AU2013243353B2 - Fused cyclopentyl antagonists of CCR2 - Google Patents

Fused cyclopentyl antagonists of CCR2 Download PDF

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Publication number
AU2013243353B2
AU2013243353B2 AU2013243353A AU2013243353A AU2013243353B2 AU 2013243353 B2 AU2013243353 B2 AU 2013243353B2 AU 2013243353 A AU2013243353 A AU 2013243353A AU 2013243353 A AU2013243353 A AU 2013243353A AU 2013243353 B2 AU2013243353 B2 AU 2013243353B2
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compound
alkyl
formula
salt
product
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AU2013243353A1 (en
Inventor
Shawn Branum
Nagy E. Fawzy
Fu-An Kang
Michael Reuman
Ronald K. Russell
Zhihua Sui
Christopher A. Teleha
Michael P. Winters
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Janssen Pharmaceutica NV
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AU2013243353A 2012-04-06 2013-04-05 Fused cyclopentyl antagonists of CCR2 Ceased AU2013243353B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261621138P 2012-04-06 2012-04-06
US61/621,138 2012-04-06
PCT/US2013/035396 WO2013152269A1 (en) 2012-04-06 2013-04-05 Fused cyclopentyl antagonists of ccr2

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AU2013243353A1 AU2013243353A1 (en) 2014-10-02
AU2013243353B2 true AU2013243353B2 (en) 2017-07-20

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AU2013243353A Ceased AU2013243353B2 (en) 2012-04-06 2013-04-05 Fused cyclopentyl antagonists of CCR2

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US (2) US8822460B2 (enExample)
EP (1) EP2834234B1 (enExample)
JP (2) JP6110474B2 (enExample)
CN (1) CN104619702B (enExample)
AU (1) AU2013243353B2 (enExample)
CA (1) CA2869647A1 (enExample)
ES (1) ES2648175T3 (enExample)
HK (1) HK1210150A1 (enExample)
WO (1) WO2013152269A1 (enExample)

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US8822460B2 (en) * 2012-04-06 2014-09-02 Janssen Pharmaceutica Nv Fused cyclopentyl antagonists of CCR2
EP2875023B1 (en) * 2012-07-19 2017-04-05 Janssen Pharmaceutica NV Octahydro-cyclopentapyrrolyl antagonists of ccr2
EP3613435A1 (en) 2015-01-28 2020-02-26 Universite De Bordeaux Chemokine receptor cxcr4 inhibitors for treating and/or preventing chronic obstructive pulmonary disease
RS62809B1 (sr) 2015-05-21 2022-02-28 Chemocentryx Inc Modulatori ccr2
CN106366091A (zh) * 2016-08-24 2017-02-01 河北艾林国际贸易有限公司 海南霉素及其衍生物的用途及其海南霉素衍生物和制备方法
US11304952B2 (en) 2017-09-25 2022-04-19 Chemocentryx, Inc. Combination therapy using a chemokine receptor 2 (CCR2) antagonist and a PD-1/PD-L1 inhibitor
EP3737367B1 (en) 2018-01-08 2024-10-02 ChemoCentryx, Inc. Ccr2 antagonists for the treatment of cutaneous t-cell lymphoma
US20190269664A1 (en) 2018-01-08 2019-09-05 Chemocentryx, Inc. Methods of treating solid tumors with ccr2 antagonists
EP3833762A4 (en) 2018-08-09 2022-09-28 Verseau Therapeutics, Inc. Oligonucleotide compositions for targeting ccr2 and csf1r and uses thereof
CN110028469B (zh) * 2019-04-28 2022-08-09 南京药石科技股份有限公司 一种非阿片类镇痛药的关键中间体的制备方法及应用
TW202300150A (zh) 2021-03-18 2023-01-01 美商薛定諤公司 環狀化合物及其使用方法

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EP2834234A1 (en) 2015-02-11
CN104619702A (zh) 2015-05-13
CA2869647A1 (en) 2013-10-10
JP6110474B2 (ja) 2017-04-05
US9150532B2 (en) 2015-10-06
EP2834234B1 (en) 2017-09-13
AU2013243353A1 (en) 2014-10-02
US20140018356A1 (en) 2014-01-16
CN104619702B (zh) 2017-09-15
WO2013152269A1 (en) 2013-10-10
US20150080588A1 (en) 2015-03-19
JP2015516968A (ja) 2015-06-18
ES2648175T3 (es) 2017-12-28
US8822460B2 (en) 2014-09-02
JP2017095499A (ja) 2017-06-01
HK1210150A1 (en) 2016-04-15

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