AU604512B2 - Octahydrobenzo(g)quinoline-3beta-carbonyl derivatives useful as dopamine receptor stimulating and prolactin secretion inhibiting agents - Google Patents

Octahydrobenzo(g)quinoline-3beta-carbonyl derivatives useful as dopamine receptor stimulating and prolactin secretion inhibiting agents Download PDF

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Publication number
AU604512B2
AU604512B2 AU81409/87A AU8140987A AU604512B2 AU 604512 B2 AU604512 B2 AU 604512B2 AU 81409/87 A AU81409/87 A AU 81409/87A AU 8140987 A AU8140987 A AU 8140987A AU 604512 B2 AU604512 B2 AU 604512B2
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AU
Australia
Prior art keywords
compound
formula
addition salt
free base
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU81409/87A
Other languages
English (en)
Other versions
AU8140987A (en
Inventor
Cyril Mahaim
Christos Papageorgiou
Trevor James Petcher
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sandoz AG
Original Assignee
Sandoz AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz AG filed Critical Sandoz AG
Publication of AU8140987A publication Critical patent/AU8140987A/en
Application granted granted Critical
Publication of AU604512B2 publication Critical patent/AU604512B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/08—Aza-anthracenes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU81409/87A 1986-11-21 1987-11-19 Octahydrobenzo(g)quinoline-3beta-carbonyl derivatives useful as dopamine receptor stimulating and prolactin secretion inhibiting agents Ceased AU604512B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3639855 1986-11-21
DE3639855 1986-11-21

Publications (2)

Publication Number Publication Date
AU8140987A AU8140987A (en) 1988-05-26
AU604512B2 true AU604512B2 (en) 1990-12-20

Family

ID=6314490

Family Applications (1)

Application Number Title Priority Date Filing Date
AU81409/87A Ceased AU604512B2 (en) 1986-11-21 1987-11-19 Octahydrobenzo(g)quinoline-3beta-carbonyl derivatives useful as dopamine receptor stimulating and prolactin secretion inhibiting agents

Country Status (22)

Country Link
JP (1) JPS63150264A (cg-RX-API-DMAC7.html)
KR (1) KR880006200A (cg-RX-API-DMAC7.html)
AT (1) AT393836B (cg-RX-API-DMAC7.html)
AU (1) AU604512B2 (cg-RX-API-DMAC7.html)
BE (1) BE1003219A3 (cg-RX-API-DMAC7.html)
CH (1) CH677668A5 (cg-RX-API-DMAC7.html)
DK (1) DK608787A (cg-RX-API-DMAC7.html)
ES (1) ES2011309A6 (cg-RX-API-DMAC7.html)
FI (1) FI875130A7 (cg-RX-API-DMAC7.html)
FR (1) FR2607134A1 (cg-RX-API-DMAC7.html)
GB (1) GB2198129B (cg-RX-API-DMAC7.html)
GR (1) GR871777B (cg-RX-API-DMAC7.html)
HU (1) HUT47914A (cg-RX-API-DMAC7.html)
IL (1) IL84538A (cg-RX-API-DMAC7.html)
IT (1) IT1211920B (cg-RX-API-DMAC7.html)
LU (1) LU87047A1 (cg-RX-API-DMAC7.html)
NL (1) NL8702680A (cg-RX-API-DMAC7.html)
NZ (1) NZ222612A (cg-RX-API-DMAC7.html)
PH (1) PH25125A (cg-RX-API-DMAC7.html)
PT (1) PT86178B (cg-RX-API-DMAC7.html)
SE (1) SE8704551L (cg-RX-API-DMAC7.html)
ZA (1) ZA878717B (cg-RX-API-DMAC7.html)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1990000896A1 (en) * 1988-07-22 1990-02-08 Sandoz Ag USE OF BENZO(g)QUINOLINES IN TREATMENT OF NICOTINE ADDICTION
TW357143B (en) * 1995-07-07 1999-05-01 Novartis Ag Benzo[g]quinoline derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4526892A (en) * 1981-03-03 1985-07-02 Farmitalia Carlo Erba, S.P.A. Dimethylaminoalkyl-3-(ergoline-8'βcarbonyl)-ureas
EP0077754B1 (en) * 1981-10-16 1990-09-26 Sandoz Ag Novel pharmaceutically active 1,2,3,4,4a,5,10,10a-octahydrobenzo(g)quinoline derivatives
GB8602372D0 (en) * 1986-01-31 1986-03-05 Sandoz Ltd Organic compounds

Also Published As

Publication number Publication date
SE8704551D0 (sv) 1987-11-19
ATA306187A (de) 1991-06-15
IT1211920B (it) 1989-11-08
HUT47914A (en) 1989-04-28
GB2198129A (en) 1988-06-08
CH677668A5 (cg-RX-API-DMAC7.html) 1991-06-14
ES2011309A6 (es) 1990-01-01
AT393836B (de) 1991-12-27
PT86178A (en) 1987-12-01
DK608787A (da) 1988-05-22
IT8748620A0 (it) 1987-11-18
JPS63150264A (ja) 1988-06-22
SE8704551L (sv) 1988-05-22
NZ222612A (en) 1991-07-26
BE1003219A3 (fr) 1992-02-04
FR2607134A1 (fr) 1988-05-27
IL84538A (en) 1991-12-12
NL8702680A (nl) 1988-06-16
FI875130A7 (fi) 1988-05-22
AU8140987A (en) 1988-05-26
ZA878717B (en) 1989-06-28
KR880006200A (ko) 1988-07-22
PT86178B (pt) 1990-11-07
GB2198129B (en) 1990-08-08
IL84538A0 (en) 1988-04-29
DK608787D0 (da) 1987-11-19
GB8727057D0 (en) 1987-12-23
FI875130A0 (fi) 1987-11-19
PH25125A (en) 1991-02-19
LU87047A1 (fr) 1988-06-13
GR871777B (en) 1988-03-24

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