Inc. | Deacetylase inhibitors and uses thereof |
| EP2326619B1 (fr) | 2008-08-01 | 2019-02-27 | Bioxiness Pharmaceuticals, Inc. | Analogues de methionine, et procedes d'utilisation de ceux-ci |
| US8716344B2 (en) | 2009-08-11 | 2014-05-06 | President And Fellows Of Harvard College | Class- and isoform-specific HDAC inhibitors and uses thereof |
| CN109970797A (zh) * | 2014-01-10 | 2019-07-05 | 葛兰素史密斯克莱知识产权（第2 号）有限公司 | 羟基甲酰胺衍生物及其用途 |
| US20180362485A1 (en) * | 2015-07-09 | 2018-12-20 | Glaxosmithkline Intellectual Property (No. 2) Limited | N-HYDROXYFORMAMIDE COMPOUNDS AND COMPOSITIONS COMPRISING THEM FOR USE AS BMP l, TLL1 AND/OR TLL2 INHIBITORS |
| US9813673B2 (en) | 2016-01-20 | 2017-11-07 | Gerard Dirk Smits | Holographic video capture and telepresence system |
| CN115197102B (zh) * | 2021-04-12 | 2023-10-20 | 山东大学 | 类肽异羟肟酸类恶性疟原虫氨肽酶抑制剂及其制备方法和应用 |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0925293A (ja) * | 1995-02-14 | 1997-01-28 | Teijin Ltd | ヒスチジル−ヒドロキサム酸誘導体 |
| AU7751598A (en) * | 1997-06-11 | 1998-12-30 | Carlton And United Breweries Limited | A container for separately storing flowable materials but allowing mixing of materials when required |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IE54551B1 (en) | 1982-01-22 | 1989-11-22 | Ici Plc | Amide derivatives |
| JPH01146896A (ja) * | 1987-12-04 | 1989-06-08 | Fuji Yakuhin Kogyo Kk | 新規なペプチジルヒドロキサム酸誘導体 |
| AU2228292A (en) * | 1991-06-14 | 1993-01-12 | Research Corporation Technologies, Inc. | Peptide derivatives of collagenase inhibitor |
| JP3597863B2 (ja) * | 1993-11-05 | 2004-12-08 | ワーナー−ランバート・コンパニー | タンパク質：ファルネシルトランスフェラーゼの置換されたジ‐およびトリペプチド阻害剤 |
| US5703092A (en) * | 1995-04-18 | 1997-12-30 | The Dupont Merck Pharmaceutical Company | Hydroxamic acid compounds as metalloprotease and TNF inhibitors |
| JPH08311096A (ja) | 1995-05-18 | 1996-11-26 | Teijin Ltd | Ｍｍｐ阻害作用を有する新規なヒスチジル−ヒドロキサム酸誘導体 |
| JPH11511137A (ja) | 1995-08-08 | 1999-09-28 | ファイブロゲン，インコーポレーテッド | コラーゲンの過剰生産に関係した疾患を治療するためのｃ−プロテイナーゼ阻害剤 |
| IT1283637B1 (it) | 1996-05-14 | 1998-04-23 | Italfarmaco Spa | Composti ad attivita' antinfiammatoria ed immunosoppressiva |
| EP0994104A4 (fr) | 1996-06-27 | 2001-09-12 | Ono Pharmaceutical Co | Derives d'aryle (sulfure, oxyde sulfonique et sulfone) et medicaments les contenant en tant que principe actif |
| WO1998015525A1 (fr) | 1996-10-07 | 1998-04-16 | Sumitomo Pharmaceuticals Co., Ltd. | Acides hydroxamiques |
| AR016751A1 (es) | 1996-11-22 | 2001-08-01 | Athena Neurosciences Inc | Metodo para inhibir la liberacion del peptido beta-amiloide en una celula, composicion farmaceutica y compuestos utiles en dicho metodo |
| FR2762315B1 (fr) | 1997-04-22 | 1999-05-28 | Logeais Labor Jacques | Derives d'amino-acides inhibiteurs des metalloproteases de la matrice extracellulaire et de la liberation du tnf alpha |
| AUPO721997A0 (en) * | 1997-06-06 | 1997-07-03 | Queensland Institute Of Medical Research, The | Anticancer compounds |
-
1999
- 1999-12-06 KR KR1020017007101A patent/KR20010080709A/ko not_active Application Discontinuation
- 1999-12-06 CN CN99814311A patent/CN1330661A/zh active Pending
- 1999-12-06 WO PCT/EP1999/009519 patent/WO2000034313A1/fr not_active Application Discontinuation
- 1999-12-06 TR TR2001/01663T patent/TR200101663T2/xx unknown
- 1999-12-06 AU AU25375/00A patent/AU772575B2/en not_active Ceased
- 1999-12-06 EP EP99968338A patent/EP1137661A1/fr not_active Withdrawn
- 1999-12-06 BR BR9916004-8A patent/BR9916004A/pt not_active IP Right Cessation
- 1999-12-06 CA CA002352740A patent/CA2352740A1/fr not_active Abandoned
- 1999-12-06 JP JP2000586755A patent/JP2002531576A/ja active Pending
- 1999-12-09 AR ARP990106263A patent/AR021596A1/es unknown
- 1999-12-10 US US09/459,201 patent/US6426402B1/en not_active Expired - Fee Related
-
2001
- 2001-06-07 ZA ZA200104672A patent/ZA200104672B/en unknown
-
2002
- 2002-02-07 US US10/072,730 patent/US6951918B2/en not_active Expired - Fee Related
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0925293A (ja) * | 1995-02-14 | 1997-01-28 | Teijin Ltd | ヒスチジル−ヒドロキサム酸誘導体 |
| AU7751598A (en) * | 1997-06-11 | 1998-12-30 | Carlton And United Breweries Limited | A container for separately storing flowable materials but allowing mixing of materials when required |
Also Published As
| Publication number | Publication date |
|---|---|
| US6426402B1 (en) | 2002-07-30 |
| TR200101663T2 (tr) | 2001-11-21 |
| CN1330661A (zh) | 2002-01-09 |
| EP1137661A1 (fr) | 2001-10-04 |
| JP2002531576A (ja) | 2002-09-24 |
| AR021596A1 (es) | 2002-07-31 |
| WO2000034313A1 (fr) | 2000-06-15 |
| US20020169133A1 (en) | 2002-11-14 |
| KR20010080709A (ko) | 2001-08-22 |
| BR9916004A (pt) | 2001-10-02 |
| US6951918B2 (en) | 2005-10-04 |
| ZA200104672B (en) | 2002-09-09 |
| AU2537500A (en) | 2000-06-26 |
| CA2352740A1 (fr) | 2000-06-15 |
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