AU2010300421B2 - Olopatadine compositions and uses thereof - Google Patents
Olopatadine compositions and uses thereof Download PDFInfo
- Publication number
- AU2010300421B2 AU2010300421B2 AU2010300421A AU2010300421A AU2010300421B2 AU 2010300421 B2 AU2010300421 B2 AU 2010300421B2 AU 2010300421 A AU2010300421 A AU 2010300421A AU 2010300421 A AU2010300421 A AU 2010300421A AU 2010300421 B2 AU2010300421 B2 AU 2010300421B2
- Authority
- AU
- Australia
- Prior art keywords
- solution composition
- olopatadine
- group
- pde4 inhibitor
- concentration
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
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Classifications
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A61P37/00—Drugs for immunological or allergic disorders
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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- Engineering & Computer Science (AREA)
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- Dermatology (AREA)
- Ophthalmology & Optometry (AREA)
- Otolaryngology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
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| US24761809P | 2009-10-01 | 2009-10-01 | |
| US61/247,618 | 2009-10-01 | ||
| PCT/US2010/051062 WO2011041640A1 (en) | 2009-10-01 | 2010-10-01 | Olopatadine compositions and uses thereof |
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| AU2010300421A1 AU2010300421A1 (en) | 2012-04-12 |
| AU2010300421B2 true AU2010300421B2 (en) | 2014-01-23 |
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Country Status (13)
| Country | Link |
|---|---|
| US (2) | US20110082145A1 (https=) |
| EP (1) | EP2482798A1 (https=) |
| JP (1) | JP5721722B2 (https=) |
| KR (1) | KR20120091037A (https=) |
| CN (1) | CN102548536A (https=) |
| AU (1) | AU2010300421B2 (https=) |
| BR (1) | BR112012007091A2 (https=) |
| CA (1) | CA2773483A1 (https=) |
| CL (1) | CL2012000801A1 (https=) |
| MX (1) | MX2012003693A (https=) |
| PH (1) | PH12012500654A1 (https=) |
| RU (1) | RU2012117141A (https=) |
| WO (1) | WO2011041640A1 (https=) |
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| TWI544922B (zh) * | 2011-05-19 | 2016-08-11 | 愛爾康研究有限公司 | 高濃度歐羅派特錠（ｏｌｏｐａｔａｄｉｎｅ）眼用組成物 |
| CN103202833A (zh) * | 2012-12-25 | 2013-07-17 | 常州市亚邦医药研究所有限公司 | 一种奥洛他定或其盐的药用组合物及其制备方法 |
| US10758550B2 (en) | 2013-10-04 | 2020-09-01 | Glenmark Specialty S.A. | Treatment of allergic rhinitis using a combination of mometasone and olopatadine |
| EP3037094A1 (en) * | 2014-12-23 | 2016-06-29 | Poifa Warszawa SA | Ophthalmic pharmaceutical composition |
| CN110117271A (zh) * | 2018-02-06 | 2019-08-13 | 中国科学院上海药物研究所 | 四氢异喹啉类化合物、其制备方法、包含此类化合物的药物组合物及其用途 |
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2010
- 2010-10-01 US US12/896,056 patent/US20110082145A1/en not_active Abandoned
- 2010-10-01 EP EP10762842A patent/EP2482798A1/en not_active Withdrawn
- 2010-10-01 MX MX2012003693A patent/MX2012003693A/es not_active Application Discontinuation
- 2010-10-01 CN CN2010800434937A patent/CN102548536A/zh active Pending
- 2010-10-01 JP JP2012532346A patent/JP5721722B2/ja not_active Expired - Fee Related
- 2010-10-01 KR KR1020127008229A patent/KR20120091037A/ko not_active Withdrawn
- 2010-10-01 PH PH1/2012/500654A patent/PH12012500654A1/en unknown
- 2010-10-01 CA CA2773483A patent/CA2773483A1/en not_active Abandoned
- 2010-10-01 WO PCT/US2010/051062 patent/WO2011041640A1/en not_active Ceased
- 2010-10-01 BR BR112012007091A patent/BR112012007091A2/pt not_active IP Right Cessation
- 2010-10-01 RU RU2012117141/15A patent/RU2012117141A/ru not_active Application Discontinuation
- 2010-10-01 AU AU2010300421A patent/AU2010300421B2/en not_active Ceased
-
2012
- 2012-03-30 CL CL2012000801A patent/CL2012000801A1/es unknown
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2013
- 2013-12-17 US US14/108,432 patent/US20140107121A1/en not_active Abandoned
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| US20070142458A1 (en) * | 2001-06-27 | 2007-06-21 | Alcon, Inc. | Olopatadine formulations for topical nasal administration |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011041640A1 (en) | 2011-04-07 |
| RU2012117141A (ru) | 2013-11-10 |
| MX2012003693A (es) | 2012-04-19 |
| US20110082145A1 (en) | 2011-04-07 |
| AU2010300421A1 (en) | 2012-04-12 |
| CA2773483A1 (en) | 2011-04-07 |
| CL2012000801A1 (es) | 2012-10-19 |
| PH12012500654A1 (en) | 2012-10-22 |
| JP5721722B2 (ja) | 2015-05-20 |
| EP2482798A1 (en) | 2012-08-08 |
| JP2013506692A (ja) | 2013-02-28 |
| CN102548536A (zh) | 2012-07-04 |
| BR112012007091A2 (pt) | 2016-04-19 |
| KR20120091037A (ko) | 2012-08-17 |
| US20140107121A1 (en) | 2014-04-17 |
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