AU2010329998B2 - Novel 24-membered cyclooctadepsipeptides from fungal strains and their use as anthelmintics or endoparasiticides - Google Patents

Novel 24-membered cyclooctadepsipeptides from fungal strains and their use as anthelmintics or endoparasiticides Download PDF

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Publication number
AU2010329998B2
AU2010329998B2 AU2010329998A AU2010329998A AU2010329998B2 AU 2010329998 B2 AU2010329998 B2 AU 2010329998B2 AU 2010329998 A AU2010329998 A AU 2010329998A AU 2010329998 A AU2010329998 A AU 2010329998A AU 2010329998 B2 AU2010329998 B2 AU 2010329998B2
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AU
Australia
Prior art keywords
xrb
cyclooctadepsipeptides
cyclooctadepsipeptide
fungal strains
esi
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Ceased
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AU2010329998A
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English (en)
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AU2010329998A1 (en
Inventor
Dietrich Ewald
Achim Harder
Thanh Dam Huynh
Klemens Krieger
Clemens Mugge
Thi Lam Huong Pham
Hardy Weisshoff
Irmtraut Zaspel
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Bayer Intellectual Property GmbH
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Bayer Intellectual Property GmbH
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Ceased legal-status Critical Current
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
AU2010329998A 2009-12-11 2010-12-07 Novel 24-membered cyclooctadepsipeptides from fungal strains and their use as anthelmintics or endoparasiticides Ceased AU2010329998B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09178799 2009-12-11
EP09178799.4 2009-12-11
PCT/EP2010/069040 WO2011069995A1 (en) 2009-12-11 2010-12-07 Novel 24-membered cyclooctadepsipeptides from fungal strains and their use as anthelmintics or endoparasiticides

Publications (2)

Publication Number Publication Date
AU2010329998A1 AU2010329998A1 (en) 2012-07-05
AU2010329998B2 true AU2010329998B2 (en) 2015-05-21

Family

ID=43480707

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2010329998A Ceased AU2010329998B2 (en) 2009-12-11 2010-12-07 Novel 24-membered cyclooctadepsipeptides from fungal strains and their use as anthelmintics or endoparasiticides

Country Status (8)

Country Link
US (1) US20120302496A1 (enExample)
EP (1) EP2509967B1 (enExample)
JP (1) JP5779787B2 (enExample)
AR (1) AR079341A1 (enExample)
AU (1) AU2010329998B2 (enExample)
TW (1) TW201138799A (enExample)
UY (1) UY33095A (enExample)
WO (1) WO2011069995A1 (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104540845B (zh) * 2012-06-13 2018-01-26 明治制果药业株式会社 新的环缩酚酸肽衍生物以及含有它的有害生物防除剂
WO2015093558A1 (ja) * 2013-12-18 2015-06-25 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 環状デプシペプチド誘導体およびそれを含んでなる有害生物防除剤
CN107835818B (zh) 2015-05-20 2022-04-29 勃林格殷格翰动物保健美国公司 驱虫缩酚酸肽化合物
KR20220003663A (ko) 2015-12-28 2022-01-10 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 구충성 뎁시펩티드 화합물
EP3541789A1 (en) 2016-11-16 2019-09-25 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
CN106749569B (zh) * 2017-03-03 2021-10-15 重庆乾泰生物医药有限公司 一种pf1022a的分离纯化方法
CN108570016B (zh) * 2017-03-10 2021-11-26 上海医药工业研究院 一种pf1022a分离纯化的方法
CN106978353B (zh) * 2017-03-10 2019-10-18 广东省微生物研究所 特氏炭角菌及其栽培方法
CN113943350B (zh) * 2021-11-02 2023-08-15 海南大学三亚南繁研究院 一种环肽化合物或其药学上可接受的盐及其制备方法和应用、药物及其应用
CN114875093B (zh) * 2022-05-20 2024-07-19 浙江海正药业股份有限公司 一种提高pf1022a发酵产量的方法
WO2025149943A1 (en) * 2024-01-09 2025-07-17 Animol Discovery, Inc. Antiparasitic cyclic depsipeptides

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO176766C (no) 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
JP3207870B2 (ja) * 1991-04-15 2001-09-10 明治製菓株式会社 環状デプシペプチドおよびその製造法
JP2873894B2 (ja) * 1992-10-19 1999-03-24 明治製菓株式会社 環状デプシペプチドおよびその製造法
DE4317432A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4341992A1 (de) 1993-12-09 1995-06-14 Bayer Ag Endoparasitizide Mittel auf Basis von offenkettigen Tetradepsipeptiden
WO1998005655A1 (en) 1996-08-07 1998-02-12 Meiji Seika Kaisha, Ltd. Process for producing cyclodepsipeptide compounds and novel cyclodepsipeptide
AU2009331930A1 (en) * 2008-12-16 2011-06-30 Bayer Animal Health Gmbh Method for producing optically active, cyclic depsipeptides comprising lactic acid and phenyl lactic acid and having 24 ring atoms, using fungus strains of Rosellinia type, and further species of Xylariaceae
US9209940B2 (en) 2009-03-16 2015-12-08 Lg Electronics Inc. Method of retransmission for supporting MIMO in synchronous HARQ

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
SUZUKI A ET AL, TETRAHEDRON LETTERS, vol. 18, no. 25, pages 2167-2170 *

Also Published As

Publication number Publication date
AU2010329998A1 (en) 2012-07-05
JP2013513567A (ja) 2013-04-22
AR079341A1 (es) 2012-01-18
EP2509967B1 (en) 2016-02-17
US20120302496A1 (en) 2012-11-29
JP5779787B2 (ja) 2015-09-16
EP2509967A1 (en) 2012-10-17
TW201138799A (en) 2011-11-16
WO2011069995A1 (en) 2011-06-16
UY33095A (es) 2011-07-29

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