AU570431B2 - Benzamide derivatives - Google Patents

Benzamide derivatives

Info

Publication number
AU570431B2
AU570431B2 AU25066/84A AU2506684A AU570431B2 AU 570431 B2 AU570431 B2 AU 570431B2 AU 25066/84 A AU25066/84 A AU 25066/84A AU 2506684 A AU2506684 A AU 2506684A AU 570431 B2 AU570431 B2 AU 570431B2
Authority
AU
Australia
Prior art keywords
benzamide derivatives
benzamide
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU25066/84A
Other languages
English (en)
Other versions
AU2506684A (en
Inventor
Renato Joos
Emilio Kyburz
Mose Da Prada
Pierre-Charles Wyss
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of AU2506684A publication Critical patent/AU2506684A/en
Application granted granted Critical
Publication of AU570431B2 publication Critical patent/AU570431B2/en
Assigned to F. HOFFMANN-LA ROCHE AG reassignment F. HOFFMANN-LA ROCHE AG Alteration of Name(s) in Register under S187 Assignors: F. HOFFMANN-LA ROCHE AG
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/77—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU25066/84A 1983-03-03 1984-02-27 Benzamide derivatives Ceased AU570431B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH1150/83 1983-03-03
CH1150/83A CH653670A5 (de) 1983-03-03 1983-03-03 Benzamid-derivate.

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU83079/87A Division AU609758B2 (en) 1983-03-03 1987-12-24 Benzamide derivatives

Publications (2)

Publication Number Publication Date
AU2506684A AU2506684A (en) 1984-09-06
AU570431B2 true AU570431B2 (en) 1988-03-17

Family

ID=4203649

Family Applications (2)

Application Number Title Priority Date Filing Date
AU25066/84A Ceased AU570431B2 (en) 1983-03-03 1984-02-27 Benzamide derivatives
AU83079/87A Ceased AU609758B2 (en) 1983-03-03 1987-12-24 Benzamide derivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU83079/87A Ceased AU609758B2 (en) 1983-03-03 1987-12-24 Benzamide derivatives

Country Status (28)

Country Link
JP (1) JPS59167552A (de)
KR (1) KR910008202B1 (de)
AR (1) AR243155A1 (de)
AT (1) AT390948B (de)
AU (2) AU570431B2 (de)
BE (1) BE899059A (de)
CA (1) CA1252794A (de)
CH (1) CH653670A5 (de)
DE (1) DE3407654C2 (de)
DK (1) DK166382C (de)
ES (3) ES8504680A1 (de)
FI (1) FI79297C (de)
FR (1) FR2541996B1 (de)
GB (1) GB2135998B (de)
GR (1) GR81866B (de)
HU (1) HU193556B (de)
IE (1) IE57004B1 (de)
IL (1) IL71078A (de)
IT (1) IT1173365B (de)
LU (1) LU85231A1 (de)
MC (1) MC1568A1 (de)
NL (1) NL8400459A (de)
NO (1) NO165999C (de)
NZ (1) NZ207272A (de)
PH (1) PH19623A (de)
PT (1) PT78187B (de)
SE (1) SE466447B (de)
ZA (1) ZA841394B (de)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU589921B2 (en) * 1984-11-23 1989-10-26 Novartis Ag N-(2-dialkylaminoethyl) benzamides process for their manufacture and their pharmaceutical use

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1261335A (en) * 1984-08-29 1989-09-26 Hoffmann-La Roche Limited/Hoffmann-La Roche Limitee Ethylenediamine monoamide derivatives
NZ219974A (en) * 1986-04-22 1989-08-29 Goedecke Ag N-(2'-aminophenyl)-benzamide derivatives, process for their preparation and their use in the control of neoplastic diseases
FR2642972B1 (fr) * 1989-02-14 1994-08-05 Inst Nat Sante Rech Med Agents pour le diagnostic et le traitement des melanomes, derives halogenes aromatiques utilisables comme de tels agents et leur preparation
WO2014155184A1 (en) * 2013-03-28 2014-10-02 Rhenovia Pharma Treatment for parkinson's disease

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0083729A1 (de) * 1982-01-07 1983-07-20 Chemie Linz Aktiengesellschaft Substituierte 1-Benzoyl-2-phenylimino-imidazolidine, deren Säureadditionssalze, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel
AU546777B2 (en) * 1983-01-03 1985-09-19 Miles Laboratories Inc. Procainamide/n-acetyl derivatives thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3342679A (en) * 1967-09-19 Parts by weight of acid chloride to react with parts of amine in
FR6557M (de) * 1967-06-20 1968-12-23 Ile De France
GB1455116A (en) * 1972-12-15 1976-11-10 Ici Ltd Pharmaceutical compositions
GB1520584A (en) * 1975-04-02 1978-08-09 Yamanouchi Pharma Co Ltd 2 - alkoxy - 5 substituted benzamide derivatives and their use in pharmaceutical compositions
DE2616486A1 (de) * 1976-04-14 1977-11-03 Basf Ag Farbstoffe der perylentetracarbonsaeurediimidreihe
CA1206964A (en) * 1980-11-12 1986-07-02 Nobuo Shinma Tetra-substituted benzene derivatives
US4808624A (en) * 1984-06-28 1989-02-28 Bristol-Myers Company Pharmacologically active substituted benzamides

