AU2007269646A1 - Fused heterocyclic inhibitors of D-amino acid oxidase - Google Patents
Fused heterocyclic inhibitors of D-amino acid oxidase Download PDFInfo
- Publication number
- AU2007269646A1 AU2007269646A1 AU2007269646A AU2007269646A AU2007269646A1 AU 2007269646 A1 AU2007269646 A1 AU 2007269646A1 AU 2007269646 A AU2007269646 A AU 2007269646A AU 2007269646 A AU2007269646 A AU 2007269646A AU 2007269646 A1 AU2007269646 A1 AU 2007269646A1
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- Australia
- Prior art keywords
- substituted
- unsubstituted
- member selected
- alkyl
- heterocycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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- C07D515/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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- C07D—HETEROCYCLIC COMPOUNDS
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Applications Claiming Priority (7)
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| US80639106P | 2006-06-30 | 2006-06-30 | |
| US60/806,391 | 2006-06-30 | ||
| US84246506P | 2006-09-05 | 2006-09-05 | |
| US60/842,465 | 2006-09-05 | ||
| US91429307P | 2007-04-26 | 2007-04-26 | |
| US60/914,293 | 2007-04-26 | ||
| PCT/US2007/015396 WO2008005456A2 (en) | 2006-06-30 | 2007-07-02 | Fused heterocyclic inhibitors of d-amino acid oxidase |
Publications (1)
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| AU2007269646A1 true AU2007269646A1 (en) | 2008-01-10 |
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| AU2007269646A Abandoned AU2007269646A1 (en) | 2006-06-30 | 2007-07-02 | Fused heterocyclic inhibitors of D-amino acid oxidase |
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| Country | Link |
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| EP (1) | EP2057162A2 (enExample) |
| JP (1) | JP2009542683A (enExample) |
| KR (1) | KR20090024823A (enExample) |
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| BR (1) | BRPI0713216A2 (enExample) |
| CA (1) | CA2659060A1 (enExample) |
| IL (1) | IL195921A0 (enExample) |
| MX (1) | MX2008016525A (enExample) |
| WO (1) | WO2008005456A2 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| CA2551952A1 (en) | 2003-12-29 | 2005-07-21 | Sepracor Inc. | Pyrrole and pyrazole daao inhibitors |
| WO2007081542A2 (en) | 2006-01-06 | 2007-07-19 | Sepracor Inc. | Tetralone-based monoamine reuptake inhibitors |
| CA2636324C (en) | 2006-01-06 | 2012-03-20 | Sepracor Inc. | Cycloalkylamines as monoamine reuptake inhibitors |
| DK2013835T3 (en) | 2006-03-31 | 2015-12-14 | Sunovion Pharmaceuticals Inc | Preparation of chiral amides and AMINES |
| US7884124B2 (en) | 2006-06-30 | 2011-02-08 | Sepracor Inc. | Fluoro-substituted inhibitors of D-amino acid oxidase |
| US7579370B2 (en) * | 2006-06-30 | 2009-08-25 | Sepracor Inc. | Fused heterocycles |
| EP2077267A4 (en) | 2006-10-18 | 2010-04-07 | Takeda Pharmaceutical | CONDENSED HETEROCYCLIC COMPOUND |
| US7902252B2 (en) * | 2007-01-18 | 2011-03-08 | Sepracor, Inc. | Inhibitors of D-amino acid oxidase |
| RU2470011C2 (ru) | 2007-05-31 | 2012-12-20 | Сепракор Инк. | Циклоалкиламины, содержащие в качестве заместителя фенил, как ингибиторы обратного захвата моноаминов |
| AR076766A1 (es) | 2009-05-14 | 2011-07-06 | Japan Tobacco Inc | Compuestos de azetidina, composiciones farmaceuticas y su uso en el tratamiento de enfermedades autoinmunes. |
| GB201111705D0 (en) * | 2011-07-07 | 2011-08-24 | Takeda Pharmaceutical | Compounds and their use |
| JO3115B1 (ar) * | 2011-08-22 | 2017-09-20 | Takeda Pharmaceuticals Co | مركبات بيريدازينون واستخدامها كمثبطات daao |
| GB201222711D0 (en) | 2012-12-17 | 2013-01-30 | Takeda Pharmaceutical | Novel compounds |
| AU2015253099B2 (en) * | 2014-04-30 | 2019-07-18 | National Chiao Tung University | Use of known compounds as D-amino acid oxidase inhibitors |
| TW202115086A (zh) * | 2019-06-28 | 2021-04-16 | 美商輝瑞大藥廠 | Bckdk抑制劑 |
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| GB9803228D0 (en) * | 1998-02-17 | 1998-04-08 | Zeneca Ltd | Chemical compounds |
| DK1088824T3 (da) * | 1999-09-30 | 2004-04-13 | Pfizer Prod Inc | Bicykliske pyrrolylamider som glycogen phosphorylase inhibitorer |
| EP1391460A1 (en) * | 1999-09-30 | 2004-02-25 | Pfizer Products Inc. | Tricyclic pyrrolyl amides as glycogen phosphorylase inhibitors |
| US20030162825A1 (en) * | 2001-11-09 | 2003-08-28 | Sepracor Inc. | D-amino acid oxidase inhibitors for learning and memory |
| AU2003272285A1 (en) * | 2002-09-06 | 2004-03-29 | Janssen Pharmaceutica, N.V. | Thienopyrrolyl and furanopyrrolyl compounds and their use as histamine h4 receptor ligands |
| CA2551952A1 (en) * | 2003-12-29 | 2005-07-21 | Sepracor Inc. | Pyrrole and pyrazole daao inhibitors |
| CA2569530C (en) * | 2004-07-01 | 2013-07-30 | Daiichi Asubio Pharma Co.,Ltd. | Thienopyrazole derivative having pde 7 inhibitory activity |
| CA2594665A1 (en) * | 2005-01-19 | 2006-07-27 | Biolipox Ab | Thienopyrroles useful in the treatment of inflammation |
| US20090306169A1 (en) * | 2005-10-06 | 2009-12-10 | Brandish Philip E | Use of Fused Pyrrole Carboxylic Acids for the Treatment of Neurodegenerative and Psychiatric Diseases and D-Amino Acid Oxidase Inhibitors |
| UA95788C2 (en) * | 2005-12-15 | 2011-09-12 | Ф. Хоффманн-Ля Рош Аг | Fused pyrrole derivatives |
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2007
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- 2007-07-02 WO PCT/US2007/015396 patent/WO2008005456A2/en not_active Ceased
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- 2007-07-02 MX MX2008016525A patent/MX2008016525A/es not_active Application Discontinuation
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- 2007-07-02 EP EP07796659A patent/EP2057162A2/en not_active Withdrawn
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2008
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Also Published As
| Publication number | Publication date |
|---|---|
| JP2009542683A (ja) | 2009-12-03 |
| EP2057162A2 (en) | 2009-05-13 |
| IL195921A0 (en) | 2009-09-01 |
| MX2008016525A (es) | 2009-03-09 |
| WO2008005456A3 (en) | 2008-07-31 |
| CA2659060A1 (en) | 2008-01-10 |
| BRPI0713216A2 (pt) | 2012-12-04 |
| KR20090024823A (ko) | 2009-03-09 |
| WO2008005456A2 (en) | 2008-01-10 |
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