AU2006227243B2 - Dosing regimes for trans-clomiphene - Google Patents
Dosing regimes for trans-clomiphene Download PDFInfo
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- AU2006227243B2 AU2006227243B2 AU2006227243A AU2006227243A AU2006227243B2 AU 2006227243 B2 AU2006227243 B2 AU 2006227243B2 AU 2006227243 A AU2006227243 A AU 2006227243A AU 2006227243 A AU2006227243 A AU 2006227243A AU 2006227243 B2 AU2006227243 B2 AU 2006227243B2
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- Prior art keywords
- clomiphene
- testosterone
- treatment
- trans
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- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- Public Health (AREA)
- General Health & Medical Sciences (AREA)
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- Chemical & Material Sciences (AREA)
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- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Pregnancy & Childbirth (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US60/664,290 | 2005-03-22 | ||
| PCT/US2006/010022 WO2006102232A2 (en) | 2005-03-22 | 2006-03-17 | Dosing regimes for trans-clomiphene |
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| AU2006227243A1 AU2006227243A1 (en) | 2006-09-28 |
| AU2006227243B2 true AU2006227243B2 (en) | 2011-10-27 |
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| US7737185B2 (en) | 2001-07-09 | 2010-06-15 | Repros Therapeutics Inc. | Methods and compositions with trans-clomiphene |
| DK1411916T3 (da) | 2001-07-09 | 2008-12-15 | Repros Therapeutics Inc | Fremgangsmåder og materialer til behandling af testosteronmangel hos mænd |
| JP5785680B2 (ja) | 2005-03-22 | 2015-09-30 | リプロス セラピューティクス インコーポレイテッド | トランス−クロミフェン用の投与レジメン |
| MY148330A (en) | 2006-10-31 | 2013-03-29 | Basf Se | Regulation of a process for producing water-absorbing polymer particles in a heated gas phase |
| CN102940619A (zh) * | 2007-10-16 | 2013-02-27 | 利普生物药剂公司 | 用于治疗代谢综合征的珠氯米芬 |
| TW201500041A (zh) * | 2008-11-07 | 2015-01-01 | Repros Therapeutics Inc | 用於代謝症候群與第２型糖尿病的反式氯米芬 |
| UA113291C2 (xx) | 2011-08-04 | 2017-01-10 | Метаболіти транскломіфену і їх застосування | |
| WO2013020215A1 (en) * | 2011-08-09 | 2013-02-14 | Adams Kenneth W | Use of aromatase inhibitor or estrogen blocker for increasing spermatogenesis or testosterone levels in males |
| AU2013221478B2 (en) * | 2012-02-14 | 2017-06-01 | Repros Therapeutics Inc. | Selective estrogen receptor modulators with short half-lives and uses thereof |
| MX2014009322A (es) * | 2012-02-29 | 2014-11-10 | Repros Therapeutics Inc | Terapia de combinacion para el tratamiento de la deficiencia androgenica. |
| ES2701400T3 (es) | 2012-05-31 | 2019-02-22 | Repros Therapeutics Inc | Formulaciones para la administración vaginal de antiprogestinas |
| HK1211852A1 (en) | 2012-11-02 | 2016-06-03 | Repros Therapeutics Inc. | Methods and compositions for treating progesterone-dependent conditions |
| HK1216502A1 (zh) * | 2012-11-02 | 2016-11-18 | Repros Therapeutics Inc. | 用於癌症治療的反式-克羅米芬 |
| CA2914503A1 (en) * | 2013-06-05 | 2014-11-12 | Repros Therapeutics Inc. | Trans-clomiphene and its analogues as agents that increase bone mineral density |
