AU2007322116B2 - Cyclohexenyl-aryl compounds for inflammation and immune-related uses - Google Patents
Cyclohexenyl-aryl compounds for inflammation and immune-related uses Download PDFInfo
- Publication number
- AU2007322116B2 AU2007322116B2 AU2007322116A AU2007322116A AU2007322116B2 AU 2007322116 B2 AU2007322116 B2 AU 2007322116B2 AU 2007322116 A AU2007322116 A AU 2007322116A AU 2007322116 A AU2007322116 A AU 2007322116A AU 2007322116 B2 AU2007322116 B2 AU 2007322116B2
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- Australia
- Prior art keywords
- optionally substituted
- methyl
- tetrahydropyridin
- phenyl
- thiazol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
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Applications Claiming Priority (3)
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| US85861006P | 2006-11-13 | 2006-11-13 | |
| US60/858,610 | 2006-11-13 | ||
| PCT/US2007/023853 WO2008063504A2 (en) | 2006-11-13 | 2007-11-12 | Cyclohexenyl-aryl compounds for inflammation and immune-related uses |
Publications (2)
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| AU2007322116A1 AU2007322116A1 (en) | 2008-05-29 |
| AU2007322116B2 true AU2007322116B2 (en) | 2013-01-10 |
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| EP (1) | EP2086326B1 (enExample) |
| JP (1) | JP5538894B2 (enExample) |
| AU (1) | AU2007322116B2 (enExample) |
| CA (1) | CA2669695C (enExample) |
| TW (1) | TWI428338B (enExample) |
| WO (1) | WO2008063504A2 (enExample) |
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| CA2640090A1 (en) * | 2006-01-25 | 2007-08-02 | Synta Pharmaceuticals Corp. | Substituted aromatic compounds for inflammation and immune-related uses |
| JP2009524683A (ja) * | 2006-01-25 | 2009-07-02 | シンタ ファーマシューティカルズ コーポレーション | 炎症および免疫関連用途のためのビニル−フェニル誘導体 |
| JP2009528273A (ja) * | 2006-01-25 | 2009-08-06 | シンタ ファーマシューティカルズ コーポレーション | 炎症および免疫関連使用用の置換ビアリール化合物 |
| CA2645434A1 (en) | 2006-03-20 | 2007-09-27 | Synta Pharmaceutical Corp. | Benzoimidazolyl-parazine compounds for inflammation and immune-related uses |
| US8779154B2 (en) * | 2006-09-26 | 2014-07-15 | Qinglin Che | Fused ring compounds for inflammation and immune-related uses |
| TWI444379B (zh) * | 2007-06-29 | 2014-07-11 | Sunesis Pharmaceuticals Inc | 有用於作為Ｒａｆ激酶抑制劑之化合物 |
| WO2009017831A1 (en) * | 2007-08-01 | 2009-02-05 | Synta Pharmaceuticals Corp. | Vinyl-aryl derivatives for inflammation and immune-related uses |
| CN101854933A (zh) | 2007-09-10 | 2010-10-06 | 钙医学公司 | 调节细胞内钙的化合物 |
| WO2009076454A2 (en) | 2007-12-12 | 2009-06-18 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| WO2010013849A1 (ja) * | 2008-08-01 | 2010-02-04 | 日本ケミファ株式会社 | Ｇｐｒ１１９作動薬 |
| US7906553B2 (en) | 2008-08-27 | 2011-03-15 | Calcimedica, Inc. | Substituted thiophene modulators of intracellular calcium |
| US8524763B2 (en) | 2008-09-22 | 2013-09-03 | Calcimedica, Inc. | Inhibitors of store operated calcium release |
| US20110118281A9 (en) * | 2008-10-01 | 2011-05-19 | Gary Bohnert | Compounds for inflammation and immune-related uses |
| US8143269B2 (en) | 2008-10-03 | 2012-03-27 | Calcimedica, Inc. | Inhibitors of store operated calcium release |
| EP2477982A4 (en) | 2009-09-16 | 2013-04-03 | Calcimedica Inc | COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM |
| US8993612B2 (en) | 2009-10-08 | 2015-03-31 | Rhizen Pharmaceuticals Sa | Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer |
