AU2016353547B9 - Cyclic peptides targeting α4β7 integrin - Google Patents

Cyclic peptides targeting α4β7 integrin Download PDF

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AU2016353547B9
AU2016353547B9 AU2016353547A AU2016353547A AU2016353547B9 AU 2016353547 B9 AU2016353547 B9 AU 2016353547B9 AU 2016353547 A AU2016353547 A AU 2016353547A AU 2016353547 A AU2016353547 A AU 2016353547A AU 2016353547 B9 AU2016353547 B9 AU 2016353547B9
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absent
betahomolys
aminomethyl
phe
phenyl
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AU2016353547A1 (en
AU2016353547B2 (en
Inventor
Sai Kumar Chakka
James Gillard
Jennifer L. HICKEY
Adam Paul KAFAL
M. Monzur MORSHED
Narendra Patel
Marc-André Poupart
Andrew L. Roughton
Manuel Perez VAZQUEZ
Gaoqiang Yang
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University of Montreal
Zealand Pharma AS
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University of Montreal
Zealand Pharma AS
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    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
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    • C07K1/1072—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups
    • C07K1/1075—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups by covalent attachment of amino acids or peptide residues
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AU2016353547A 2015-11-11 2016-11-14 Cyclic peptides targeting α4β7 integrin Active AU2016353547B9 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562254003P 2015-11-11 2015-11-11
US62/254,003 2015-11-11
PCT/CA2016/000274 WO2017079820A1 (en) 2015-11-11 2016-11-14 CYCLIC PEPTIDES TARGETING α4β7 INTEGRIN

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AU2016353547A1 AU2016353547A1 (en) 2018-06-28
AU2016353547B2 AU2016353547B2 (en) 2020-08-06
AU2016353547B9 true AU2016353547B9 (en) 2020-12-03

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US (4) US11072616B2 (enExample)
EP (2) EP3377471A4 (enExample)
JP (1) JP6961586B2 (enExample)
KR (1) KR102867019B1 (enExample)
CN (2) CN109071430A (enExample)
AU (1) AU2016353547B9 (enExample)
CA (2) CA3004641A1 (enExample)
WO (2) WO2017079821A1 (enExample)

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EP3377471A4 (en) 2015-11-11 2019-11-20 Encycle Therapeutics, Inc. FRAGMENT SYNTHESIS OF CYCLIC PEPTIDES
EP3939989A1 (en) 2016-11-11 2022-01-19 Zealand Pharma A/S Cyclic peptides multimers targeting alpha 4beta 7 integrin
KR20200015540A (ko) * 2017-05-10 2020-02-12 인사이클 세라퓨틱스, 인코포레이티드 α4β7 인테그린을 타겟팅하는 호모데틱 사이클릭 펩타이드
CN110551178B (zh) * 2018-06-01 2020-07-21 深圳翰宇药业股份有限公司 一种含脯氨酸的首尾环肽合成方法
JP7670618B2 (ja) * 2019-03-14 2025-04-30 エフ・ホフマン－ラ・ロシュ・アクチェンゲゼルシャフト 環状ペプチド抗生物質
JP2021106565A (ja) * 2019-12-27 2021-07-29 国立大学法人 東京大学 ライブラリーの製造方法、環状ペプチド、ＦＸＩＩａ結合剤、及びＩＦＮＧＲ１結合剤
EP4101929A4 (en) * 2019-12-27 2024-05-22 The University of Tokyo BANK CONSTRUCTION METHOD, CYCLIC PEPTIDE, FXIIA BINDER AND IFNGR1 BINDER
TWI908822B (zh) 2020-06-29 2025-12-21 丹麥商西蘭製藥公司 化合物
KR20240116921A (ko) 2021-12-20 2024-07-30 질랜드 파마 에이/에스 화합물
WO2026018016A1 (en) * 2024-07-19 2026-01-22 C4X Discovery Limited Therapeutic compounds
WO2026018017A1 (en) * 2024-07-19 2026-01-22 C4X Discovery Limited Therapeutic compounds

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