AU2005210083B2 - Novel combination of anticholinergic and beta mimetics for the treatment of respiratory diseases - Google Patents
Novel combination of anticholinergic and beta mimetics for the treatment of respiratory diseases Download PDFInfo
- Publication number
- AU2005210083B2 AU2005210083B2 AU2005210083A AU2005210083A AU2005210083B2 AU 2005210083 B2 AU2005210083 B2 AU 2005210083B2 AU 2005210083 A AU2005210083 A AU 2005210083A AU 2005210083 A AU2005210083 A AU 2005210083A AU 2005210083 B2 AU2005210083 B2 AU 2005210083B2
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- AU
- Australia
- Prior art keywords
- use according
- daily dose
- pharmaceutical
- formoterol
- glycopyrrolate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
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Classifications
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- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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- A—HUMAN NECESSITIES
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- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
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| US54195704P | 2004-02-06 | 2004-02-06 | |
| US60/541,957 | 2004-02-06 | ||
| PCT/EP2005/000649 WO2005074900A2 (en) | 2004-02-06 | 2005-01-24 | NOVEL COMBINATION OF ANTICHOLINERGIC AND β MIMETICS FOR THE TREATMENT OF RESPIRATORY DISEASES |
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| AU2005210083A1 AU2005210083A1 (en) | 2005-08-18 |
| AU2005210083B2 true AU2005210083B2 (en) | 2010-03-11 |
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| NO (1) | NO337128B1 (enExample) |
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| SI (1) | SI1718336T1 (enExample) |
| WO (1) | WO2005074900A2 (enExample) |
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| ES2165768B1 (es) | 1999-07-14 | 2003-04-01 | Almirall Prodesfarma Sa | Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen. |
| WO2005074918A1 (en) * | 2004-02-06 | 2005-08-18 | Benzstrasse 1 D-61352 Bad Homburd | The combination of anticholinergics and glucocorticoids for the long-term treatment of asthma and copd |
| GB0410398D0 (en) * | 2004-05-10 | 2004-06-16 | Arakis Ltd | The treatment of respiratory disease |
| ES2257152B1 (es) * | 2004-05-31 | 2007-07-01 | Laboratorios Almirall S.A. | Combinaciones que comprenden agentes antimuscarinicos y agonistas beta-adrenergicos. |
| ES2389231T3 (es) * | 2005-12-21 | 2012-10-24 | Meda Pharma Gmbh & Co. Kg | Combinación de anticolinérgicos, glucocorticoides y agonistas de beta2 para el tratamiento de enfermedades inflamatorias |
| US20080031828A1 (en) * | 2006-08-03 | 2008-02-07 | Boehringer Ingelheim International Gmbh | Method for the Treatment of Dyspnea Comprising Combined Administration of Tiotropium Salts and Salts of Salmeterol |
| EP1944018A1 (en) * | 2007-01-10 | 2008-07-16 | CHIESI FARMACEUTICI S.p.A. | Micronised particles of low-dosage strength active agents for powder formulations for inhalation |
| GB0801876D0 (en) * | 2008-02-01 | 2008-03-12 | Vectura Group Plc | Suspension formulations |
| NZ587561A (en) * | 2008-02-26 | 2012-10-26 | Elevation Pharmaceuticals Inc | Method and system for the treatment of chronic obstructive pulmonary disease with nebulized anticholinergic administrations (an muscarinic antagnoist) |
| US20100055045A1 (en) | 2008-02-26 | 2010-03-04 | William Gerhart | Method and system for the treatment of chronic obstructive pulmonary disease with nebulized anticholinergic administrations |
| EP2100598A1 (en) | 2008-03-13 | 2009-09-16 | Laboratorios Almirall, S.A. | Inhalation composition containing aclidinium for treatment of asthma and chronic obstructive pulmonary disease |
| EP2100599A1 (en) | 2008-03-13 | 2009-09-16 | Laboratorios Almirall, S.A. | Inhalation composition containing aclidinium for treatment of asthma and chronic obstructive pulmonary disease |
