AU2022270088A1 - Contraceptive compounds and methods - Google Patents

Contraceptive compounds and methods Download PDF

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Publication number
AU2022270088A1
AU2022270088A1 AU2022270088A AU2022270088A AU2022270088A1 AU 2022270088 A1 AU2022270088 A1 AU 2022270088A1 AU 2022270088 A AU2022270088 A AU 2022270088A AU 2022270088 A AU2022270088 A AU 2022270088A AU 2022270088 A1 AU2022270088 A1 AU 2022270088A1
Authority
AU
Australia
Prior art keywords
compound
pharmaceutically acceptable
acceptable salt
independently selected
optionally substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
AU2022270088A
Other languages
English (en)
Inventor
Narsihmulu CHERYALA
Ingrid Gunda Georg
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
University of Minnesota System
Original Assignee
University of Minnesota Twin Cities
University of Minnesota System
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by University of Minnesota Twin Cities, University of Minnesota System filed Critical University of Minnesota Twin Cities
Publication of AU2022270088A1 publication Critical patent/AU2022270088A1/en
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Orthopedics, Nursing, And Contraception (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU2022270088A 2021-05-04 2022-05-03 Contraceptive compounds and methods Pending AU2022270088A1 (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US202163184014P 2021-05-04 2021-05-04
US63/184,014 2021-05-04
US202263307943P 2022-02-08 2022-02-08
US63/307,943 2022-02-08
US202263326524P 2022-04-01 2022-04-01
US63/326,524 2022-04-01
PCT/US2022/027506 WO2022235693A1 (en) 2021-05-04 2022-05-03 Contraceptive compounds and methods

Publications (1)

Publication Number Publication Date
AU2022270088A1 true AU2022270088A1 (en) 2023-11-23

Family

ID=81854578

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2022270088A Pending AU2022270088A1 (en) 2021-05-04 2022-05-03 Contraceptive compounds and methods

Country Status (9)

Country Link
US (3) US11780828B2 (https=)
EP (1) EP4334309A1 (https=)
JP (1) JP7828661B2 (https=)
KR (1) KR20240004737A (https=)
AU (1) AU2022270088A1 (https=)
CA (1) CA3217096A1 (https=)
IL (1) IL308171A (https=)
MX (1) MX2023012958A (https=)
WO (1) WO2022235693A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7828661B2 (ja) * 2021-05-04 2026-03-12 リージェンツ オブ ザ ユニバーシティ オブ ミネソタ 避妊薬の化合物及び方法
WO2025251031A1 (en) * 2024-05-30 2025-12-04 Yourchoice Therapeutics, Inc. Contraceptive compounds and dosing for the same

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4559157A (en) 1983-04-21 1985-12-17 Creative Products Resource Associates, Ltd. Cosmetic applicator useful for skin moisturizing
LU84979A1 (fr) 1983-08-30 1985-04-24 Oreal Composition cosmetique ou pharmaceutique sous forme aqueuse ou anhydre dont la phase grasse contient un polyether oligomere et polyethers oligomeres nouveaux
US4820508A (en) 1987-06-23 1989-04-11 Neutrogena Corporation Skin protective composition
US4992478A (en) 1988-04-04 1991-02-12 Warner-Lambert Company Antiinflammatory skin moisturizing composition and method of preparing same
US4938949A (en) 1988-09-12 1990-07-03 University Of New York Treatment of damaged bone marrow and dosage units therefor
CN1255396C (zh) * 1996-03-18 2006-05-10 卫材株式会社 含有稠环的羧酸衍生物
US7105566B2 (en) * 2002-10-22 2006-09-12 Allergan, Inc. Methods of treatment during vascular procedures
AU2015365738B2 (en) * 2014-12-19 2020-07-23 Galderma Research & Development Novel compounds, synthesis method thereof and use of same in medicine and in cosmetics
WO2017201200A1 (en) * 2016-05-19 2017-11-23 Orphagen Pharmaceuticals, Inc. Therapeutic compositions containing rar-alpha antagonists
WO2019014468A1 (en) * 2017-07-13 2019-01-17 Io Therapeutics, Inc. RECEPTOR SUBTYPE AND RETINOID COMPOUNDS AND SELECTIVE REXINOIDS OF A FUNCTION IN COMBINATION WITH IMMUNE MODULATORS FOR ANTICANCER IMMUNOTHERAPY
EP3709990A4 (en) * 2017-11-17 2021-12-01 The Regents of the University of California MANIPULATION OF THE RETIC ACID SIGNAL PATH
JP7828661B2 (ja) * 2021-05-04 2026-03-12 リージェンツ オブ ザ ユニバーシティ オブ ミネソタ 避妊薬の化合物及び方法

Also Published As

Publication number Publication date
US20250276962A1 (en) 2025-09-04
US20220388993A1 (en) 2022-12-08
US12281105B2 (en) 2025-04-22
EP4334309A1 (en) 2024-03-13
KR20240004737A (ko) 2024-01-11
CA3217096A1 (en) 2022-11-10
JP7828661B2 (ja) 2026-03-12
IL308171A (en) 2023-12-01
MX2023012958A (es) 2024-01-05
JP2024516023A (ja) 2024-04-11
US11780828B2 (en) 2023-10-10
US20240109872A1 (en) 2024-04-04
WO2022235693A1 (en) 2022-11-10

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