| CN108883083A (zh) * | 2016-02-25 | 2018-11-23 | 艾森潘帕克制药股份有限公司 | 两种氯米芬异构体的口服剂型及使用其治疗继发性腺功能减退症的方法 |
| CA2989364C (en) | 2016-04-22 | 2021-07-20 | F.I.S. - Fabbrica Italiana Sintetici S.P.A. | Process for the preparation of enclomiphene citrate having needle shaped crystal habit. |
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- 2006-03-17 EP EP11153365A patent/EP2392322A3/en not_active Withdrawn
- 2006-03-17 RU RU2007138867/15A patent/RU2413508C2/ru active
- 2006-03-17 EP EP06738985A patent/EP1865938A4/en not_active Ceased
- 2006-03-17 WO PCT/US2006/010022 patent/WO2006102232A2/en not_active Ceased
- 2006-03-17 NZ NZ560551A patent/NZ560551A/en not_active IP Right Cessation
- 2006-03-17 CN CN2006800089841A patent/CN101163467B/zh not_active Expired - Fee Related
- 2006-03-17 CA CA3071412A patent/CA3071412A1/en not_active Abandoned
- 2006-03-17 PL PL383444A patent/PL383444A1/pl unknown
- 2006-03-17 US US11/815,542 patent/US8247456B2/en not_active Expired - Fee Related
- 2006-03-17 CA CA002597700A patent/CA2597700A1/en not_active Abandoned
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- 2006-03-17 KR KR1020077021707A patent/KR20070114187A/ko not_active Ceased
- 2006-03-17 AU AU2006227243A patent/AU2006227243B2/en not_active Ceased
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2007
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2014
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- 2017-11-17 JP JP2017221743A patent/JP2018024712A/ja active Pending
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20040097597A1 (en) * | 2001-07-09 | 2004-05-20 | Zonagen, Inc. | Methods and compositions with trans-clomiphene |
| WO2006019916A1 (en) * | 2004-07-14 | 2006-02-23 | Repros Therapeutics Inc. | Trans-clomiphene for the treatment of benign prostate hypertrophy, prostate cancer, hypogonadism, elevated triglycerides and high cholesterol |
| WO2006084153A2 (en) * | 2005-02-04 | 2006-08-10 | Repros Therapeutics Inc. | Methods and materials with trans-clomiphene for the treatment of male infertility |
Also Published As
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| CN101163467A (zh) | 2008-04-16 |
| US20090215907A1 (en) | 2009-08-27 |
| RU2413508C2 (ru) | 2011-03-10 |
| EP1865938A4 (en) | 2008-09-24 |
| RU2007138867A (ru) | 2009-04-27 |
| ZA200707774B (en) | 2009-09-30 |
| JP5785680B2 (ja) | 2015-09-30 |
| EP1865938A2 (en) | 2007-12-19 |
| JP6270281B2 (ja) | 2018-01-31 |
| US20120309839A1 (en) | 2012-12-06 |
| US8247456B2 (en) | 2012-08-21 |
| CN101163467B (zh) | 2012-07-18 |
| BRPI0609389A2 (pt) | 2010-03-30 |
| US8519004B2 (en) | 2013-08-27 |
| CA2597700A1 (en) | 2006-09-28 |
| PL383444A1 (pl) | 2008-03-17 |
| KR20070114187A (ko) | 2007-11-29 |
| JP2018024712A (ja) | 2018-02-15 |
| NZ560551A (en) | 2010-02-26 |
| MX2007010659A (es) | 2007-11-08 |
| JP2008534503A (ja) | 2008-08-28 |
| WO2006102232A2 (en) | 2006-09-28 |
| EP2392322A2 (en) | 2011-12-07 |
| HK1119070A1 (en) | 2009-02-27 |
| EP2392322A3 (en) | 2012-02-22 |
| AU2006227243A1 (en) | 2006-09-28 |
| WO2006102232A3 (en) | 2007-04-12 |
| CA3071412A1 (en) | 2006-09-28 |
| JP2015044867A (ja) | 2015-03-12 |
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| MK14 | Patent ceased section 143(a) (annual fees not paid) or expired |