| EP2221048A1 (en) | 2009-02-18 | 2010-08-25 | Siegfried Generics International AG | Pharmaceutical composition for inhalation |
| EP3106149B1 (en) * | 2009-05-29 | 2019-11-20 | Pearl Therapeutics, Inc. | Compositions for pulmonary delivery of long-acting muscarinic antagonists and long-acting beta-2 adrenergic receptor agonists and associated methods and systems |
| US8815258B2 (en) | 2009-05-29 | 2014-08-26 | Pearl Therapeutics, Inc. | Compositions, methods and systems for respiratory delivery of two or more active agents |
| US20110132355A1 (en) * | 2009-06-09 | 2011-06-09 | William Gerhart | Treatment of chronic obstructive pulmonary disease with nebulized beta 2-agonist or combined nebulized beta 2-agonist and anticholinergic administration |
| CA2785349C (en) * | 2009-12-23 | 2018-07-03 | Chiesi Farmaceutici S.P.A. | Combination therapy for copd |
| WO2011076842A2 (en) * | 2009-12-23 | 2011-06-30 | Chiesi Farmaceutici S.P.A. | Aerosol formulation for copd |
| BR112012015335B1 (pt) * | 2009-12-23 | 2021-05-18 | Chiesi Farmaceutici S.P.A. | formulação de aerossol para doença pulmonar obstrutiva crõnica |
| RS53391B2 (sr) * | 2009-12-23 | 2023-09-29 | Chiesi Farm Spa | Kombinovana terapija copd-a (hroničnih obstruktivnih bolesti pluća) |
| RU2013142268A (ru) | 2011-02-17 | 2015-03-27 | Сипла Лимитед | Фармацевтическая композиция |
| JO3510B1 (ar) * | 2011-03-04 | 2020-07-05 | Heptares Therapeutics Ltd | استخدام جلايكوبيرولات لعلاج عدم انتظام دقات القلب |
| EP2510928A1 (en) | 2011-04-15 | 2012-10-17 | Almirall, S.A. | Aclidinium for use in improving the quality of sleep in respiratory patients |
| BR112013029507A2 (pt) * | 2011-05-17 | 2019-09-24 | Pearl Therapeutics Inc | método para tratar uma doença ou um distúrbio |
| BR112015022784B1 (pt) | 2013-03-15 | 2023-02-14 | Pearl Therapeutics, Inc | Método de condicionamento de material cristalino micronizado e sistemas de condicionamento |
| DK3089735T3 (en) * | 2013-12-30 | 2018-09-17 | Chiesi Farm Spa | STABLE PRESSURE AEROSOL SOLUTION COMPOSITION OF GLYCOPYRRONIUM BROMIDE AND FORMOTEROL COMBINATION |
| CN105848642A (zh) * | 2013-12-30 | 2016-08-10 | 奇斯药制品公司 | 格隆溴铵和福莫特罗组合的稳定的加压气雾剂溶液组合物 |
| WO2017077488A1 (en) * | 2015-11-04 | 2017-05-11 | Glenmark Pharmaceuticals Limited | An inhalable fixed dose powder composition comprising glycopyrronium and formoterol |
| CA3152578A1 (en) | 2019-12-02 | 2021-06-10 | Enrico Zambelli | Stainles steel can for pressurised metered dose inhalers |
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| US20010027789A1 (en) * | 1999-12-18 | 2001-10-11 | Joachim Goede | Storage system for powdered pharmaceuticals, and inhaler equipped with this system |
| WO2001076575A2 (en) * | 2000-04-07 | 2001-10-18 | Arakis Ltd. | The treatment of respiratory diseases |
| US20020115681A1 (en) * | 1999-05-12 | 2002-08-22 | Karl-Heinz Bozung | Medicament compositions containing anticholinergically-effective compounds and salmeterol |
| WO2002078671A1 (de) * | 2001-03-30 | 2002-10-10 | Jagotec Ag | Medizinische aerosolformulierungen |
| US20020151597A1 (en) * | 2001-04-17 | 2002-10-17 | Dey L.P. | Bronchodilating compositions and methods |
| US6475467B1 (en) * | 1998-08-04 | 2002-11-05 | Jago Research Ag | Medicinal aerosol formulations |
| US6645466B1 (en) * | 1998-11-13 | 2003-11-11 | Jago Research Ag | Dry powder for inhalation |
| US20040002548A1 (en) * | 1999-05-12 | 2004-01-01 | Boehringer Ingelheim Pharma Kg | Medicament compositions containing anticholinergically-effective compounds and betamimetics |
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|---|---|---|---|---|
| WO1998000016A1 (en) * | 1996-07-01 | 1998-01-08 | Sepracor, Inc. | Methods and compositions for treating urinary incontinence using enantiomerically enriched (r,r)-glycopyrrolate |
| EP1369414A1 (de) | 1996-11-11 | 2003-12-10 | Christian R. Noe | Enantiomerenreine Arylcycloalkyl-Hydroxycarbonsäureester, Verfahren zu ihrer Herstellung und ihre Verwendung als Muskarinrezeptor-Modulatoren |