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0083729A1 (de) * 1982-01-07 1983-07-20 Chemie Linz Aktiengesellschaft Substituierte 1-Benzoyl-2-phenylimino-imidazolidine, deren Säureadditionssalze, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel
AU546777B2 (en) * 1983-01-03 1985-09-19 Miles Laboratories Inc. Procainamide/n-acetyl derivatives thereof

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU589921B2 (en) * 1984-11-23 1989-10-26 Novartis Ag N-(2-dialkylaminoethyl) benzamides process for their manufacture and their pharmaceutical use

Also Published As

Publication number Publication date
DK147584D0 (da) 1984-02-29
AU2506684A (en) 1984-09-06
DK166382B (da) 1993-05-10
FR2541996A1 (fr) 1984-09-07
PT78187B (en) 1986-08-05
GB2135998A (en) 1984-09-12
AU609758B2 (en) 1991-05-09
KR910008202B1 (ko) 1991-10-11
NZ207272A (en) 1987-07-31
SE466447B (sv) 1992-02-17
NO165999C (no) 1991-05-15
FI840734A0 (fi) 1984-02-22
FI79297C (fi) 1989-12-11
DE3407654A1 (de) 1984-09-06
ES530230A0 (es) 1985-05-01
FI840734A (fi) 1984-09-04
ES8506601A1 (es) 1985-08-16
DK166382C (da) 1993-09-27
LU85231A1 (de) 1985-09-12
NO840797L (no) 1984-09-04
PH19623A (de) 1986-06-04
DK147584A (da) 1984-09-04
ATA72484A (de) 1990-01-15
KR840009077A (ko) 1984-12-24
GB8405486D0 (en) 1984-04-04
ES8504680A1 (es) 1985-05-01
PT78187A (en) 1984-04-01
DE3407654C2 (de) 1994-04-07
IE57004B1 (en) 1992-03-11
IE840512L (en) 1984-09-03
AR243155A1 (es) 1993-07-30
CA1252794A (en) 1989-04-18
IL71078A0 (en) 1984-05-31
ES537045A0 (es) 1985-08-16
IT8419778A0 (it) 1984-02-23
CH653670A5 (de) 1986-01-15
MC1568A1 (fr) 1985-02-04
IT1173365B (it) 1987-06-24
SE8401190L (sv) 1984-09-04
JPS59167552A (ja) 1984-09-21
NO165999B (no) 1991-02-04
AU8307987A (en) 1988-06-16
HU193556B (en) 1987-10-28
FR2541996B1 (fr) 1987-12-11
NL8400459A (nl) 1984-10-01
ES537046A0 (es) 1985-08-16
IL71078A (en) 1987-12-31
GB2135998B (en) 1986-09-24
ZA841394B (en) 1985-06-26
SE8401190D0 (sv) 1984-03-02
ES8506600A1 (es) 1985-08-16
GR81866B (de) 1984-12-12
BE899059A (fr) 1984-09-03
FI79297B (fi) 1989-08-31
AT390948B (de) 1990-07-25
JPH0430389B2 (de) 1992-05-21

Similar Documents

Publication Publication Date Title
AU2290088A (en) Halogen-aniline derivatives
AU567140B2 (en) Sulphonamido-benzamide derivatives
AU571494B2 (en) 1- phenyl-2-azole-ethylamino-carbonyl derivatives
AU2951884A (en) Tetrahydropyridazinone derivatives
AU3320184A (en) Pyridoinole derivatives
AU2983384A (en) Spirosuccinimide derivatives
AU570047B2 (en) 3-phenyl-4-cyanopyrrole derivatives
AU562795B2 (en) Pyrrolo-thiazole derivatives
AU3608284A (en) Acylamino-s-triazine derivatives
AU3276284A (en) Acylindole derivatives
AU565020B2 (en) 1-benzazepine derivatives
AU563515B2 (en) 3-indolecarboxamide derivatives
AU3022984A (en) Formamidoxime derivatives
AU573268B2 (en) 2-azacycloalkylthiopenem derivatives
AU3668384A (en) Tetrazole-5-carboxamide derivatives
AU570431B2 (en) Benzamide derivatives
AU2559584A (en) 2-cyano-imidazopyridine derivatives
AU3492584A (en) Phenylethanamine derivatives
AU558705B2 (en) Gonadoliberine derivatives
AU568527B2 (en) Carboxy-thiazolopyrimidine derivatives
AU567189B2 (en) Azolyl-tetrahydrofuran-2-ylidene-methane derivatives
AU3540584A (en) Pyrimidoisoquinoline derivatives
AU2769084A (en) Bispiperidine derivatives
AU566160B2 (en) Azolyl-tetrahydrofuran-2-ylidene-methane derivatives
AU3644984A (en) Iminomethyl-azolyl derivatives