AU2010236346B2 - 4-azetidinyl-1-phenyl-cyclohexane antagonists of CCR2 - Google Patents

4-azetidinyl-1-phenyl-cyclohexane antagonists of CCR2 Download PDF

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Publication number
AU2010236346B2
AU2010236346B2 AU2010236346A AU2010236346A AU2010236346B2 AU 2010236346 B2 AU2010236346 B2 AU 2010236346B2 AU 2010236346 A AU2010236346 A AU 2010236346A AU 2010236346 A AU2010236346 A AU 2010236346A AU 2010236346 B2 AU2010236346 B2 AU 2010236346B2
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alkyl
phenyl
prepared
compound
azetidin
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AU2010236346A1 (en
Inventor
Cuifen Hou
Heather Rae Hufnagel
Dana L. Johnson
Zhihua Sui
Xuqing Zhang
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Janssen Pharmaceutica NV
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Janssen Pharmaceutica NV
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AU2010236346A 2009-04-17 2010-04-15 4-azetidinyl-1-phenyl-cyclohexane antagonists of CCR2 Ceased AU2010236346B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17030709P 2009-04-17 2009-04-17
US61/170,307 2009-04-17
PCT/US2010/031265 WO2010121046A1 (en) 2009-04-17 2010-04-15 4-azetidinyl-1-phenyl-cyclohexane antagonists of ccr2

Publications (2)

Publication Number Publication Date
AU2010236346A1 AU2010236346A1 (en) 2011-11-03
AU2010236346B2 true AU2010236346B2 (en) 2015-01-22

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AU2010236346A Ceased AU2010236346B2 (en) 2009-04-17 2010-04-15 4-azetidinyl-1-phenyl-cyclohexane antagonists of CCR2

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US (2) US20100267689A1 (enExample)
EP (1) EP2419419B1 (enExample)
JP (1) JP5675773B2 (enExample)
KR (1) KR20120006544A (enExample)
CN (1) CN102459227B (enExample)
AR (1) AR076328A1 (enExample)
AU (1) AU2010236346B2 (enExample)
BR (1) BRPI1016189A2 (enExample)
CA (1) CA2758934A1 (enExample)
ES (1) ES2528625T3 (enExample)
MX (1) MX2011010964A (enExample)
NZ (1) NZ595432A (enExample)
TW (1) TW201102377A (enExample)
WO (1) WO2010121046A1 (enExample)

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GB201617454D0 (en) * 2016-10-14 2016-11-30 Heptares Therapeutics Limited Pharmaceutical compounds
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MA50665A (fr) 2017-09-25 2020-08-05 Chemocentryx Inc Polythérapie utilisant un antagoniste du récepteur 2 de la chimiokine (ccr2) et un inhibiteur pd-1/pd-l1
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US20100267689A1 (en) 2010-10-21
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