| US6585958B1 (en) | 1998-07-24 | 2003-07-01 | Jago Research Ag | Medicinal aerosol formulations |
| GB0008485D0 (en) * | 2000-04-07 | 2000-05-24 | Glaxo Group Ltd | Pharmaceutical compositions |
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2005
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- 2005-01-24 PL PL05701139T patent/PL1718336T3/pl unknown
- 2005-01-24 JP JP2006551761A patent/JP5524442B2/ja not_active Expired - Fee Related
- 2005-01-24 SI SI200530323T patent/SI1718336T1/sl unknown
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- 2005-01-24 WO PCT/EP2005/000649 patent/WO2005074900A2/en not_active Ceased
- 2005-01-24 CN CNA2005800019327A patent/CN1905902A/zh active Pending
- 2005-01-24 HR HR20080439T patent/HRP20080439T3/xx unknown
- 2005-01-24 PT PT05701139T patent/PT1718336E/pt unknown
- 2005-01-24 RU RU2006132036/15A patent/RU2438660C2/ru not_active Application Discontinuation
- 2005-01-24 CA CA2550841A patent/CA2550841C/en not_active Expired - Fee Related
- 2005-01-24 AT AT05701139T patent/ATE399027T1/de active
- 2005-01-24 DK DK05701139T patent/DK1718336T3/da active
- 2005-01-24 AU AU2005210083A patent/AU2005210083B2/en not_active Ceased
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- 2005-01-24 ES ES05701139T patent/ES2309705T3/es not_active Expired - Lifetime
- 2005-02-07 US US11/051,469 patent/US20050175549A1/en not_active Abandoned
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2006
- 2006-07-11 US US11/483,693 patent/US20060252815A1/en not_active Abandoned
- 2006-08-31 NO NO20063882A patent/NO337128B1/no not_active IP Right Cessation
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2007
- 2007-07-30 US US11/882,109 patent/US7985766B2/en active Active
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2008
- 2008-09-10 CY CY20081100967T patent/CY1108326T1/el unknown
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| US6475467B1 (en) * | 1998-08-04 | 2002-11-05 | Jago Research Ag | Medicinal aerosol formulations |
| US6645466B1 (en) * | 1998-11-13 | 2003-11-11 | Jago Research Ag | Dry powder for inhalation |
| US20020115681A1 (en) * | 1999-05-12 | 2002-08-22 | Karl-Heinz Bozung | Medicament compositions containing anticholinergically-effective compounds and salmeterol |
| US20040002548A1 (en) * | 1999-05-12 | 2004-01-01 | Boehringer Ingelheim Pharma Kg | Medicament compositions containing anticholinergically-effective compounds and betamimetics |
| US20010027789A1 (en) * | 1999-12-18 | 2001-10-11 | Joachim Goede | Storage system for powdered pharmaceuticals, and inhaler equipped with this system |
| WO2001076575A2 (en) * | 2000-04-07 | 2001-10-18 | Arakis Ltd. | The treatment of respiratory diseases |
| WO2002078671A1 (de) * | 2001-03-30 | 2002-10-10 | Jagotec Ag | Medizinische aerosolformulierungen |
| US20020151597A1 (en) * | 2001-04-17 | 2002-10-17 | Dey L.P. | Bronchodilating compositions and methods |
Also Published As
| Publication number | Publication date |
|---|---|
| RU2006132036A (ru) | 2008-03-20 |
| US7985766B2 (en) | 2011-07-26 |
| SI1718336T1 (sl) | 2008-10-31 |
| PL1718336T3 (pl) | 2008-11-28 |
| EP1718336B1 (en) | 2008-06-25 |
| WO2005074900A3 (en) | 2006-04-06 |
| AU2005210083A1 (en) | 2005-08-18 |
| JP2007520506A (ja) | 2007-07-26 |
| CN1905902A (zh) | 2007-01-31 |
| NO337128B1 (no) | 2016-01-25 |
| DK1718336T3 (da) | 2008-10-20 |
| CA2550841C (en) | 2012-10-02 |
| NO20063882L (no) | 2006-10-26 |
| NZ548302A (en) | 2010-04-30 |
| PT1718336E (pt) | 2008-08-28 |
| CY1108326T1 (el) | 2014-02-12 |
| RU2438660C2 (ru) | 2012-01-10 |
| ES2309705T3 (es) | 2008-12-16 |
| HRP20080439T3 (hr) | 2008-10-31 |
| US20070270481A1 (en) | 2007-11-22 |
| ATE399027T1 (de) | 2008-07-15 |
| WO2005074900A2 (en) | 2005-08-18 |
| DE602005007708D1 (de) | 2008-08-07 |
| CA2550841A1 (en) | 2005-08-18 |
| EP1718336A2 (en) | 2006-11-08 |
| US20060252815A1 (en) | 2006-11-09 |
| JP5524442B2 (ja) | 2014-06-18 |
| US20050175549A1 (en) | 2005-08-11 |
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