| US8377970B2 (en) | 2009-10-08 | 2013-02-19 | Rhizen Pharmaceuticals Sa | Modulators of calcium release-activated calcium channel |
| JP2013511279A (ja) | 2009-11-20 | 2013-04-04 | アムジエン・インコーポレーテツド | 抗Ｏｒａｉ１抗原結合蛋白及びその使用 |
| US20190192510A1 (en) * | 2010-02-01 | 2019-06-27 | Nippon Chemiphar Co., Ltd. | Gpr119 agonist |
| US10703722B2 (en) | 2010-04-27 | 2020-07-07 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| CA2797533A1 (en) | 2010-04-27 | 2011-11-10 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| PL2563776T3 (pl) | 2010-04-27 | 2017-01-31 | Calcimedica Inc | Związki, które modulują wewnątrzkomórkowy wapń |
| WO2012027710A2 (en) | 2010-08-27 | 2012-03-01 | Calcimedica Inc. | Compounds that modulate intracellular calcium |
| US20130289071A1 (en) * | 2010-11-09 | 2013-10-31 | Synta Pharmaceuticals Corp. | Tetrazolyl-tetrahydropyridine compounds for inflammation and immune-related uses |
| US20120316182A1 (en) | 2011-06-10 | 2012-12-13 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| WO2013059677A1 (en) | 2011-10-19 | 2013-04-25 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| US9512116B2 (en) | 2012-10-12 | 2016-12-06 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| EA036265B1 (ru) | 2015-02-27 | 2020-10-20 | Кальцимедика, Инк. | Лечение панкреатита |
| CA2995094A1 (en) | 2015-08-07 | 2017-02-16 | Calcimedica, Inc. | Use of crac channel inhibitors for the treatment of stroke and traumatic brain injury |
| KR101798840B1 (ko) | 2017-05-17 | 2017-11-17 | 주식회사 레고켐 바이오사이언스 | 신규 오토탁신 저해 화합물 및 이를 함유하는 약제학적 조성물 |
| US10961242B2 (en) | 2017-05-17 | 2021-03-30 | Legochem Biosciences, Inc. | Compounds as autotaxin inhibitors and pharmaceutical compositions comprising the same |
| MX2021003094A (es) | 2018-09-14 | 2021-05-12 | Rhizen Pharmaceuticals A G | Composiciones que comprenden un inhibidor de crac y un corticosteroide y métodos de uso de estas. |
| CA3167339A1 (en) | 2020-01-13 | 2021-07-22 | Verge Analytics, Inc. | Substituted pyrazolo-pyrimidines and uses thereof |
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| US20050107399A1 (en) * | 2003-09-11 | 2005-05-19 | Kemia, Inc. | Cytokine inhibitors |
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-
2007
- 2007-11-12 WO PCT/US2007/023853 patent/WO2008063504A2/en not_active Ceased
- 2007-11-12 AU AU2007322116A patent/AU2007322116B2/en not_active Ceased
- 2007-11-12 EP EP07853118.3A patent/EP2086326B1/en not_active Not-in-force
- 2007-11-12 JP JP2009536338A patent/JP5538894B2/ja not_active Expired - Fee Related
- 2007-11-12 US US11/938,779 patent/US20080207641A1/en not_active Abandoned
- 2007-11-12 CA CA2669695A patent/CA2669695C/en not_active Expired - Fee Related
- 2007-11-13 TW TW096142793A patent/TWI428338B/zh not_active IP Right Cessation
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050107399A1 (en) * | 2003-09-11 | 2005-05-19 | Kemia, Inc. | Cytokine inhibitors |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2008063504A2 (en) | 2008-05-29 |
| JP2010509342A (ja) | 2010-03-25 |
| AU2007322116A1 (en) | 2008-05-29 |
| TWI428338B (zh) | 2014-03-01 |
| TW200829585A (en) | 2008-07-16 |
| US20080207641A1 (en) | 2008-08-28 |
| WO2008063504A3 (en) | 2008-08-28 |
| EP2086326A2 (en) | 2009-08-12 |
| JP5538894B2 (ja) | 2014-07-02 |
| CA2669695A1 (en) | 2008-05-29 |
| CA2669695C (en) | 2012-10-30 |
| EP2086326B1 (en) | 2014-01-08 |
| EP2086326A4 (en) | 2011-03-09 |
| HK1133553A1 (en) | 2010-04-01 |
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